Design, synthesis and biological evaluations of novel oxindoles as HIV-1 non-nucleoside reverse transcriptase inhibitors. Part I

Bioorganic and Medicinal Chemistry Letters

Volumn 16, Issue 8, 2006, Pages 2105-2108

  Jiang, Tao ^a   Kuhen, Kelli L ^a   Wolff, Karen ^a   Yin, Hong ^a   Bieza, Kimberly ^a   Caldwell, Jeremy ^a   Bursulaya, Badry ^a   Wu, Tom Yao Hsing ^b   He, Yun ^a  

^a GENOMICS INSTITUTE OF THE NOVARTIS RESEARCH FOUNDATION   (United States)

^b SCRIPPS RESEARCH INSTITUTE   (United States)

Author keywords

AIDS; HIV; Inhibitor; Oxindole; Reverse transcriptase; SAR

Indexed keywords

DELAVIRDINE; EFAVIRENZ; INDOLE DERIVATIVE; NEVIRAPINE; RNA DIRECTED DNA POLYMERASE INHIBITOR;

ARTICLE; CELL ASSAY; DRUG DESIGN; DRUG MONITORING; DRUG POTENCY; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; HUMAN IMMUNODEFICIENCY VIRUS 1; NONHUMAN; STRUCTURE ACTIVITY RELATION; VIRUS REPLICATION;

ANTI-HIV AGENTS; DRUG RESISTANCE, VIRAL; HIV-1; INDOLES; REVERSE TRANSCRIPTASE INHIBITORS; STEREOISOMERISM; STRUCTURE-ACTIVITY RELATIONSHIP; VIRUS REPLICATION;

HUMAN IMMUNODEFICIENCY VIRUS 1;

EID: 33644807569     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2006.01.073     Document Type: Article

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