Interparticle van der Waals force in powder flowability and compactibility

International Journal of Pharmaceutics

Volumn 280, Issue 1-2, 2004, Pages 77-93

  Li, Qin ^a   Rudolph, Victor ^a   Weigl, Bernhard ^b   Earl, Alan ^c  

^a UNIVERSITY OF QUEENSLAND   (Australia)

^b BASF SE   (Germany)

^c Qld 4106   (Australia)

Author keywords

Compactibility; Flowability; Hausner ratio; Interparticle adhesion force; Tablet strength; Van der Waals force

Indexed keywords

EXCIPIENT; PARACETAMOL;

ARTICLE; FLOW RATE; FORCE; MATERIAL STATE; PARTICULATE MATTER; POWDER; PRIORITY JOURNAL; TABLET; VALIDATION PROCESS;

CHEMISTRY, PHARMACEUTICAL; COMPRESSIVE STRENGTH; PARTICLE SIZE; POWDERS;

EID: 3242672320     PISSN: 03785173     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ijpharm.2004.05.001     Document Type: Article

References (41)

1. Abdullah E.C., Geldart D. The use of bulk density measurements as flowability indicators. Powder Technol. 102:1999;151-165
2. Alderborn, G., 1996. Particle dimensions. In: Nystrom, C. (Ed.), Pharmaceutical Powder Compaction Technology. Marcel Dekker, Inc., New York, pp. 245-282.
3. Beach E.R., Tormoen G.W., Drelich J., Han R. Pull-off force measurements between rough surfaces by atomic force microscopy. J. Colloid Interface Sci. 247:2002;84-99
4. Beyer T., Day G.M., Price S.L. The prediction, morphology, and mechanical properties of the polymorphs of paracetamol. J. Am. Chem. Soc. 123:2001;5086-5094
5. Bolhuis, G.K., Chowhan, Z.T., 1996. Materials for direct compaction. In: Nystrom, C. (Ed.), Pharmaceutical Powder Compaction Technology. Marcel Dekker, Inc., pp. 419-500.
6. Davies, P.N., Newton, J.M., 1996. Mechanical strength. In: Nystrom, C. (Ed.), Pharmaceutical Powder Compaction Technology. Marcel Dekker, New York, pp. 165-191.
7. Derjaguin, B.V., Abrikosova, I.I., Lifshitz, E.M., 1956. Q. Rev. Chem. Soc. 10, 295.
8. Fachaux J.M., Guyot-Hermann A.M., Guyot J.C., Conflant P., Drache M., Veesler S., Boistelle R. Pure Paracetamol for direct compression: part I. Development of sintered-like crystals of Paracetamol. Powder Technol. 82:1995a;123-128
9. Fachaux J.M., Guyot-Hermann A.M., Guyot J.C., Conflant P., Drache M., Veesler S., Boistelle R. Pure Paracetamol for direct compression: part II. Study of the physicochemical and mechanical properties of sintered-like crystals of Paracetamol. Powder Technol. 82:1995b;129-133
10. Fuhrer, C., 1996. Interparticulate attraction mechanisms. In: Nystrom, C. (Ed.), Pharmaceutical Powder Compaction Techology. Marcel Dekker, Inc., New York.
11. Garekani H.A., Ford J.L., Rubinstein M.H., Rajabi-Siahboomi A.R. Highly compressible paracetamol: I: crystallization and characterization. Int. J. Pharm. 208:2000;87-89
12. Geldart D., Harnby N., Wong A.C. Fluidization of cohesive powders. Powder Technol. 37:1984;25-37
13. Geldart D., Wong A.C.Y. Fluidization of powders showing degrees of cohesiveness: I. Bed expansion. Chem. Eng. Sci. 39:1984;1481-1488
14. Gotzinger M., Peukert W. Dispersive forces of particle-surface interactions: direct AFM measurements and modelling. Powder Technol. 130:2003;102-109
15. Guerin E., Tchoreloff P., Leclerc B., Tanguy D., Deleuil M., Couarraze G. Rheological characterization of pharmaceutical powders using tap testing, shear cell and mercury porosimeter. Int. J. Pharm. 189:1999;91-103
