메뉴 건너뛰기




Volumn 113, Issue 1, 2006, Pages 80-88

The "inverted cup" - A novel in vitro release technique for drugs in lipid formulations

Author keywords

In vitro release; In vitro in vivo correlation; Local anaesthetics; Parenteral depot formulations; Sciatic nerve block

Indexed keywords

BIOMEDICAL ENGINEERING; DRUG PRODUCTS; PHARMACOKINETICS; PHASE TRANSITIONS; VISCOSITY;

EID: 33744529011     PISSN: 01683659     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.jconrel.2006.03.015     Document Type: Article
Times cited : (11)

References (35)
  • 2
    • 0021843298 scopus 로고
    • Clinical pharmacokinetics of the depot antipsychotics
    • Jann M.W., Ereshefsky L., and Saklad S.R. Clinical pharmacokinetics of the depot antipsychotics. Clin. Pharmacokinet. 10 4 (1985) 315-333
    • (1985) Clin. Pharmacokinet. , vol.10 , Issue.4 , pp. 315-333
    • Jann, M.W.1    Ereshefsky, L.2    Saklad, S.R.3
  • 3
    • 0002885683 scopus 로고
    • Note on the subcutaneous absorption of oils by rats and mice, with special reference to the assay of oestrin
    • Deanesly R., and Parkes A.S. Note on the subcutaneous absorption of oils by rats and mice, with special reference to the assay of oestrin. J. Physiol. 78 (1933) 155-160
    • (1933) J. Physiol. , vol.78 , pp. 155-160
    • Deanesly, R.1    Parkes, A.S.2
  • 4
    • 0026578594 scopus 로고
    • A prospective randomized comparison of intramuscular or intravaginal natural progesterone as a luteal phase and early pregnancy supplement
    • Smitz J., Devroey P., Faguer B., Bourgain C., Camus M., and Van Steirteghem A.C. A prospective randomized comparison of intramuscular or intravaginal natural progesterone as a luteal phase and early pregnancy supplement. Hum. Reprod. 7 (1992) 168-175
    • (1992) Hum. Reprod. , vol.7 , pp. 168-175
    • Smitz, J.1    Devroey, P.2    Faguer, B.3    Bourgain, C.4    Camus, M.5    Van Steirteghem, A.C.6
  • 5
    • 0033383771 scopus 로고    scopus 로고
    • Repeated intramuscular injections of testosterone undecanoate for substitution therapy in hypogonadal men
    • Nieschlag E., Buchter D., Von Eckardstein S., Abshagen K., Simoni M., and Behre H.M. Repeated intramuscular injections of testosterone undecanoate for substitution therapy in hypogonadal men. Clin. Endocrinol. 51 (1999) 757-763
    • (1999) Clin. Endocrinol. , vol.51 , pp. 757-763
    • Nieschlag, E.1    Buchter, D.2    Von Eckardstein, S.3    Abshagen, K.4    Simoni, M.5    Behre, H.M.6
  • 6
    • 0031911977 scopus 로고    scopus 로고
    • The pharmacokinetics and bioavailability of dihydroartemisin, arteether, artemether, artesunic acid and artelinic acid in rats
    • Li Q.-G., Peggins O.J., Fleckenstein L.L., Masonic K., Heiffer M.H., and Brewer T.G. The pharmacokinetics and bioavailability of dihydroartemisin, arteether, artemether, artesunic acid and artelinic acid in rats. J. Pharm. Pharmacol. 50 (1998) 173-182
    • (1998) J. Pharm. Pharmacol. , vol.50 , pp. 173-182
    • Li, Q.-G.1    Peggins, O.J.2    Fleckenstein, L.L.3    Masonic, K.4    Heiffer, M.H.5    Brewer, T.G.6
  • 7
    • 0035013368 scopus 로고    scopus 로고
    • Inclusion of lignocaine base into a polar lipid formulation - in vitro release, duration of peripheral nerve block and arterial blood concentrations in the rat
    • Dyhre H., Wallin R., Björkman S., Engström S., and Renck H. Inclusion of lignocaine base into a polar lipid formulation - in vitro release, duration of peripheral nerve block and arterial blood concentrations in the rat. Acta Anaesthesiol. Scand. 45 (2001) 583-589
    • (2001) Acta Anaesthesiol. Scand. , vol.45 , pp. 583-589
    • Dyhre, H.1    Wallin, R.2    Björkman, S.3    Engström, S.4    Renck, H.5
  • 8
    • 0035997889 scopus 로고    scopus 로고
