A collaborative hit-to-lead investigation leveraging medicinal chemistry expertise with high throughput library design, synthesis and purification capabilities

Combinatorial Chemistry and High Throughput Screening

Volumn 9, Issue 2, 2006, Pages 123-130

  Yang, X ^a   Parker, D ^a   Whitehead, L ^a   Ryder, N S ^a   Weidmann, B ^a   Stabile Harris, M ^b   Kizer, D ^b   McKinnon, M ^b   Smellie, A ^b   Powers, D ^b  

^a NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH   (United States)

^b ARQULE INC   (United States)

Author keywords

Antiinfectives; High throughput screening; Hit to lead; Laboratory automation; Library design; Parallel synthesis; Resource management

Indexed keywords

ARTICLE; CHEMISTRY; DRUG PURIFICATION; DRUG SYNTHESIS; HIGH THROUGHPUT SCREENING; MEDICAL RESEARCH; MOLECULAR MODEL; PRIORITY JOURNAL;

CHEMISTRY, PHARMACEUTICAL; COMBINATORIAL CHEMISTRY TECHNIQUES; COMPUTING METHODOLOGIES; COOPERATIVE BEHAVIOR; DRUG DESIGN; SYSTEMS INTEGRATION;

EID: 33645730356     PISSN: 13862073     EISSN: None     Source Type: Journal    
DOI: 10.2174/138620706775541891     Document Type: Article

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