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Volumn 60, Issue 3, 2006, Pages 121-126

Synthesis of aminoacyl thiaolidones as potential antitumour agents

Author keywords

4 Thiazolidone; Antitumour agents; Peptidyl derivatives

Indexed keywords

4 THIAZOLIDINONE DERIVATIVE; AMINOACYLTHIAOLIDONE DERIVATIVE; ANTINEOPLASTIC AGENT; UNCLASSIFIED DRUG;

EID: 33645417997     PISSN: 07533322     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.biopha.2006.01.005     Document Type: Article
Times cited : (8)

References (34)
  • 1
    • 27744594382 scopus 로고    scopus 로고
    • Câncer e agentes antineoplásicos ciclo celular específicos e ciclo celular não específicos que interagem com o DNA: Uma introdu̧ão
    • V.L. Almeida, A. Leitão, L.C.B. Reina, C.A. Montanari, C.L. Donnici, and M.T.P. Lopes Câncer e agentes antineoplásicos ciclo celular específicos e ciclo celular não específicos que interagem com o DNA: Uma introdu̧ão Quim. Nova 28 2005 118 129
    • (2005) Quim. Nova , vol.28 , pp. 118-129
    • Almeida, V.L.1    Leitão, A.2    Reina, L.C.B.3    Montanari, C.A.4    Donnici, C.L.5    Lopes, M.T.P.6
  • 2
    • 0036080202 scopus 로고    scopus 로고
    • Anti-cancer agents
    • S. Eckhardt Anti-cancer agents Curr. Med. Chem. 2 2002 419 439
    • (2002) Curr. Med. Chem. , vol.2 , pp. 419-439
    • Eckhardt, S.1
  • 3
    • 0020607978 scopus 로고
    • Plasmin activated pro-drugs for cancer chemotherapy. Synthesis and biological activity of peptidyl derivatives of doxorubicin
    • P.K. Chakravarty, P.L. Carl, M. Weber, and J. Katzenellenbogen Plasmin activated pro-drugs for cancer chemotherapy. Synthesis and biological activity of peptidyl derivatives of doxorubicin J. Med. Chem. 26 1983 633 638
    • (1983) J. Med. Chem. , vol.26 , pp. 633-638
    • Chakravarty, P.K.1    Carl, P.L.2    Weber, M.3    Katzenellenbogen, J.4
  • 4
    • 0023097983 scopus 로고
    • Selective cytotoxicity of a system L specific amino acid nitrogen mustard
    • D. Haines, R. Fuller, S. Ahmad, D. Vistica, and V. Marquez Selective cytotoxicity of a system L specific amino acid nitrogen mustard J. Med. Chem. 30 1987 542 547
    • (1987) J. Med. Chem. , vol.30 , pp. 542-547
    • Haines, D.1    Fuller, R.2    Ahmad, S.3    Vistica, D.4    Marquez, V.5
  • 5
    • 0035300427 scopus 로고    scopus 로고
    • Extracellularly tumor-activated prodrugs for the selective chemotherapy of cancer: Application to doxirubicin and preliminary in vitro and in vivo studies
    • A. Trouet, A. Passioukov, K. Derpoorten, A.M. Fernandez, J. Abarca-Quinones, and R. Baurain Extracellularly tumor-activated prodrugs for the selective chemotherapy of cancer: application to doxirubicin and preliminary in vitro and in vivo studies Cancer Res. 61 2001 2843 2846
    • (2001) Cancer Res. , vol.61 , pp. 2843-2846
    • Trouet, A.1    Passioukov, A.2    Derpoorten, K.3    Fernandez, A.M.4    Abarca-Quinones, J.5    Baurain, R.6
  • 6
    • 0023912390 scopus 로고
    • Peptide derivatives of primaquine as potential antimalarial agents
    • A. Philip, J. Kepler, B. Johnson, and F. Carrol Peptide derivatives of primaquine as potential antimalarial agents J. Chem. Soc. 31 1988 870 874