    • In-vitro release of bupivacaine from injectable lipid formulations investigated by a single drop technique-relation to duration of action in-vivo
    • Söderberg L., Dyhre H., Roth B., and Björkman S. In-vitro release of bupivacaine from injectable lipid formulations investigated by a single drop technique-relation to duration of action in-vivo. J. Pharm. Pharmacol. 54 (2002) 747-755
    • (2002) J. Pharm. Pharmacol. , vol.54 , pp. 747-755
    • Söderberg, L.1    Dyhre, H.2    Roth, B.3    Björkman, S.4
  • 9
    • 0037123707 scopus 로고    scopus 로고
    • In vivo release of bupivacaine from subcutaneously administered oily solution. Comparison with in vitro release
    • Larsen D.B., Joergensen S., Olsen N.V., Hansen S.H., and Larsen C. In vivo release of bupivacaine from subcutaneously administered oily solution. Comparison with in vitro release. J. Control. Release 81 (2002) 145-154
    • (2002) J. Control. Release , vol.81 , pp. 145-154
    • Larsen, D.B.1    Joergensen, S.2    Olsen, N.V.3    Hansen, S.H.4    Larsen, C.5
  • 10
    • 33644865613 scopus 로고    scopus 로고
    • Ultralong peripheral nerve block by lidocaine:prilocaine 1:1 mixture in a lipid depot formulation: comparison of in vitro, in vivo and effect kinetics
    • Söderberg L., Dyhre H., Roth B., and Björkman S. Ultralong peripheral nerve block by lidocaine:prilocaine 1:1 mixture in a lipid depot formulation: comparison of in vitro, in vivo and effect kinetics. Anesthesiology 104 (2006) 110-121
    • (2006) Anesthesiology , vol.104 , pp. 110-121
    • Söderberg, L.1    Dyhre, H.2    Roth, B.3    Björkman, S.4
  • 11
    • 0002906786 scopus 로고
    • Drug delivery from cubic and other lipid-water phases
    • Engström S. Drug delivery from cubic and other lipid-water phases. Lipid Technol. 2 (1990) 42-45
    • (1990) Lipid Technol. , vol.2 , pp. 42-45
    • Engström, S.1
  • 12
    • 0026527630 scopus 로고
    • Phase behaviour of the lignocaine-monoolein-water system
    • Engström S., and Engström L. Phase behaviour of the lignocaine-monoolein-water system. Int. J. Pharm. 79 (1992) 113-122
    • (1992) Int. J. Pharm. , vol.79 , pp. 113-122
    • Engström, S.1    Engström, L.2
  • 13
    • 0026457460 scopus 로고
    • A study of polar lipid drug carrier systems undergoing a thermoreversible lamellar-to-cubic phase transition
    • Engström S., Lindahl L., Wallin R., and Engblom J. A study of polar lipid drug carrier systems undergoing a thermoreversible lamellar-to-cubic phase transition. Int. J. Pharm. 86 (1992) 137-145
    • (1992) Int. J. Pharm. , vol.86 , pp. 137-145
    • Engström, S.1    Lindahl, L.2    Wallin, R.3    Engblom, J.4
  • 14
    • 0026641726 scopus 로고
    • Formulation of a drug delivery system based on a mixture of monoglycerides and triglycerides for use in the treatment of periodontal disease
    • Norling T., Lading P., Engström S., Larsson K., Krog N., and Nissen S.S. Formulation of a drug delivery system based on a mixture of monoglycerides and triglycerides for use in the treatment of periodontal disease. J. Clin. Periodontol. 19 (1992) 687-692
    • (1992) J. Clin. Periodontol. , vol.19 , pp. 687-692
    • Norling, T.1    Lading, P.2    Engström, S.3    Larsson, K.4    Krog, N.5    Nissen, S.S.6
  • 15
    • 0028944067 scopus 로고
    • Phase diagram of soybean phosphatidylcholine-diacylglycerol-water studied by x-ray diffraction and 31P- and pulsed field gradient 1H-NMR: evidence for reversed micelles in the cubic phase
    • Oradd G., Lindblom G., Fontell K., and Ljusberg-Wahren H. Phase diagram of soybean phosphatidylcholine-diacylglycerol-water studied by x-ray diffraction and 31P- and pulsed field gradient 1H-NMR: evidence for reversed micelles in the cubic phase. Biophys. J. 68 (1995) 1856-1863
    • (1995) Biophys. J. , vol.68 , pp. 1856-1863
    • Oradd, G.1    Lindblom, G.2    Fontell, K.3    Ljusberg-Wahren, H.4
