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Volumn 23, Issue 4, 2006, Pages 680-688

Analysis of in vitro skin permeation of 22-oxacalcitriol having a complicated metabolic pathway

Author keywords

22 oxacalcitriol; Diffusion model; Rat skin; Skin metabolism; Skin permeation

Indexed keywords

22 OXACALCITRIOL; DRUG METABOLITE;

EID: 33646411475     PISSN: 07248741     EISSN: 1573904X     Source Type: Journal    
DOI: 10.1007/s11095-006-9781-z     Document Type: Article
Times cited : (11)

References (24)
  • 1
    • 0025084188 scopus 로고
    • Enhanced delivery of zidovudine through rat and human skin via ester prodrugs
    • T. Seki T. Kawaguchi K. Juni 1990 Enhanced delivery of zidovudine through rat and human skin via ester prodrugs Pharm. Res. 7 948 952
    • (1990) Pharm. Res. , vol.7 , pp. 948-952
    • Seki, T.1    Kawaguchi, T.2    Juni, K.3
  • 2
    • 0025336831 scopus 로고
    • Carboxylic ester hydrolase activity in hairless and athymic nude mouse skin
    • M. K. Ghosh A. K. Mitra 1990 Carboxylic ester hydrolase activity in hairless and athymic nude mouse skin Pharm. Res. 7 251 255
    • (1990) Pharm. Res. , vol.7 , pp. 251-255
    • Ghosh, M.K.1    Mitra, A.K.2
  • 3
    • 0028139958 scopus 로고
    • Effects of epidermal/dermal separation methods and ester chain configuration on the bioconversion of a homologous series of methotrexate dialkyl esters in dermal and epidermal homogenates of hairless mouse skin
    • J. J. Fort A. K. Mitra 1994 Effects of epidermal/dermal separation methods and ester chain configuration on the bioconversion of a homologous series of methotrexate dialkyl esters in dermal and epidermal homogenates of hairless mouse skin Int. J. Pharm. 102 241 247
    • (1994) Int. J. Pharm. , vol.102 , pp. 241-247
    • Fort, J.J.1    Mitra, A.K.2
  • 4
    • 0023655003 scopus 로고
    • Cytochrome P-450 dependent metabolism of testosterone in rat skin
    • H. Mukhtar M. Athar D. R. Bickers 1987 Cytochrome P-450 dependent metabolism of testosterone in rat skin Biochem. Biophys. Res. Commun. 145 749 753
    • (1987) Biochem. Biophys. Res. Commun. , vol.145 , pp. 749-753
    • Mukhtar, H.1    Athar, M.2    Bickers, D.R.3
  • 5
    • 0022413127 scopus 로고
    • Distribution and sub-cellular localization of drug metabolizing enzymes in the skin
    • M. J. Finnen M. L. Herdman S. Shuster 1985 Distribution and sub-cellular localization of drug metabolizing enzymes in the skin Br. J. Dermatol. 113 713 721
    • (1985) Br. J. Dermatol. , vol.113 , pp. 713-721
    • Finnen, M.J.1    Herdman, M.L.2    Shuster, S.3
  • 6
    • 0018671731 scopus 로고
    • Physical model evaluation of topical prodrug delivery-simultaneous transport and bioconversion of vidarabine-5′-valerate I: Physical model development
    • C. D. Yu J. L. Fox N. F. H. Ho W. I. Higuchi 1979 Physical model evaluation of topical prodrug delivery-simultaneous transport and bioconversion of vidarabine-5′-valerate I: physical model development J. Pharm. Sci. 68 1341 1346
    • (1979) J. Pharm. Sci. , vol.68 , pp. 1341-1346
    • Yu, C.D.1    Fox, J.L.2    Ho, N.F.H.3    Higuchi, W.I.4
  • 7
    • 0025205114 scopus 로고
