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Volumn 339, Issue 2, 2006, Pages 59-66

Synthesis and characterization of thiol containing furoxan derivatives as coligands for the preparation of potential bioreductive radiopharmaceuticals

(10) Cerecetto, Hugo a,d González, Mercedes a Onetto, Silvia a Risso, Mariela a Rey, Ana a,e Giglio, Javier a León, Elsa a León, Alba a Pilatti, Pierina b Fernández, Marcelo c

a UNIVERSIDAD DE LA REPÚBLICA (Uruguay)

b Liceo Juan Lacaze (Uruguay)

c INSTITUTO DE INVESTIGACIONES BIOLÓGICAS CLEMENTE ESTABLE (Uruguay)

d Facultad de Ciencias (Uruguay)

e Facultad de Química (Uruguay)

Author keywords

1,2,5 Oxadiazole N oxide derivatives; Bioreductive99mTc radiopharmaceuticals; Solid tumour imaging

Indexed keywords

1,2,5 OXADIAZOLE N OXIDE DERIVATIVE; 2 NITROIMIDAZOLE DERIVATIVE; 3 (4 MERCAPTOPHENYLMETHYLIDENHYDRAZINOCARBONYLOXYMETHYL) 4 PHENYL 1,2,5 OXADIAZOLE N 2 OXIDE; 3 MERCAPTOMETHYL 4 PHENYL 1,2,5 OXADIAZOLE N 2 OXIDE; DISULFIDE; FUROXAN DERIVATIVE; LIGAND; N,N BIS(2 MERCAPTOETHYL) N',N' DIETHYLETHYLENEDIAMINE; RADIOPHARMACEUTICAL AGENT; TECHNETIUM 99M; THIOL DERIVATIVE; UNCLASSIFIED DRUG; XANTHIC ACID DERIVATIVE;

ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL MODEL; ANIMAL TISSUE; ARTICLE; CARBON NUCLEAR MAGNETIC RESONANCE; CONTROLLED STUDY; DRUG CLEARANCE; DRUG DISTRIBUTION; DRUG EXCRETION; DRUG SYNTHESIS; DRUG UPTAKE; FEMALE; HEPATOBILIARY SYSTEM; HYPOXIA; INFRARED SPECTROSCOPY; MASS SPECTROMETRY; MICROANALYSIS; MOUSE; MOUSE STRAIN; NONHUMAN; PRIORITY JOURNAL; PROTON NUCLEAR MAGNETIC RESONANCE; RADIOCHEMISTRY; REDUCTION; SARCOMA; SOLID TUMOR; THIN LAYER CHROMATOGRAPHY; URINARY EXCRETION;

ANIMALS; FEMALE; LIGANDS; MICE; OXADIAZOLES; RADIOPHARMACEUTICALS; SULFHYDRYL COMPOUNDS; TECHNETIUM; TISSUE DISTRIBUTION;

EID: 33144460671 PISSN: 03656233 EISSN: None Source Type: Journal
DOI: 10.1002/ardp.200500172 Document Type: Article

Times cited : (13)

References (39)

1
- 0000122198
- R. Holm, E. Solomon, Chem. Rev. 1996, 96, 2237-2238.
- (1996) Chem. Rev. , vol.96 , pp. 2237-2238
- Holm, R.¹ Solomon, E.²

2
- 0001381567
- C. Orvig, M. Abrams, Chem. Rev. 1999, 99, 2201-2203.
- (1999) Chem. Rev. , vol.99 , pp. 2201-2203
- Orvig, C.¹ Abrams, M.²

3
- 11444251794
- S. Jurisson, D. Berning, W. Jia, D. Ma, Chem. Rev. 1993, 93. 1137-1156;
- (1993) Chem. Rev. , vol.93 , pp. 1137-1156
- Jurisson, S.¹ Berning, D.² Jia, W.³ Ma, D.⁴

4
- 0012725753
- W. Volkert, T. Hoffman, Chem. Rev. 1999, 99, 2269-2292.
- (1999) Chem. Rev. , vol.99 , pp. 2269-2292
- Volkert, W.¹ Hoffman, T.²

