Octapeptide analogs of somatostatin containing α,α-dialkylated amino acids with potent anticancer activity

International Journal of Peptide Research and Therapeutics

Volumn 12, Issue 2, 2006, Pages 179-185

  Prasad, Sudhanand ^a   Mathur, Archna ^a   Sharma, Rajan ^a   Gupta, Neena ^a   Ahuja, Rinku ^a   Jaggi, Manu ^a   Singh, Anu T ^a   Mukherjee, Rama ^a  

^a DABUR RESEARCH FOUNDATION   (India)

Author keywords

, dialkylated amino acids; Anticancer peptides; Somatostatin

Indexed keywords

2 AMINO 2 METHYLPROPIONIC ACID; AMINO ACID DERIVATIVE; CYCLOLEUCINE; CYSTEINE; DISULFIDE; OCTAPEPTIDE; PEPTIDE DERIVATIVE; SOMATOSTATIN DERIVATIVE;

ANTINEOPLASTIC ACTIVITY; ARTICLE; CANCER INHIBITION; COLON TUMOR; CONFORMATIONAL TRANSITION; DISULFIDE BOND; DRUG DESIGN; DRUG POTENCY; DRUG SCREENING; DRUG SYNTHESIS; IN VIVO STUDY; MOUSE; NONHUMAN; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; NUDE MOUSE; PEPTIDE SYNTHESIS; PROTEIN CONFORMATION; PROTEIN STRUCTURE; STRUCTURE ANALYSIS; TUMOR REGRESSION; TUMOR XENOGRAFT;

MUS MUSCULUS;

EID: 33745059934     PISSN: 15733149     EISSN: 15733904     Source Type: Journal    
DOI: 10.1007/s10989-005-9005-0     Document Type: Article

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