  • 16
    • 0031774918 scopus 로고    scopus 로고
    • Drug compatibility with the sponge phases formed in monoolein, water, and propylene glycol or poly(ethylene glycol)
    • Alfons K., and Engstrom S. Drug compatibility with the sponge phases formed in monoolein, water, and propylene glycol or poly(ethylene glycol). J. Pharm. Sci. 87 12 (1998) 1527-1530
    • (1998) J. Pharm. Sci. , vol.87 , Issue.12 , pp. 1527-1530
    • Alfons, K.1    Engstrom, S.2
  • 17
    • 0031441595 scopus 로고    scopus 로고
    • Progress in the development of ultra-long-acting local anesthetics
    • Kuzma P.J., Kline M.D., Calkins M.D., and Staats P.S. Progress in the development of ultra-long-acting local anesthetics. Reg. Anesth. 22 (1997) 543-551
    • (1997) Reg. Anesth. , vol.22 , pp. 543-551
    • Kuzma, P.J.1    Kline, M.D.2    Calkins, M.D.3    Staats, P.S.4
  • 18
    • 33644984488 scopus 로고    scopus 로고
    • Methods to assess in vitro drug release from injectable polymeric particulate systems
    • D'Souza S.S., and DeLuca P.P. Methods to assess in vitro drug release from injectable polymeric particulate systems. Pharm. Res. 23 3 (2006) 460-474
    • (2006) Pharm. Res. , vol.23 , Issue.3 , pp. 460-474
    • D'Souza, S.S.1    DeLuca, P.P.2
  • 20
    • 0035858365 scopus 로고    scopus 로고
    • Regulatory perspectives on in vitro (dissolution)/in vivo (bioavailability) correlations
    • Uppoor V.R.S. Regulatory perspectives on in vitro (dissolution)/in vivo (bioavailability) correlations. J. Control. Release 73 (2001) 127-132
    • (2001) J. Control. Release , vol.73 , pp. 127-132
    • Uppoor, V.R.S.1
  • 21
    • 33744521132 scopus 로고    scopus 로고
    • European Pharmacopoeia Ed. 4, supplement 4.8, Council of Europe, EDQM, 2004, p. 189-199, 3245-3250, 3895-3901.
  • 22
    • 33744510926 scopus 로고    scopus 로고
    • USP 28, United States Pharmacopoeial Convention, Inc., Rockville, MD, p. 2412-2414.
  • 23
    • 0027504825 scopus 로고
    • Conventional versus novel conditions for the in vitro dissolution testing of parenteral slow release formulations: application to doxepin parenteral dosage forms
    • Gido C., Langguth P., Kreuter J., Winter G., Woog H., and Mutschler E. Conventional versus novel conditions for the in vitro dissolution testing of parenteral slow release formulations: application to doxepin parenteral dosage forms. Pharmazie 48 (1993) 764-769
    • (1993) Pharmazie , vol.48 , pp. 764-769
    • Gido, C.1    Langguth, P.2    Kreuter, J.3    Winter, G.4    Woog, H.5    Mutschler, E.6
  • 24
    • 0028286485 scopus 로고
    • Predictions of in vivo plasma concentrations from in vitro release kinetics: application to doxepin parenteral (i.m.) suspensions in lipophilic vehicles in dogs
    • Gido C., Langguth P., and Mutschler E. Predictions of in vivo plasma concentrations from in vitro release kinetics: application to doxepin parenteral (i.m.) suspensions in lipophilic vehicles in dogs. Pharm. Res. 11 6 (1994) 800-808
    • (1994) Pharm. Res. , vol.11 , Issue.6 , pp. 800-808
    • Gido, C.1    Langguth, P.2    Mutschler, E.3
  • 25
    • 0030734317 scopus 로고    scopus 로고
    • Rotating dialysis cell as in vitro release method for oily parenteral depot solutions
    • Schultz K., Mollgaard B., Frokjaer S., and Larsen C. Rotating dialysis cell as in vitro release method for oily parenteral depot solutions. Int. J. Pharm. 157 (1997) 163-169
    • (1997) Int. J. Pharm. , vol.157 , pp. 163-169
    • Schultz, K.1    Mollgaard, B.2    Frokjaer, S.3    Larsen, C.4
  • 26
    • 0033867779 scopus 로고    scopus 로고
    • Assessment of rate of drug release from oil vehicle using a rotating dialysis cell
    • Larsen D.H., Fredholt K., and Larsen C. Assessment of rate of drug release from oil vehicle using a rotating dialysis cell. Eur. J. Pharm. Sci. 11 (2000) 223-229