5
- 25144503630
- American Pharmacists Association, Washington DC
- R. Kowalsky, S. Fallen, Radiopharmaceuticals in Nuclear Pharmacy and Nuclear Medicine Second Edition, American Pharmacists Association, Washington DC. 2004, 1 -15;
- (2004) Radiopharmaceuticals in Nuclear Pharmacy and Nuclear Medicine Second Edition , pp. 1-15
- Kowalsky, R.¹ Fallen, S.²

6
- 0027218815
- M. J. Abrams, B. A. Murrer, Science 1993, 261, 725-730.
- (1993) Science , vol.261 , pp. 725-730
- Abrams, M.J.¹ Murrer, B.A.²

7
- 0000167554
- B. Johannsen, H. Spies, Transitions Met. Chem. 1997, 22, 318-320.
- (1997) Transitions Met. Chem. , vol.22 , pp. 318-320
- Johannsen, B.¹ Spies, H.²

8
- 0001294083
- S. Jurisson, J. Lydon, Chem. Rev. 1999, 99, 2205-2218.
- (1999) Chem. Rev. , vol.99 , pp. 2205-2218
- Jurisson, S.¹ Lydon, J.²

9
- 0032342440
- J. Dilworth, S. Parrot, Chem. Soc. Rev. 1998, 27, 43-55.
- (1998) Chem. Soc. Rev. , vol.27 , pp. 43-55
- Dilworth, J.¹ Parrot, S.²

10
- 0008883289
- S. Liu, D. Eduards, Chem. Rev. 1999, 99, 2235-2268.
- (1999) Chem. Rev. , vol.99 , pp. 2235-2268
- Liu, S.¹ Eduards, D.²

11
- 0031797593
- R. Yyer, E. Engelhardt, C. Stobbe, R. Schneider, J. Chapman, Int. J. Radiation Oncology Biol. Phys. 1998, 42, 741-745.
- (1998) Int. J. Radiation Oncology Biol. Phys. , vol.42 , pp. 741-745
- Yyer, R.¹ Engelhardt, E.² Stobbe, C.³ Schneider, R.⁴ Chapman, J.⁵

12
- 0028167554
- K. E. Linder, Y. W. Chan, J. E. Cyr, M. F. Malley, D. P. Nowotnik, A. D. Nunn, J. Med. Chem. 1994, 37, 9-17;
- (1994) J. Med. Chem. , vol.37 , pp. 9-17
- Linder, K.E.¹ Chan, Y.W.² Cyr, J.E.³ Malley, M.F.⁴ Nowotnik, D.P.⁵ Nunn, A.D.⁶

13
- 0031981258
- J. Chapman, E. Engelhardt, C. Stobbe, R. Schneider, G. Hanks, Radiotherapy and Oncology 1998, 46, 229-237;
- (1998) Radiotherapy and Oncology , vol.46 , pp. 229-237
- Chapman, J.¹ Engelhardt, E.² Stobbe, C.³ Schneider, R.⁴ Hanks, G.⁵

14
- 0033959159
- T. Melo, J. Duncan, J. R. Ballinger, A. M. Rauth, J. Nucl. Med. 2000, 41, 169-176;
- (2000) J. Nucl. Med. , vol.41 , pp. 169-176
- Melo, T.¹ Duncan, J.² Ballinger, J.R.³ Rauth, A.M.⁴

15
- 1642452629
- T. Chu, S. Hu, B. Wei, Y. Wang, X. Liu, X. Wang, Bioorg. Med. Chem. Lett. 2004, 14, 747-749.
- (2004) Bioorg. Med. Chem. Lett. , vol.14 , pp. 747-749
- Chu, T.¹ Hu, S.² Wei, B.³ Wang, Y.⁴ Liu, X.⁵ Wang, X.⁶

16
- 0035468733
- H. Cerecetto, M. González, Minirev. Med. Chem. 2001, 1, 219-231.
- (2001) Minirev. Med. Chem. , vol.1 , pp. 219-231
- Cerecetto, H.¹ González, M.²