    • Quantitaton of simultaneous diffusion and metabolism of β-estradiol in hairless mouse skin: Enzyme distribution and intrinsic diffusion/metabolism parameters
    • P. Liu W. I. Higuchi A.-H. Ghanem T. Kurihara-Bergstrom W. R. Good 1990 Quantitaton of simultaneous diffusion and metabolism of β-estradiol in hairless mouse skin: enzyme distribution and intrinsic diffusion/metabolism parameters Int. J. Pharm. 64 7 25
    • (1990) Int. J. Pharm. , vol.64 , pp. 7-25
    • Liu, P.1    Higuchi, W.I.2    Ghanem, A.-H.3    Kurihara-Bergstrom, T.4    Good, W.R.5
  • 8
    • 0030591404 scopus 로고    scopus 로고
    • Analysis of in vitro skin penetration of acyclovir prodrugs based on a diffusion model with a metabolic process
    • H. Bando M. Sahashi T. Takagi F. Yamashita Y. Takakura M. Hashida 1996 Analysis of in vitro skin penetration of acyclovir prodrugs based on a diffusion model with a metabolic process Int. J. Pharm. 135 91 102
    • (1996) Int. J. Pharm. , vol.135 , pp. 91-102
    • Bando, H.1    Sahashi, M.2    Takagi, T.3    Yamashita, F.4    Takakura, Y.5    Hashida, M.6
  • 9
    • 0028270058 scopus 로고
    • Diffusion and metabolism of prednisolone farnesylate in viable skin of the hairless mouse
    • K. Tojo K. Yamada T. Hikita 1994 Diffusion and metabolism of prednisolone farnesylate in viable skin of the hairless mouse Pharm. Res. 11 393 397
    • (1994) Pharm. Res. , vol.11 , pp. 393-397
    • Tojo, K.1    Yamada, K.2    Hikita, T.3
  • 10
    • 0028826222 scopus 로고
    • Physical model relating diffusional transport and concurrent metabolism of peptides in metabolically active cell sheet
    • I. Steinsträsser R. Sperb H. P. Merkle 1995 Physical model relating diffusional transport and concurrent metabolism of peptides in metabolically active cell sheet J. Pharm. Sci. 84 1332 1341
    • (1995) J. Pharm. Sci. , vol.84 , pp. 1332-1341
    • Steinsträsser, I.1    Sperb, R.2    Merkle, H.P.3
  • 11
    • 0030591413 scopus 로고    scopus 로고
    • Analysis of in vitro rat skin permeation and metabolism of SM-10902, prodrug of synthetic prostacyclin analogue
    • K. Sato T. Mine 1996 Analysis of in vitro rat skin permeation and metabolism of SM-10902, prodrug of synthetic prostacyclin analogue Int. J. Pharm. 135 127 136
    • (1996) Int. J. Pharm. , vol.135 , pp. 127-136
    • Sato, K.1    Mine, T.2
  • 12
    • 0034616620 scopus 로고    scopus 로고
    • Modeling of diffusion and concurrent metabolism in cutaneous tissue
    • P. Boderke K. Schittkowski M. Wolf H. P. Merkle 2000 Modeling of diffusion and concurrent metabolism in cutaneous tissue J. Theor. Biol. 204 393 407
    • (2000) J. Theor. Biol. , vol.204 , pp. 393-407
    • Boderke, P.1    Schittkowski, K.2    Wolf, M.3    Merkle, H.P.4
  • 13
    • 0032883599 scopus 로고    scopus 로고
    • Simultaneous transport and metabolism of ethyl nicotinate in hairless rat skin after its topical application: The effect of enzyme distribution in skin
    • K. Sugibayashi T. Hayashi Y. Morimoto 1999 Simultaneous transport and metabolism of ethyl nicotinate in hairless rat skin after its topical application: the effect of enzyme distribution in skin J. Control. Release 62 201 208
    • (1999) J. Control. Release , vol.62 , pp. 201-208
