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Volumn 14, Issue 9, 2006, Pages 2896-2903

Synthesis and transdermal permeation-enhancing activity of ketone, amide, and alkane analogs of Transkarbam 12

(4) Holas, Tomáš a Vávrová, Kateřina a Klimentová, Jana a Hrabálek, Alexandr a

a Charles University in Prague Faculty of Pharmacy (Czech Republic)

Author keywords

Carbamate; Hydrogen bonding; Percutaneous absorption; Permeation enhancer; Structure activity relationships; Transdermal drug delivery

Indexed keywords

5 (DODECYLOXYCARBONYL)PENTYLAMMONIUM 5 (DODECYLOXYCARBONYL)PENTYLCARBAMATE; 5 (OCTAN 2 YLCARBAMOYL)PENTYLAMMONIUM 5 (OCTAN 2 YLCARBAMOYL)PENTYLCARBAMATE; 5 DECYLCARBAMOYLPENTYLAMMONIUM 5 DECYLCARBAMOYLPENTYLCARBAMATE; 5 DODECYLCARBAMOYLPENTYLAMMONIUM 5 DODECYLCARBAMOYLPENTYLCARBAMATE; 5 HEPTYLCARBAMOYLPENTYLAMMONIUM 5 HEPTACYLCARBAMOYLPENTYLCARBAMATE; 5 HEXYLCARBAMOYLPENTYLAMMONIUM 5 HEXYLCARBAMOYLPENTYLCARBAMATE; 5 NONYLCARBAMOYLPENTYLAMMONIUM 5 NONYLCARBAMOYLPENTYLCARBAMATE; 5 OCTADECYLCARBAMOYLPENTYLAMMONIUM 5 OCTADECYLCARBAMOYLPENTYLCARBAMATE; 5 OCTYLCARBAMOYLPENTYLAMMONIUM 5 OCTYLCARBAMOYLPENTYLCARBAMATE; 6 OXOHEPTADECYLAMMONIUM 6 OXOHEPTADECYLCARBAMATE; CARBAMIC ACID DERIVATIVE; CARBENE; MYRISTIC ACID ISOPROPYL ESTER; OCTADECYLAMMONIUM OCTADECYLCARBAMATE; PENETRATION ENHANCING AGENT; PROPYLENE GLYCOL; THEOPHYLLINE; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; CONTROLLED STUDY; DRUG ACTIVITY; DRUG EFFECT; DRUG PENETRATION; DRUG SYNTHESIS; NONHUMAN;

ADJUVANTS, PHARMACEUTIC; ALKANES; AMIDES; ANIMALS; CARBAMATES; KETONES; MODELS, MOLECULAR; SKIN ABSORPTION; STRUCTURE-ACTIVITY RELATIONSHIP; SWINE; THEOPHYLLINE;

ANIMALIA; SUIDAE;

EID: 33645005238 PISSN: 09680896 EISSN: None Source Type: Journal
DOI: 10.1016/j.bmc.2005.12.006 Document Type: Article

Times cited : (18)

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