17
- 0035042457
- H. Cerecetto, M. González, S. Onetto, M. Risso, P. Saenz, G. Seoane, A. M. Bruno, J. Alarcón, C. Olea-Azar, A. López de Ceráin, O. Ezpeleta, A. Monge, Med. Chem. Res. 2001, 10, 328-337;
- (2001) Med. Chem. Res. , vol.10 , pp. 328-337
- Cerecetto, H.¹ González, M.² Onetto, S.³ Risso, M.⁴ Saenz, P.⁵ Seoane, G.⁶ Bruno, A.M.⁷ Alarcón, J.⁸ Olea-Azar, C.⁹ López De Ceráin, A.¹⁰ Ezpeleta, O.¹¹ Monge, A.¹²

18
- 3042762404
- H. Cerecetto, M. González, S. Onetto, P. Saenz, O. Ezpeleta, A. López de Ceráin, A. Monge, Arch. Pharm. Pharm. Med. Chem. 2004, 337, 247-258;
- (2004) Arch. Pharm. Pharm. Med. Chem. , vol.337 , pp. 247-258
- Cerecetto, H.¹ González, M.² Onetto, S.³ Saenz, P.⁴ Ezpeleta, O.⁵ López De Ceráin, A.⁶ Monge, A.⁷

19
- 4544287322
- H. Cerecetto, M. González, M. Risso, P. Saenz, C. Olea-Azar, A. M. Bruno, A. Azqueta, A. López de Ceráin, A. Monge, Arch. Pharm. Pharm. Med. Chem. 2004, 337, 271-280;
- (2004) Arch. Pharm. Pharm. Med. Chem. , vol.337 , pp. 271-280
- Cerecetto, H.¹ González, M.² Risso, M.³ Saenz, P.⁴ Olea-Azar, C.⁵ Bruno, A.M.⁶ Azqueta, A.⁷ López De Ceráin, A.⁸ Monge, A.⁹

20
- 12144272242
- H. Cerecetto, M. González, M. L. Lavaggi, A. Azqueta, A. López de Ceráin, A. Monge, J. Med. Chem. 2005, 48, 21-23;
- (2005) J. Med. Chem. , vol.48 , pp. 21-23
- Cerecetto, H.¹ González, M.² Lavaggi, M.L.³ Azqueta, A.⁴ López De Ceráin, A.⁵ Monge, A.⁶

21
- 21044444841
- M. H. Torre, D. Gambino, J. Araujo, H. Cerecetto, M. González, M. L. Lavaggi, A. Azqueta, A. López de Cerain, A. Monge, U. Abram, A. J. Costa-Filho, Eur. J. Med. Chem. 2005, 40, 473-480.
- (2005) Eur. J. Med. Chem. , vol.40 , pp. 473-480
- Torre, M.H.¹ Gambino, D.² Araujo, J.³ Cerecetto, H.⁴ González, M.⁵ Lavaggi, M.L.⁶ Azqueta, A.⁷ López De Cerain, A.⁸ Monge, A.⁹ Abram, U.¹⁰ Costa-Filho, A.J.¹¹

22
- 0031693970
- A. Monge, A. López de Ceráin, O. Ezpeleta, H. Cerecetto, E. Dias, R. Di Maio, M. Gonzalez, S. Onetto, M. Risso, G. Seoane, F. Zinola, C. Olea-Azar, Pharmazie 1998, 53, 698-702;
- (1998) Pharmazie , vol.53 , pp. 698-702
- Monge, A.¹ López De Ceráin, A.² Ezpeleta, O.³ Cerecetto, H.⁴ Dias, E.⁵ Di Maio, R.⁶ Gonzalez, M.⁷ Onetto, S.⁸ Risso, M.⁹ Seoane, G.¹⁰ Zinola, F.¹¹ Olea-Azar, C.¹²

23
- 0035492204
- M. Boiani, H. Cerecetto, M. González, M. Risso, C. Olea-Azar, O. E. Piro, E. E. Castellano, A. López de Ceráin, O. Ezpeleta, A. Monge, Eur. J. Med. Chem. 2001, 36, 771-782;
- (2001) Eur. J. Med. Chem. , vol.36 , pp. 771-782
- Boiani, M.¹ Cerecetto, H.² González, M.³ Risso, M.⁴ Olea-Azar, C.⁵ Piro, O.E.⁶ Castellano, E.E.⁷ López De Ceráin, A.⁸ Ezpeleta, O.⁹ Monge, A.¹⁰