    • (1988) J. Chem. Soc. , vol.31 , pp. 870-874
    • Philip, A.1    Kepler, J.2    Johnson, B.3    Carrol, F.4
  • 7
    • 9644273900 scopus 로고    scopus 로고
    • Synthesis, antitumour and antimicrobial activities of new peptidyl derivatives containing the 1,3-benzodioxole system. Eur
    • A.C.L. Leite, K.P. da Silva, I.A. de Souza, J.M. De Araújo, and D.J. Brondani Synthesis, antitumour and antimicrobial activities of new peptidyl derivatives containing the 1,3-benzodioxole system. Eur J. Med. Chem. 39 2004 1059 1065
    • (2004) J. Med. Chem. , vol.39 , pp. 1059-1065
    • Leite, A.C.L.1    Da Silva, K.P.2    De Souza, I.A.3    De Araújo, J.M.4    Brondani, D.J.5
  • 8
    • 0035415493 scopus 로고    scopus 로고
    • Prodrug strategies in cancer therapy
    • W.A. Denny Prodrug strategies in cancer therapy Eur. J. Med. Chem. 36 2001 577 595
    • (2001) Eur. J. Med. Chem. , vol.36 , pp. 577-595
    • Denny, W.A.1
  • 9
    • 0032535999 scopus 로고    scopus 로고
    • Cancer treatment by targets drug delivery to tumor vasculature in a mouse model
    • W. Arap, R. Pasqualini, and E. Ruoslahti Cancer treatment by targets drug delivery to tumor vasculature in a mouse model Science 279 1998 377 380
    • (1998) Science , vol.279 , pp. 377-380
    • Arap, W.1    Pasqualini, R.2    Ruoslahti, E.3
  • 10
    • 0030988859 scopus 로고    scopus 로고
    • 8-(1H-Imidazol-1-yl)-7-nitro-4(5H)-imidazo[1,2-a]quinoxalinone and related compounds: Synthesis and structure-activity relationships for the AMPA-type non-NMDA receptor
    • J. Ohmori, M. Shimizu-Sasamata, M. Okada, and S. Sakamoto 8-(1H-Imidazol-1-yl)-7-nitro-4(5H)-imidazo[1,2-a]quinoxalinone and related compounds: synthesis and structure-activity relationships for the AMPA-type non-NMDA receptor J. Med. Chem. 40 1997 2053 2058
    • (1997) J. Med. Chem. , vol.40 , pp. 2053-2058
    • Ohmori, J.1    Shimizu-Sasamata, M.2    Okada, M.3    Sakamoto, S.4
  • 11
    • 0033520964 scopus 로고    scopus 로고
    • New pyrazole containing bicarboxylic alpha-amino acids: Mimics of the cis amide bond
    • L. Luca, M. Falorni, G. Giacomelli, and A. Porcheddu New pyrazole containing bicarboxylic alpha-amino acids: mimics of the cis amide bond Tetrahedron Lett. 40 1999 8701 8705
    • (1999) Tetrahedron Lett. , vol.40 , pp. 8701-8705
    • Luca, L.1    Falorni, M.2    Giacomelli, G.3    Porcheddu, A.4
  • 12
    • 0033889329 scopus 로고    scopus 로고
    • Synthesis of optically active alpha-amino acids containing pyrazolyl ring as substituent
    • L. Luca, M. Falorni, G. Giacomelli, A. Porcheddu, and A.M. Spanedda Synthesis of optically active alpha-amino acids containing pyrazolyl ring as substituent Synthesis (Mass.) 9 2000 1295 1301
    • (2000) Synthesis (Mass.) , vol.9 , pp. 1295-1301
    • Luca, L.1    Falorni, M.2    Giacomelli, G.3    Porcheddu, A.4    Spanedda, A.M.5
  • 14
    • 0025037115 scopus 로고
    • Synthesis and anti-human-immunodeficiency-virus (HIV-1) activity of 3′-deoxy-3′-(triazol-1-il) thymidines and 2′,3′-dideoxy- 3′-(triazol-1-yl)uridines, and inhibition of reverse transcriptase by their 5′-triphosphates
