Physical stability, centrifugation tests, and entrapment efficiency studies of carnauba wax-decyl oleate nanoparticles used for the dispersion of inorganic sunscreens in aqueous media

European Journal of Pharmaceutics and Biopharmaceutics

Volumn 63, Issue 2, 2006, Pages 115-127

  Villalobos Hernandez J R ^a   Muller Goymann C C ^a  

^a TECHNICAL UNIVERSITY OF BRAUNSCHWEIG   (Germany)

Author keywords

Centrifugation; Entrapment efficiency; Inorganic sunscreens; Nanosuspensions; Physical stability; Transmission electron microscopy

Indexed keywords

BARIUM SULFATE; NANOPARTICLE; OLEIC ACID; PLANT EXTRACT; STRONTIUM; SUNSCREEN; TITANIUM DIOXIDE; UNCLASSIFIED DRUG; WAX;

AQUEOUS SOLUTION; ARTICLE; CARNAUBA; CARNAUBA WAX; CENTRIFUGATION; DISPERSION; DRUG FORMULATION; DRUG STABILITY; ENCAPSULATION; MATHEMATICAL COMPUTING; MEDICINAL PLANT; PARTICLE SIZE; TEMPERATURE; TRANSMISSION ELECTRON MICROSCOPY;

CENTRIFUGATION; DRUG STABILITY; MICROSCOPY, ELECTRON, TRANSMISSION; NANOTECHNOLOGY; OLEIC ACID; PARTICLE SIZE; SUNSCREENING AGENTS; TEMPERATURE; TITANIUM; WATER; WAXES;

EID: 33646833799     PISSN: 09396411     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ejpb.2006.01.005     Document Type: Article

References (37)

