Development of pharmacophoric models on 5,6-diarylimidazo[2.1-b]thiazole for selective inhibition of cyclooxygenase-2 enzyme

Indian Journal of Pharmaceutical Sciences

Volumn 66, Issue 2, 2004, Pages 193-201

  Sharma, R ^a   Prathipati, P ^b   Chaturvedi, S C ^c   Saxena, A K ^b  

^a DEVI AHILYA UNIVERSITY   (India)

^b CENTRAL DRUG RESEARCH INSTITUTE   (India)

^c SHRI G S INSTITUTE OF TECHNOLOGY AND SCIENCE   (India)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 33744820652     PISSN: 0250474X     EISSN: 19983743     Source Type: Journal    
DOI: None     Document Type: Article

References (24)

1. Vane, J.R., Nature, 231, 1971, 232.
2. Lombardino, J.G., In; Nonsteroidal Anti-inflammatory Drugs: Wiley-Interscience / John Wiley & Sons, New York, 1985, 255.
3. Fu, J.Y., Masferrer, J.L., Seibert, K., Raz, A. and Needleman P., J. Biol. Chem., 265, 1990, 16737.
4. Seibert, K., Zhang, Y., Leahy, K., Hauser, S., Masferrer, J. and Isakson, P., Adv. Exp. Med. Biol., 400A, 1997, 167.
5. Kujubu, D.A., Fletcher, B.S., Varnum, B.C., Lim, R.W. and Herschman, H.R., J. Biol. Chem., 266, 1991, 12866.
6. Lee, S.H., Soyoola, E., Chanmugan, P., Hart, S., Sun, W., Zhong, S., Liou, D., Simmons, D. and Hwang, D., J. Biol. Chem., 267, 1992, 25934.
7. O'sullivan, M.G., Huggins, E.M. Jr. and Mc Call, C.E., Biochem. Biophys. Res. Commun, 191, 1993, 1294.
8. Dannhardt, G. and Kiefer, W., Eur. J. Med. Chem., 36, 2001, 109.
9. Reitz, D.B. and Seibert, K., Ann. Rep. Med. Chem., 30, 1995, 179.
10. Pairet, M., Churchill, W., Roman, R.J., Haber, S.B., Kerr, J.S., Scmidt, W.K., Smith, C., Hewes W.E. and Ackerman, N.R., J. Pharmacol. Exp. Ther., 254, 1990, 180.
11. Desmond, R., Dolling, U., Marcune, B., Tillyer, R. and Tschaen D., World Patent No. WO96/08482, 1996, Through Chem. Abstr., 1996, 125, 86474.
12. Gans, K.R., Galbraith, W., Roman, R.J., Haber, S.B., Kerr, J., Scmidt, S., Smith C., Hewas, E. and Ackerman N.R., J. Pharmacol. Exp. Ther., 1990, 254, 180.
13. Therien, M., Brideau, C., Chan, C.C., Cromlish, W.A., Gauthier, J.Y., Gordon, R., Greig , G., Kargman, S., Lau, C.K., Leblanc, Y., Li, C-S., O'Neill, G.P., Riendeau, D., Roy, P., Wang , Z., Xu, L. and Prasit, P., Bioorg. Med. Chem. Letters, 1997, 7, 47.
14. Apex-3D version 1.4 user guide, Biosym MSI, San Diego, Sept. 1993.
15. Insight II version 2.3.0, Biosym MSI, San Diego, Sept. 1993.
16. Discover version 3.1 user guide, Biosym MSI, San Diego, Sept. 1993.
17. Dabur-osguthorpe, P., Roberts, V.A., Ostguthorpe, D.J., Wolf, J., Genset, M. and Hagler, A.T., Proteins Struct. Func. Genet., 1988, 4, 31.
18. Powell, M.J.D. Math. Program., 197, 241.
19. Stewart, J.J.P., QCPF Bull., 1990, 455.
20. Ghose, A.K. and Crippen, G.M., J. Chem. Inf. Comput Sci., 1987, 27, 21.
21. Viswanadhan, V.N., Ghose, A.K., Revankar, G.R. and Robins, R.K., J. Chem. Inf. Comput. Sci., 1989, 29, 103.
22. Golender, V.E. and Vorpagel, E.R., In; Kubinyi, H., Eds., 3D QSAR in Drug Design Theory, Methods and Application, Escom, Leiden, 1993, 137.
23. Golennder, V.E. and Rozenblit, A.B., In; Logical and Combinatorial Algorithms Drug Design, Research Studies Press, Letchworth, 1983, 1.
24. Pandya, T., Pandey, S.K., Tiwari, M., Chaturvedi, S.C. and Saxena, A.K., Bioorg. Med. Chem., 2001, 9, 291.