    • K. Hirota, H. Hosono, Y. Kitade, Y. Maki, and C.K. Chu Synthesis and anti-human-immunodeficiency-virus (HIV-1) activity of 3′-deoxy-3′- (triazol-1-il) thymidines and 2′,3′-dideoxy-3′-(triazol-1-yl) uridines, and inhibition of reverse transcriptase by their 5′- triphosphates Chem. Pharm. Bull. (Tokyo) 38 1990 2597 2602
    • (1990) Chem. Pharm. Bull. (Tokyo) , vol.38 , pp. 2597-2602
    • Hirota, K.1    Hosono, H.2    Kitade, Y.3    Maki, Y.4    Chu, C.K.5
  • 15
    • 37049073557 scopus 로고
    • Trans. Crystal-structure and quantum electronic analyses of pitrazepin, a gamma aminobutyric acid (GABA) receptor antagonist
    • T. Boulanger, D.P. Vercauteren, G. Evrard, and F. Durant Trans. Crystal-structure and quantum electronic analyses of pitrazepin, a gamma aminobutyric acid (GABA) receptor antagonist J. Chem. Soc. Perkin. 2 1989 217 219
    • (1989) J. Chem. Soc. Perkin. , vol.2 , pp. 217-219
    • Boulanger, T.1    Vercauteren, D.P.2    Evrard, G.3    Durant, F.4
  • 16
    • 0026684706 scopus 로고
    • Rationally designed dipeptoid analogs of CCK - acid mimics of the potent and selective nonpeptide CCK-B receptor antagonist CI-988
    • M.J. Drysdale, M.C. Pritchard, and D.C. Horwell Rationally designed dipeptoid analogs of CCK - acid mimics of the potent and selective nonpeptide CCK-B receptor antagonist CI-988 J. Med. Chem. 35 1992 2597 2604
    • (1992) J. Med. Chem. , vol.35 , pp. 2597-2604
    • Drysdale, M.J.1    Pritchard, M.C.2    Horwell, D.C.3
  • 17
    • 0033807919 scopus 로고    scopus 로고
    • Use of 3,5-disubstituted 1,2,4-triazoles for the synthesis of peptidomimetics
    • J. Cesar, and M. Sollner Use of 3,5-disubstituted 1,2,4-triazoles for the synthesis of peptidomimetics Synth. Commun. 30 2000 41 47
    • (2000) Synth. Commun. , vol.30 , pp. 41-47
    • Cesar, J.1    Sollner, M.2
  • 19
    • 0034932539 scopus 로고    scopus 로고
    • N-terminal carboxyl and tetrazole-containing amides as adjuvants to Grb2 SH2 domain ligand binding
    • T.R. Burke, Z.J. Yao, Y. Gao, J.X. Wu, X. Zhu, and J.H. Luo N-terminal carboxyl and tetrazole-containing amides as adjuvants to Grb2 SH2 domain ligand binding Bioorg. Med. Chem. 9 2001 1439 1442
    • (2001) Bioorg. Med. Chem. , vol.9 , pp. 1439-1442
    • Burke, T.R.1    Yao, Z.J.2    Gao, Y.3    Wu, J.X.4    Zhu, X.5    Luo, J.H.6
  • 22
    • 10744233763 scopus 로고    scopus 로고
    • Combinatorial modification of natural products: Synthesis and in vivo analysis of derivatives of thiazole peptide antibiotic GE2270 A: A-ring modifications
    • J. Clough, S. Chen, E.M. Gordon, C. Hackbarth, S. Larn, and J. Trias Combinatorial modification of natural products: synthesis and in vivo analysis of derivatives of thiazole peptide antibiotic GE2270 A: a-ring modifications Bioorganic & Med. Chem. Lett. 13 2003 3409 3414
    • (2003) Bioorganic & Med. Chem. Lett. , vol.13 , pp. 3409-3414
    • Clough, J.1    Chen, S.2    Gordon, E.M.3    Hackbarth, C.4    Larn, S.5    Trias, J.6
  • 23
    • 0036501101 scopus 로고    scopus 로고
    • Synthesis, characterization and biological activity of novel 4-thiazolidinones, 1,3,4-oxadiazoles and some related compounds
