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0029046233
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Synthesis of 1,2,4-oxadiazole-, 1,3,4-oxadiazole-, and 1,2,4-triazole-derived dipeptidomimetics
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0032492712
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Pyrazoles, 1,2,4-triazoles, and tetrazoles as surrogates for cis-amide bonds in boronate ester thrombin inhibitors
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(b) Duncia, J. V.; Santella III, J. B.; Higley, C. A.; VanAtten, M. K.; Weber, P. C.; Alexander, R. S.; Kettner, C. A.; Pruitt, J. R.; Liauw, A. Y.; Quan, M. L.; Knabb, R. M.; Wexler, R. R. Pyrazoles, 1,2,4-triazoles, and tetrazoles as surrogates for cis-amide bonds in boronate ester thrombin inhibitors. Bioorg. Med. Chem. Lett. 1998, 8, 775-780;
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0026776275
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Synthesis and muscarinic activities of quinuclidin-3-yltriazole and -tetrazole derivatives
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(d) Wadswoith, H. J.; Jenkins, S. M.; Orlek, B. S.; Cassidy, F.; Clark, M. S. G.; Brown, F.; Riley, G. J.; Graves, D.; Hawlins, J.; Naylor, C. B. Synthesis and muscarinic activities of quinuclidin-3-yltriazole and -tetrazole derivatives. J. Med. Chem. 1992, 35, 1280-1290;
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Substituent variation in azabicyclic triazole- And tetrazole-based muscarinic receptor ligands
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(e) Jenkins, S. M.; Wadsworth, H. J.; Bromidge, S.; Orlek, B. S.; Wyman, P. A.; Riley, G. J.; Hawkins, J. Substituent variation in azabicyclic triazole- and tetrazole-based muscarinic receptor ligands. J. Med. Chem. 1992, 35, 2392-2406.
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Efficient and regiospecific one-pot synthesis of substituted 1,2,4-triazoles
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Synthèse et activité analgésique dans la série des triazoles-1,2,4
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Clemence, F.; Joliveau-Maushart, C.; Meier, J.; Cerede, J.; Delevallée, F.; Benzoni, J.; Deraedt, R. Synthèse et activité analgésique dans la série des triazoles-1,2,4. Eur. J. Med. Chem. 1985, 20, 257-266.
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Studies of substituted N-benzoyl-2-pyridinecarboxamides: Reactions with acyl chlorides and other electrophiles
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Novel pyrimidine rearrangement reaction: A new synthesis of 4-formylimidazoles
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A convenient synthetic approach to 1,5-diiodonaphthalene derivatives
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Lawson, E. C.; Maryanoff, B. E.; Hoekstra, W. J. A convenient synthetic approach to 1,5-diiodonaphthalene derivatives. Tetrahedron Lett. 2000, 41, 4533-4536.
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Discovery of 4,5-diphenyl-1,2,4-triazole derivatives as a novel class of selective antagonists for the human VIA receptor
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Kakefuda, A.; Suzuki, T.; Tobe, T.; Tahara, A.; Sakamoto, S.; Tsukamoto, S. Discovery of 4,5-diphenyl-1,2,4-triazole derivatives as a novel class of selective antagonists for the human VIA receptor. Bioorg. Med. Chem. Lett. 2002, 10, 1905-1912.
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A mild method for the formation and in situ reaction of imidoyl chlorides: Conversion of pyridine 1-oxides to 2-aminopyridine amides
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The synthesis of spirocyclic [1,2,4]triazolo[4,3-a]quinolines as potential ligands for the benzodiazepine receptor
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Reiter, L. A.; Berg, G. E. The synthesis of spirocyclic [1,2,4]triazolo[4,3-a]quinolines as potential ligands for the benzodiazepine receptor. Heterocycles 1992, 34, 771-780.
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Efficient monohydroxyarylation (or alkylation) and symmetrical bis-hydroxyarylation (or alkylation) of 2,5-dimethyl-1,3,4-thiadiazole
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Cousin, P.; Anselme, G.; Courtois, G.; Mesnard, D. Efficient monohydroxyarylation (or alkylation) and symmetrical bis-hydroxyarylation (or alkylation) of 2,5-dimethyl-1,3,4-thiadiazole. Synth. Commun. 1999, 29, 145-156.
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A new protocol for the synthesis of N(1)-unsubstituted 2-substituted 2-imidazolines
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Jones, C. F. R.; Dimopoulos, P. A new protocol for the synthesis of N(1)-unsubstituted 2-substituted 2-imidazolines. Tetrahedron 2000, 56, 2061-2074.
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An efficient oxidation of acid hydrazides to N,N′-diacylhydrazines using copper(II) acetate in solvent-free conditions under microwave irradiation
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For an example of oxidation of hydrazides to deacyl hydrazides, see Mogilaiah, K.; Prashanthi, M.; Rhandeer Reddy, G. An efficient oxidation of acid hydrazides to N,N′-diacylhydrazines using copper(II) acetate in solvent-free conditions under microwave irradiation. Synth. Commun. 2003, 33, 3741-3745.
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