    • (2000) Eur. J. Pharm. Sci. , vol.11 , pp. 223-229
    • Larsen, D.H.1    Fredholt, K.2    Larsen, C.3
  • 27
    • 0033860043 scopus 로고    scopus 로고
    • Modification of in vitro drug release rate from oily parenteral depots using a formulation approach
    • Fredholt K., Larsen D.H., and Larsen C. Modification of in vitro drug release rate from oily parenteral depots using a formulation approach. Eur. J. Pharm. Sci. 11 (2000) 231-237
    • (2000) Eur. J. Pharm. Sci. , vol.11 , pp. 231-237
    • Fredholt, K.1    Larsen, D.H.2    Larsen, C.3
  • 28
    • 0034963991 scopus 로고    scopus 로고
    • Addition of hydrogen bond donating excipients to oil solution: effect on in vitro drug release rate and viscosity
    • Larsen D.B., Fredholt K., and Larsen C. Addition of hydrogen bond donating excipients to oil solution: effect on in vitro drug release rate and viscosity. Eur. J. Pharm. Sci. 13 (2001) 403-410
    • (2001) Eur. J. Pharm. Sci. , vol.13 , pp. 403-410
    • Larsen, D.B.1    Fredholt, K.2    Larsen, C.3
  • 29
    • 0037203654 scopus 로고    scopus 로고
    • Characteristics of drug substances in oily solutions. Drug release rate, partitioning and solubility
    • Larsen D.B., Parshad H., Fredholt K., and Larsen C. Characteristics of drug substances in oily solutions. Drug release rate, partitioning and solubility. Int. J. Pharm. 232 (2002) 107-117
    • (2002) Int. J. Pharm. , vol.232 , pp. 107-117
    • Larsen, D.B.1    Parshad, H.2    Fredholt, K.3    Larsen, C.4
  • 30
    • 0041666519 scopus 로고    scopus 로고
    • Assessment of drug salt release from solutions, suspensions and in situ suspensions using a rotating dialysis cell
    • Parshad H., Frydenvang K., Liljefors T., and Cornett C. Assessment of drug salt release from solutions, suspensions and in situ suspensions using a rotating dialysis cell. Eur. J. Pharm. Sci. 19 (2003) 263-272
    • (2003) Eur. J. Pharm. Sci. , vol.19 , pp. 263-272
    • Parshad, H.1    Frydenvang, K.2    Liljefors, T.3    Cornett, C.4
  • 31
    • 18044371878 scopus 로고    scopus 로고
    • Characterization of the rotating dialysis cell as an in vitro model potentially useful for simulation of the pharmacokinetic fate of intra-articularly administered drugs
    • Pedersen B.T., Ostergaard J., Larsen S.W., and Larsen C. Characterization of the rotating dialysis cell as an in vitro model potentially useful for simulation of the pharmacokinetic fate of intra-articularly administered drugs. Eur. J. Pharm. Sci. 25 (2005) 73-79
    • (2005) Eur. J. Pharm. Sci. , vol.25 , pp. 73-79
    • Pedersen, B.T.1    Ostergaard, J.2    Larsen, S.W.3    Larsen, C.4
  • 32
    • 0342702115 scopus 로고
    • Effect of dosage form on drug absorption a frequent variable in clinical pharmacology
    • Levy G. Effect of dosage form on drug absorption a frequent variable in clinical pharmacology. Arch. Int. Pharmacodyn. Ther. 152 (1964) 59-68
    • (1964) Arch. Int. Pharmacodyn. Ther. , vol.152 , pp. 59-68
    • Levy, G.1
  • 33
    • 0020082978 scopus 로고
    • In vitro-in vivo correlation, a time scaling problem? Basic considerations on in vitro dissolution testing
    • Brockmeier D., and von Hattingberg H.M. In vitro-in vivo correlation, a time scaling problem? Basic considerations on in vitro dissolution testing. Arzneimittelforschung 32 (1982) 248-251
    • (1982) Arzneimittelforschung , vol.32 , pp. 248-251
    • Brockmeier, D.1    von Hattingberg, H.M.2
  • 34
    • 0024114562 scopus 로고
    • A note regarding curve fitting with a sum of exponentials
    • Ronald A., and Veng-Pedersen P. A note regarding curve fitting with a sum of exponentials. Biopharm. Drug Dispos. 9 (1988) 579-586
    • (1988) Biopharm. Drug Dispos. , vol.9 , pp. 579-586
    • Ronald, A.1    Veng-Pedersen, P.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.