ARTICLE;
CARBON NUCLEAR MAGNETIC RESONANCE;
DRUG STRUCTURE;
DRUG SYNTHESIS;
PROTON NUCLEAR MAGNETIC RESONANCE;
STEROIDOGENESIS;
STRUCTURE ACTIVITY RELATION;
CHEMICAL STRUCTURE;
CHEMISTRY;
CONFORMATION;
NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY;
SYNTHESIS;
MAGNETIC RESONANCE SPECTROSCOPY;
MOLECULAR CONFORMATION;
MOLECULAR STRUCTURE;
NITRILES;
STEROIDS;
New steroids with antiprogestational and antiglucocorticoid activities
Neef G., Beier S., Elger W., Henderson D., and Wiechert R. New steroids with antiprogestational and antiglucocorticoid activities. Steroids 44 (1984) 349-372
The synthesis of 11β -alkyl-19-norsteroids: a novel class of potent steroid hormones. The synthesis of 11β -methyl and 11β -ethylestradiol
Baran J.S., Langford D.D., Laos I., and Liang C.D. The synthesis of 11β -alkyl-19-norsteroids: a novel class of potent steroid hormones. The synthesis of 11β -methyl and 11β -ethylestradiol. Tetrahedron 33 (1977) 609-616
Dialkylation of 2,3-butanedione diketal with 1,8-bis(trimethylsilyl)-2,6-octadiene (BISTRO). Application to the synthesis of estrone derivatives
Pellissier H., and Santelli M. Dialkylation of 2,3-butanedione diketal with 1,8-bis(trimethylsilyl)-2,6-octadiene (BISTRO). Application to the synthesis of estrone derivatives. Tetrahedron 52 (1996) 9093-9100
Synthesis of (+/-)-B(9a)-homo-C-nor-3-methoxy-12-oxa-17-vinylestra-1,3,5(10)-trienes
Wilmouth S., Pellissier H., and Santelli M. Synthesis of (+/-)-B(9a)-homo-C-nor-3-methoxy-12-oxa-17-vinylestra-1,3,5(10)-trienes. Tetrahedron 54 (1998) 13805-13812
Efficient synthesis of new steroids possessing an aromatic A-ring with a 2-hydroxy or a 2-fluoro substituent
Maurin P., Ibrahim-Ouali M., and Santelli M. Efficient synthesis of new steroids possessing an aromatic A-ring with a 2-hydroxy or a 2-fluoro substituent. Eur. J. Org. Chem. (2002) 151-156
A very short synthesis of steroids from 1,3-butadiene and benzocyclobutenes
Michellys P.-Y., Maurin M., Toupet L., Pellissier H., and Santelli M. A very short synthesis of steroids from 1,3-butadiene and benzocyclobutenes. J. Org. Chem. 66 (2001) 115-122
Convenient general synthetic method for 1,4- and 1,5-diketones by palladium catalyzed oxidation of α-allyl and α-3-butenyl ketones
Tsuji J., Shimizu I., and Yamamoto K. Convenient general synthetic method for 1,4- and 1,5-diketones by palladium catalyzed oxidation of α-allyl and α-3-butenyl ketones. Tetrahedron Lett. 34 (1976) 2975-2976
Regiochemistry of Wacker-type oxidation of vinyl group in the presence of neighboring oxygen functions
Michellys P.-Y., Pellissier H., and Santelli M. Regiochemistry of Wacker-type oxidation of vinyl group in the presence of neighboring oxygen functions. Tetrahedron 53 (1997) 7577-7586
Stereochemistry of transmetalation in the palladium-catalyzed coupling of acid-chlorides and organotin
Labadie J.W., and Stille J.K. Stereochemistry of transmetalation in the palladium-catalyzed coupling of acid-chlorides and organotin. J. Am. Chem. Soc. 105 (1983) 669-670
Mechanisms of the palladium-catalyzed couplings of acid-chlorides with organotin reagent
Labadie J.W., and Stille J.K. Mechanisms of the palladium-catalyzed couplings of acid-chlorides with organotin reagent. J. Am. Chem. Soc. 105 (1983) 6129-6137
Stereoselective synthesis of (+)-testosterone via intramolecular 1,3-dipolar cycloaddition of nitrile oxide
Ihara M., Tokunaga Y., and Fukumoto K. Stereoselective synthesis of (+)-testosterone via intramolecular 1,3-dipolar cycloaddition of nitrile oxide. Tetrahedron 47 (1991) 6635-6648
A novel synthetic approach to steroids via intramolecular 1,3-dipolar cycloaddition-a highly stereocontrolled synthesis of testosterone
Ihara M., Tokunaga Y., Tainguchi N., and Fukumoto K. A novel synthetic approach to steroids via intramolecular 1,3-dipolar cycloaddition-a highly stereocontrolled synthesis of testosterone. J. Org. Chem. 55 (1990) 4497-4498
Saline hydrides and superbases in organic reactions. IV: rapid stereospecific methylation of alcohols and glycols with sodium hydride/methyl iodide
Brown C.A., and Barton D. Saline hydrides and superbases in organic reactions. IV: rapid stereospecific methylation of alcohols and glycols with sodium hydride/methyl iodide. Synthesis 6 (1974) 434-436
Acyclic stereoselection. 40: Steric effects, as well as sigma-star-orbital energies, are important in diastereoface differentiation in additions to chiral aldehydes
Lodge E.P., and Heathcock C.H. Acyclic stereoselection. 40: Steric effects, as well as sigma-star-orbital energies, are important in diastereoface differentiation in additions to chiral aldehydes. J. Am. Chem. Soc. 109 (1987) 3353-3361
[[(4,5-Dihydro-2-oxazolyl)phenoxy]alkyl]isoxazoles - Inhibitors of picornavirus uncoating
Diana G.D., Mc Kinlay M.A., Otto M.J., Akullian V., and Oglesby R.C. [[(4,5-Dihydro-2-oxazolyl)phenoxy]alkyl]isoxazoles - Inhibitors of picornavirus uncoating. J. Med. Chem. 28 (1985) 1906-1910
Comfa analysis of the interactions of antipicornavirus compounds in the binding pocket of human rhinovirus-14
Diana G.D., Kowalczyk P., Teasurywala A.M., and Oglesby R.C. Comfa analysis of the interactions of antipicornavirus compounds in the binding pocket of human rhinovirus-14. J. Med. Chem. 35 (1992) 1002-1008
Synthetic utility of the palladium-catalyzed coupling reaction of acid-chlorides with organotins
Labadie J.W., Tueting D., and Stille J.K. Synthetic utility of the palladium-catalyzed coupling reaction of acid-chlorides with organotins. J. Org. Chem. 48 (1983) 4634-4642
Mercuration demercuration of aliphatic isocyanates-a new mild route to primary amines
Malanga C., Urso A., and Lardicci L. Mercuration demercuration of aliphatic isocyanates-a new mild route to primary amines. Tetrahedron Lett. 36 (1995) 8859-8860