    • S.G. Kücukgüzel, E. Oruc, E.S. Rollas, F. Sahin, and A. Özbek Synthesis, characterization and biological activity of novel 4-thiazolidinones, 1,3,4-oxadiazoles and some related compounds Eur. J. Med. Chem. 37 2002 197 203
    • (2002) Eur. J. Med. Chem. , vol.37 , pp. 197-203
    • Kücukgüzel, S.G.1    Oruc, E.2    Rollas, E.S.3    Sahin, F.4    Özbek, A.5
  • 25
    • 0021873308 scopus 로고
    • Synthesis and anti-inflammatory activity of thiazolidinones and imidazolidinones derivated from thiosemicarbazones
    • I.P. Singh, A. Saxena, and K. Shanker Synthesis and anti-inflammatory activity of thiazolidinones and imidazolidinones derivated from thiosemicarbazones Eur. J. Med. Chem. Ther. 20-3 1985 283 287
    • (1985) Eur. J. Med. Chem. Ther. , vol.20 , Issue.3 , pp. 283-287
    • Singh, I.P.1    Saxena, A.2    Shanker, K.3
  • 26
    • 0028074368 scopus 로고
    • Synthesis and anticonvulsivant activity of new 4-thiazolidone and 4-thiazoline derivatives
    • E. Medime, and G. Çapan Synthesis and anticonvulsivant activity of new 4-thiazolidone and 4-thiazoline derivatives Farmaco 49 1994 449 453
    • (1994) Farmaco , vol.49 , pp. 449-453
    • Medime, E.1    Çapan, G.2
  • 27
    • 0034525453 scopus 로고    scopus 로고
    • Synthesis and in vitro antitumour activity evaluation of 1-aryl-1H,3H-thiazolo[3,4-b]quinazolines
    • S. Grasso, N. Micale, A.M. Monforte, P. Monforte, S. Polimeni, and M. Zappalá Synthesis and in vitro antitumour activity evaluation of 1-aryl-1H,3H-thiazolo[3,4-b]quinazolines Eur. J. Med. Chem. 35 2000 1115 1119
    • (2000) Eur. J. Med. Chem. , vol.35 , pp. 1115-1119
    • Grasso, S.1    Micale, N.2    Monforte, A.M.3    Monforte, P.4    Polimeni, S.5    Zappalá, M.6
  • 28
    • 0031800659 scopus 로고    scopus 로고
    • Some reactions of 2-cyanomethylimidazo[4,5-b]pyridine with isothiocyanates. Antituberculotic activity of the obtained compounds
    • L. Bukowski, M. Janowiec, Z. Zwolska-Kwiek, and Z. Andrzejczyk Some reactions of 2-cyanomethylimidazo[4,5-b]pyridine with isothiocyanates. Antituberculotic activity of the obtained compounds Pharmazie 53 1998 373 378
    • (1998) Pharmazie , vol.53 , pp. 373-378
    • Bukowski, L.1    Janowiec, M.2    Zwolska-Kwiek, Z.3    Andrzejczyk, Z.4
  • 32
    • 0035289779 scopus 로고    scopus 로고
    • Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings
    • C. Lipinski, A.F. Lombardo, B.W. Dominy, and P. Feeney Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings Adv. Drug 46 2001 3 26
    • (2001) Adv. Drug , vol.46 , pp. 3-26
    • Lipinski, C.1    Lombardo, A.F.2    Dominy, B.W.3    Feeney, P.4
  • 33
    • 1642575965 scopus 로고    scopus 로고
    • Passage of cell-penetrating peptides across a human epithelial cell layer in vitro
    • M.E. Lindgren, M.M. Hallbrink, A.U. Elmquist, and M. Langel Passage of cell-penetrating peptides across a human epithelial cell layer in vitro Biochem. J. 377 2004 69 76
    • (2004) Biochem. J. , vol.377 , pp. 69-76
    • Lindgren, M.E.1    Hallbrink, M.M.2    Elmquist, A.U.3    Langel, M.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.