1. Müller R.H., Radtke M., and Wissing S. Solid lipid nanoparticles (SLN) and nanostructured lipid carriers (NLC) in cosmetic and dermatological preparations. Adv. Drug Deliv. Rev. 54 (2002) S131-S155
2. 1H NMR study. Int. J. Pharm. 205 (2000) 15-21
3. Mehnert W., and Mäder K. Solid lipid nanoparticles. Production, characterization and applications. Adv. Drug Deliv. Rev. 47 (2001) 165-196
4. Saupe A., Wissing S.A., Lenk A., Schmidt C., and Müller R.H. Solid lipid nanoparticles (SLN) and nanostructured lipid carriers (NLC) - structural investigations on two different carrier systems. Bio-Med. Mat. Eng. 15 (2005) 393-402
5. Müller R.H., Radtke M., and Wissing S.A. Nanostructured lipid matrices for improved microencapsulation of drugs. Int. J. Pharm. 242 (2002) 121-128
6. J. R. Villalobos-Hernández, C. C. Müller-Goymann, Evaluation of a novel nanoparticulate carrier system for inorganic sunscreens based on carnauba wax and decyl oleate, in: Proceedings of the International Meeting on Pharmaceutics, Biopharmaceuticals, and Pharmaceutical Technology, Nuerenberg, March 2004, pp. 487-488.
7. W. Grimm, Basic principles of stability testing, in: W. Grimm, K. Krummen (Eds.), Stability Testing in the EC, Japan and the USA, Wissenschaftliche Verlagsgesellschaft mbH, Stuttgart, Germany, 1984, pp. 189-204.
8. Weiner N. Introduction. In: Liebermann H.A., Rieger M.M., and Banker S. (Eds). Pharmaceutical Dosage Forms: Disperse Systems vol. 1 (1996), Marcel Dekker, New York, NY 1-14
9. P.H. Stahl, Basic principles of stability testing, in: W. Grimm, K. Krummen (Eds.), Stability Testing in the EC, Japan and the USA, Wissenschaftliche Verlagsgesellschaft mbH, Stuttgart, Germany, 1984, pp. 45-65.
10. A.K. Reng, Stabilitätsprüfungen von dispersen Zubereitungen, in: Asche, D. Essig, C. Schmidt (Eds.), Technologie von Salben, Suspensionen und Emulsionen, Wissenschaftliche Verlagsgesellschaft mbH, Stuttgart, Germany, 1984, pp. 189-204.
11. Nash R. Pharmaceutical suspensions. In: Liebermann H.A., Rieger M.M., and Banker S. (Eds). Pharmaceutical Dosage Forms: Disperse Systems vol. 2 (1996), Marcel Dekker, New York, NY 1-46
12. Falkiewicz M.J. Theory of suspensions. In: Liebermann H.A., Rieger M.M., and Banker S. (Eds). Pharmaceutical Dosage Forms: Disperse Systems vol. 1 (1996), Marcel Dekker, New York, NY 32-41
13. W. Grimm, General concept of stability testing, in: W. Grimm, K. Krummen (Eds.), Stability Testing in the EC, Japan and the USA, Wissenschaftliche Verlagsgesellschaft mbH, Stuttgart, Germany, 1984, pp. 191-223.
14. Santoro M.I.R.M., Almança Gonçalves Da Costa D., Oliveira E., Kedor-Hackmann E.R.M., and Singh A.K. The effect of packaging materials on the stability of sunscreen emulsions. Int. J. Pharm. 297 (2005) 197-203
15. Bhargava H.N., Nicolai D.W., and Oza B.J. Topical suspensions. In: Liebermann H.A., Rieger M.M., and Banker S. (Eds). Pharmaceutical Dosage Forms: Disperse Systems vol. 2 (1996), Marcel Dekker, New York, NY 183-242
16. Müller R.H., Mäder K., and Gohla S. Solid lipid nanoparticles for controlled delivery - a review of the state of art. Eur. J. Pharm. Biopharm. 50 (2000) 161-177
17. Westesen K., Bunjes H., and Koch M.H.J. Physicochemical characterization of lipid nanoparticles and evaluation of their drug loading capacity and sustained release potential. J. Control Release 48 (1997) 223-236
18. Müller R.H., Mäder K., and Gohla S. Solid lipid nanoparticles (SLN) for controlled drug delivery - a review of the state of art. Eur. J. Pharm. Biopharm. 50 (2000) 161-167
19. Wissing S.A., Kayser O., and Müller R.H. Solid lipid nanoparticles for parenteral drug delivery. Adv. Drug Deliv. Rev. 56 (2004) 1257-1272
20. Freitas C., and Müller R.H. Correlation between long-term stability of solid lipid nanoparticles (SLN™) and crystallinity of the lipid phase. Eur. J. Pharm. Biopharm. 47 (1999) 125-132
21. Lim S., and Kim C. Formulation parameters determining the physicochemical characteristics of solid lipid nanoparticles loaded with all-trans retinoic acid. Int. J. Pharm. 234 (2002) 135-146
22. Jiménez M.M., Pelletier J., Bobin M.F., and Martini M.C. Influence of encapsulation on the in vitro percutaneous absorption of octyl methoxycinnamate. Int. J. Pharm. 272 (2004) 45-55
23. Marchais H., Benali S., Irache J.M., Tharasse-Bloch C., Lafont O., and Orecchioni A.M. Entrapment efficiency and initial release of phenylbutazone from nanocapsules prepared from different polyesters. Drug Dev. Ind. Pharm. 24 9 (1998) 833-888
24. Tiarks F., Landfester K., and Antonietti M. Encapsulation of carbon black by miniemulsion polymerisation. Macromol. Chem. Phys. 202 (2001) 51-60
25. Jores K., Mehnert W., Drechsler M., Bunjes H., Johann C., and Mäder K. Investigations on the structure of solid lipid nanoparticles by photon correlation spectroscopy, field-flow fractionation and transmission electron microscopy. J. Control Release 95 (2004) 217-227
26. Villalobos-Hernández J.R., and Müller-Goymann C.C. Novel nanoparticulate carrier systems based on carnauba wax an decyl oleate for the dispersion of inorganic sunscreens in aqueous media. Eur. J. Pharm. Biopharm. 60 (2005) 113-122
27. Müller R.H., and Böhm B.H.L. Dispersion techniques for laboratory and industrial scale processing. Wissenschaftliche Verlagsgesellschaft mbH Stuttgart (2001) 16-29
28. Cheng X.Y., Liang J.X., and Li Q.G. Construction of RNA-containing virus-like nanoparticles expression vector with cysteine residues on surface and fluorescent decoration. Yi Chuang Xue Bao 32 (2005) 874-878
29. Müller R.H. Zetapotential und Partikelladung in der Laborpraxis. Wissenschaftliche Verlagsgesellschaft mbH Stuttgart (1996) 52-53
30. Müller R.H., and Schuhmann R. Teilchengrößenmessung in der Laborpraxis. Wissenschaftliche Verlagsgesellschaft mbH Stuttgart (1996) 23-30
31. Talsma H., van Steenbergen M.J., and Crommelin D.J.A. The cryoprotection of liposomes 2. Effect of the particle size on the crytallization behavior and marker retention. Cryobiology 29 (1992) 80-86
32. Souto E.B., Wissing S.A., Barbosa C.M., and Müller R.H. Development of a controlled release formulation based on SLN and NLC for topical clotrimazole delivery. Int. J. Pharm. 278 (2004) 71-77
33. Crowe L.M., Crowe J.H., Rudolph A., Wormersley C., and Appel L. Preservation of freeze-dried liposomes by trehalose. Arch. Biochem. Biophys. Acta 242 (1985) 240-247
34. Crowe L.M., Wormersley C., Crowe J.H., Reid D., Appel L., and Rudolph A. prevention of fusion and leakage in freeze-dried liposomes by carbohydrations. Arch. Biochem. Biophys. Acta 861 (1986) 131-140
35. Lippacher A., Müller R.H., and Mäder K. Liquid and semisolid SLN™ dispersions for topical application: rheological characterization. Eur. J. Pharm. Biopharm. 58 (2004) 561-567
36. de Chasteignier S., Cavé G., Fessi H., Devissaguet J.P., and Puisieux F. Freeze-Drying of itraconazole-loaded nanosphere suspensions: a feasibility study. Drug Dev. Res. 38 (1996) 116-124
37. Müller-Goymann C.C. Physicochemical characterization of colloidal drug delivery systems such as reverse micelles, vesicles, liquid crystals and nanoparticles for topical administration. Eur. J. Pharm. Biopharm. 58 (2004) 343-356