24
- 2142662867
- M. Boiani, H. Cerecetto, M. González, Farmaco 2004, 59, 405-412;
- (2004) Farmaco , vol.59 , pp. 405-412
- Boiani, M.¹ Cerecetto, H.² González, M.³

25
- 85081437323
- in press
- G. Aguirre, M. Boiani, H. Cerecetto, M. Fernández, M. González, E. León, C. Pintos, S. Raymondo, C. Arredondo, J. P. Pacheco, M. A. Basombrio, Pharmazie 2006, in press.
- (2006) Pharmazie
- Aguirre, G.¹ Boiani, M.² Cerecetto, H.³ Fernández, M.⁴ González, M.⁵ León, E.⁶ Pintos, C.⁷ Raymondo, S.⁸ Arredondo, C.⁹ Pacheco, J.P.¹⁰ Basombrio, M.A.¹¹

26
- 0031728616
- A. Monge, A. López de Ceráin, O. Ezpeleta, H. Cerecetto, E. Dias, R. Di Maio, M. González, S. Onetto, G. Seoane, L. Suescun, R. Mariezcurrena, Pharmazie 1998, 53, 758-764.
- (1998) Pharmazie , vol.53 , pp. 758-764
- Monge, A.¹ López De Ceráin, A.² Ezpeleta, O.³ Cerecetto, H.⁴ Dias, E.⁵ Di Maio, R.⁶ González, M.⁷ Onetto, S.⁸ Seoane, G.⁹ Suescun, L.¹⁰ Mariezcurrena, R.¹¹

27
- 0033645456
- H. Cerecetto, M. González, M. Risso, G. Seoane, A. López, de Ceráin, O. Ezpeleta, A. Monge, L. Suescun, A. Mombrú, A. M. Bruno, Arch. Pharm. Pharm. Med. Chem. 2000, 333, 387-393.
- (2000) Arch. Pharm. Pharm. Med. Chem. , vol.333 , pp. 387-393
- Cerecetto, H.¹ González, M.² Risso, M.³ Seoane, G.⁴ López De Ceráin, A.⁵ Ezpeleta, O.⁶ Monge, A.⁷ Suescun, L.⁸ Mombrú, A.⁹ Bruno, A.M.¹⁰

28
- 85081439101
- S. Mastrostamatis, M. Papadopoulos, I. Pirmettis, E. Paschali, A Varvarigou, C. Stassinopoulou, C. Raptopoulou, A. Terzis, E. Chiotellis J. Med. Chem. 1994, 37, 3312-3218;
- (1994) J. Med. Chem. , vol.37 , pp. 3312-13218
- Mastrostamatis, S.¹ Papadopoulos, M.² Pirmettis, I.³ Paschali, E.⁴ Varvarigou, A.⁵ Stassinopoulou, C.⁶ Raptopoulou, C.⁷ Terzis, A.⁸ Chiotellis, E.⁹

29
- 2742532205
- I. Pirmettis, M. Papadopoulos, S. Mastrostamatis, C. Raptopoulou, A. Terzis, E. Chiotellis, Inorg. Chem. 1996, 35, 1685-1691.
- (1996) Inorg. Chem. , vol.35 , pp. 1685-1691
- Pirmettis, I.¹ Papadopoulos, M.² Mastrostamatis, S.³ Raptopoulou, C.⁴ Terzis, A.⁵ Chiotellis, E.⁶

30
- 0034644268
- M. Friebe, A. Mahmood, H Spies, R. Berger, B. Johannsen, A. Mohamed, M. Eisenhut, C. Bolzati, A. Davis, A. Jones, J. Med. Chem. 2000, 43, 2745-2752;
- (2000) J. Med. Chem. , vol.43 , pp. 2745-2752
- Friebe, M.¹ Mahmood, A.² Spies, H.³ Berger, R.⁴ Johannsen, B.⁵ Mohamed, A.⁶ Eisenhut, M.⁷ Bolzati, C.⁸ Davis, A.⁹ Jones, A.¹⁰