    • Sugibayashi, K.1    Hayashi, T.2    Morimoto, Y.3
  • 15
    • 0032811171 scopus 로고    scopus 로고
    • Topical application for the treatment of psoriasis vulgaris: A placebo-controlled, double-blind, dose-finding study with active comparator
    • J. N. W. N. Barker R. E. Ashton R. Marks R. I. Harris J. Berth-Jones 1999 Topical application for the treatment of psoriasis vulgaris: a placebo-controlled, double-blind, dose-finding study with active comparator Br. J. Dermatol. 141 274 278
    • (1999) Br. J. Dermatol. , vol.141 , pp. 274-278
    • Barker, J.N.W.N.1    Ashton, R.E.2    Marks, R.3    Harris, R.I.4    Berth-Jones, J.5
  • 18
    • 0022410469 scopus 로고
    • Skin penetration and metabolism of topically applied chemicals in six mammalian species, including man: An in vitro study with benzo[a]pyrene and testosterone
    • J. Kao F. K. Patterson J. Hall 1985 Skin penetration and metabolism of topically applied chemicals in six mammalian species, including man: an in vitro study with benzo[a]pyrene and testosterone Toxicol. Appl. Pharmacol. 81 502 516
    • (1985) Toxicol. Appl. Pharmacol. , vol.81 , pp. 502-516
    • Kao, J.1    Patterson, F.K.2    Hall, J.3
  • 20
    • 0027365445 scopus 로고
    • Metabolism of propranolol during percutaneous absorption in human skin
    • J. I. Ademola C. A. Chow R. C. Wester H. I. Maibach 1993 Metabolism of propranolol during percutaneous absorption in human skin J. Pharm. Sci. 82 767 770
    • (1993) J. Pharm. Sci. , vol.82 , pp. 767-770
    • Ademola, J.I.1    Chow, C.A.2    Wester, R.C.3    Maibach, H.I.4
  • 21
    • 0027469562 scopus 로고
    • An automated in vitro dermal absorption procedure: III. in vivo and in vitro comparison with the insect repellent N,N-diethyl-m-toluamide in mouse, rat, guinea pig, pig, human and tissue-cultured skin
    • R. P. Moody B. Nadeau 1993 An automated in vitro dermal absorption procedure: III. In vivo and in vitro comparison with the insect repellent N,N-diethyl-m-toluamide in mouse, rat, guinea pig, pig, human and tissue-cultured skin Toxicol. In Vitro 7 167 176
    • (1993) Toxicol. in Vitro , vol.7 , pp. 167-176
    • Moody, R.P.1    Nadeau, B.2
  • 23
    • 0037403454 scopus 로고    scopus 로고
    • Toxicokinetics and metabolism of N-[14C]N-methyl-2-pyrrolidone in male Sprague- Dawley rats: In vivo and in vitro percutaneous absorption
    • J. P. Payan I. Boudry D. Beydon J. P. Fabry M. C. Grandclaude E. Ferrari J. C. Andre 2003 Toxicokinetics and metabolism of N-[14C]N-methyl-2-pyrrolidone in male Sprague- Dawley rats: in vivo and in vitro percutaneous absorption Drug Metab. Dispos. 31 659 669
    • (2003) Drug Metab. Dispos. , vol.31 , pp. 659-669
    • Payan, J.P.1    Boudry, I.2    Beydon, D.3    Fabry, J.P.4    Grandclaude, M.C.5    Ferrari, E.6    Andre, J.C.7
  • 24
    • 0023698532 scopus 로고
    • Analysis of drug penetration through skin considering donor concentration decrease
    • M. Hashida H. Okano H. Sezaki 1988 Analysis of drug penetration through skin considering donor concentration decrease J. Pharmacobio-dyn. 11 636 644
    • (1988) J. Pharmacobio-dyn. , vol.11 , pp. 636-644
    • Hashida, M.1    Okano, H.2    Sezaki, H.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.