Synthesis and antibacterial activity of 1β-methyl-2-[5-(1,2- disubstituted ethyl)pyrrolidin-3-ylthio]carbapenem derivatives

Archiv der Pharmazie

Volumn 339, Issue 2, 2006, Pages 67-73

  Ahn, Soo Hyun ^a   Jeon, Heechol ^a   Choi, Joung Hoon ^a   Baek, Daejin ^b   Seo, Seen Hee ^c   Cho, Jung Hyuck ^c   Oh, Chang Hyun ^c  

^a Hanyang University   (South Korea)

^b Hanseo University   (South Korea)

^c Korea Institute of Science and Technology   (South Korea)

Author keywords

1 Methylcarbapenem; Antibacterial activity; Substituent effect

Indexed keywords

1BETA METHYLCARBAPENEM DERIVATIVE; 6 (1 HYDROXYETHYL) 2 [[5 (1 HYDROXY 2 ETHOXYCARBONYL)ETHYL]PYRROLIDIN 3 YL THIOL] 1 METHYLCARBAPEN 2 EM 3 CARBOXYLIC ACID; ANTIINFECTIVE AGENT; IMIPENEM; MEROPENEM; PYRROLIDINE DERIVATIVE; UNCLASSIFIED DRUG; VANCOMYCIN;

ANTIBACTERIAL ACTIVITY; ARTICLE; BACTERIUM CULTURE; BURKHOLDERIA CEPACIA; CONTROLLED STUDY; CORYNEBACTERIUM DIPHTHERIAE; DRUG POTENCY; DRUG SYNTHESIS; ENTEROBACTER CLOACAE; GRAM NEGATIVE BACTERIUM; GRAM POSITIVE BACTERIUM; INFRARED SPECTROSCOPY; MASS SPECTROMETRY; METHICILLIN RESISTANT STAPHYLOCOCCUS AUREUS; MINIMUM INHIBITORY CONCENTRATION; NONHUMAN; PRIORITY JOURNAL; PROTON NUCLEAR MAGNETIC RESONANCE; PSEUDOMONAS AERUGINOSA; STRUCTURE ACTIVITY RELATION;

ANTI-BACTERIAL AGENTS; CARBAPENEMS; MICROBIAL SENSITIVITY TESTS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 33144469140     PISSN: 03656233     EISSN: None     Source Type: Journal    
DOI: 10.1002/ardp.200500139     Document Type: Article

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