31
- 0035855595
- M. Friebe, A. Mahmood, C. Bolzati, A. Drews, B. Johannsen, M. Eisenhut, D. Kraemer, A. Davis, A. Jones, J. Med. Chem. 2001, 44, 3132-3140;
- (2001) J. Med. Chem. , vol.44 , pp. 3132-3140
- Friebe, M.¹ Mahmood, A.² Bolzati, C.³ Drews, A.⁴ Johannsen, B.⁵ Eisenhut, M.⁶ Kraemer, D.⁷ Davis, A.⁸ Jones, A.⁹

32
- 0036164064
- A. León, A. Rey, L. Mallo, M. Papadopoulos, I. Pirmettis, E. León, M. Pagano, E. Manta, M. Incerti, C. Raptopoulou, A. Terzis, E. Chiotellis, Nucl. Med. Biol. 2002, 29, 217-226.
- (2002) Nucl. Med. Biol. , vol.29 , pp. 217-226
- León, A.¹ Rey, A.² Mallo, L.³ Papadopoulos, M.⁴ Pirmettis, I.⁵ León, E.⁶ Pagano, M.⁷ Manta, E.⁸ Incerti, M.⁹ Raptopoulou, C.¹⁰ Terzis, A.¹¹ Chiotellis, E.¹²

33
- 12344273021
- H. Cerecetto, W. Porcal, Mini Rev. Med. Chem. 2005, 5, 57-71.
- (2005) Mini Rev. Med. Chem. , vol.5 , pp. 57-71
- Cerecetto, H.¹ Porcal, W.²

34
- 85081437801
- Academic Press Inc.
- nd Ed., Academic Press Inc., 1989, Vol. 3, 586-599.
- (1989) nd Ed. , vol.3 , pp. 586-599
- Sandler, S.R.¹ Karo, W.²

35
- 48749138921
- R. N. Young, J. Y. Gauthier, W. Coombs, Tet. Lett. 1984, 25, 1753-1756.
- (1984) Tet. Lett. , vol.25 , pp. 1753-1756
- Young, R.N.¹ Gauthier, J.Y.² Coombs, W.³

36
- 0034732189
- A. Rey, M. Papadopoulos, L. Mallo, I. Pirmettis, E. León, C. Raptopoulou, E. Manta, E. Chiotellis, A. León, J. Lab. Cpd. Radiopharm. 2000, 43, 347-358;
- (2000) J. Lab. Cpd. Radiopharm. , vol.43 , pp. 347-358
- Rey, A.¹ Papadopoulos, M.² Mallo, L.³ Pirmettis, I.⁴ León, E.⁵ Raptopoulou, C.⁶ Manta, E.⁷ Chiotellis, E.⁸ León, A.⁹

37
- 12944288239
- A. Rey, I. Pirmettis, M. Pelecanou, M. Papadopoulos, C. Raptopoulou, L. Mallo, C. Stassinopoulou, A. Terzis, E. Chiotellis, A. Leon, Inorg. Chem. 2000, 39, 4211-4218;
- (2000) Inorg. Chem. , vol.39 , pp. 4211-4218
- Rey, A.¹ Pirmettis, I.² Pelecanou, M.³ Papadopoulos, M.⁴ Raptopoulou, C.⁵ Mallo, L.⁶ Stassinopoulou, C.⁷ Terzis, A.⁸ Chiotellis, E.⁹ Leon, A.¹⁰

38
- 0035146970
- A. Rey, M. Papadopoulos, E. León, L. Mallo, I. Pirmettis, E. Manta, C. Raptopoulou, E. Chiotellis, A. Leon., Appl. Radiat. Isot. 2001, 53, 429-434.
- (2001) Appl. Radiat. Isot. , vol.53 , pp. 429-434
- Rey, A.¹ Papadopoulos, M.² León, E.³ Mallo, L.⁴ Pirmettis, I.⁵ Manta, E.⁶ Raptopoulou, C.⁷ Chiotellis, E.⁸ Leon, A.⁹

39
- 0001912909
- J. Corbin, K. Miller, N. Pariyadath, S. Wherland, L. Bruce, E. Stiefel, Inorg. Chim. Acta. 1984, 90, 41-51.
- (1984) Inorg. Chim. Acta. , vol.90 , pp. 41-51
- Corbin, J.¹ Miller, K.² Pariyadath, N.³ Wherland, S.⁴ Bruce, L.⁵ Stiefel, E.⁶

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