Diastereoselectivity in the solid-phase synthesis of peptide heterocycle hybrids

Tetrahedron Letters

Volumn 45, Issue 33, 2004, Pages 6333-6336

  Grimes Jr , John H ^a   Zheng, Weifan ^a   Kohn, Wayne D ^a  

^a ELI LILLY AND COMPANY   (United States)

Author keywords

2 D NMR; Peptide heterocycle; Solid phase synthesis; Stereoselective cyclization

Indexed keywords

HETEROCYCLIC COMPOUND; HYBRID PROTEIN;

ARTICLE; CONFORMATIONAL TRANSITION; NUCLEAR MAGNETIC RESONANCE; SOLID; STEREOCHEMISTRY; STRUCTURE ANALYSIS; SYNTHESIS;

THIA;

EID: 3242742816     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.tetlet.2004.06.075     Document Type: Article

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7. 3CN) followed by lyophilization