16. Hiestand E.N. Dispersion forces and plastic deformation in tablet bond. J. Pharm. Sci. 74:1985;768-770
17. Hiestand E.N. Tablet bond: I. A theoretical model. Int. J. Pharm. 67:1991;217-229
18. Jivraj M., Martini L.G., Thomson C.M. An overview of the different excipients useful for the direct compression of tablets. Pharm. Sci. Technol. Today. 3:2000;58-63
19. Johnson K.L., Kendall K., Roberts A.D. Surface energy and the contact of elastic solids. Proc. R. Soc. Lond. A. 324:1971;301-313
20. Kawakita, K., Ludde, K.-H., 1970. Some considerations on powder compression equations, Powder Technol., 61-68.
21. Kibbe, A.H., 2000. Handbook of Pharmaceutical Excipients. Pharmaceutical press.
22. Krupp H. Particle adhesion theory and experiment. Adv. Colloid Interface Sci. 1:1967;111-239
23. Leuenberger H. The compressibility and compactibility of powder systems. Int. J. Pharm. 12:1982;41-55
24. Martino P.D., Guyot-Hermann A.-M., Conflant P., Drache P., Guyot J.-C. A new pure Paracetamol for direct compression: the orthorhombic form. Int. J. Pharm. 128:1996;1-8
25. Molerus O. Interpretation of Geldart's type A, B, C and D powders by taking into account interparticle cohesion forces. Powder Technol. 33:1982;81-87
26. Muzzio F.J., Shinbrot T., Glasser B.J. Powder technology in the pharmaceutical industry: the need to catch up fast. Powder Technol. 124:2002;1-7
27. Newton J.M., Cook D.T. The strength of tablets of mixed components. J. Pharm. Pharmacol. 29:1977;247-249
28. Podczeck F., Newton J.M., James M.B. Variations in the adhesion force between a drug and carrier particles as a result of changes in the relative humidity of the air. Int. J. Pharm. 149:1997;151-160
29. Quintanilla, M.A.S., Castellanos, A., Valverde, J.M., 2001. Correlation between bulk stresses and interparticle cotnact forces in fine powders. Phys. Rev. E. 64, 031301(1-9).
30. Rabinovich Y.I., Adler J.J., Ata A., Singh R.K., Moudgil B.M. Adhesion between nanoscale rough surfaces I. role of asperity geometry. J. Colloid Interface Sci. 232:2000a;10-16
31. Rabinovich Y.I., Adler J.J., Ata A., Singh R.K., Moudgil B.M. Adhesion between nanoscale rough surfaces II. measurement and comparison with theory. J. Colloid Interface Sci. 232:2000b;17-24
32. Rumpf, H., 1962. In: Knepper, W.A. (Ed.), Agglomeration. Interscience, New York, pp. 379.
33. Rumpf, H., 1970. Zur Theorie der Zugfestigkeit von Agglomeraten bei Kraftübertragung an Kontaktpunkten. Chemie-Ing. Technik, 538.
34. Rumpf, H., 1990. Particle Technology. London, Chapman & Hall.
35. Schussele A., Bauer-Brandl A. Note on the mesaurement of flowability according to the European Pharmacopoeia. Int. J. Pharm. 257:2003;301-304
36. Staniforth, J., 2002. Powder flow. In: Aulton, M.E. (Ed.), Pharmaceutics: The Science of Dosage Form Design. Churchill Livingstone, pp. 197-210.
37. Szabó-Révész, P., Göczõ, H., Pintye-Hódi, Kásajr, P., Erõs, I., Hasznos-Nezdei, M., Farkas, B., 2001. Development of spherical crystal agglomerates of an aspartic acid salt for direct tablet making, Powder Technol. 114, 118-124.
38. van de Lagemaat J., Benkstein K.D., Frank A.J. Relation between particle coordination number and porosity in nanoparticle films: implications to dye-sensitized solar cells. J. Phys. Chem. B. 105:2001;12433-12436
39. van Veen B., Maarschalk K.V.D.V., Bolhuis G.K., Zuurman K., Frijlink H.W. Tensile strength of tablets containing two materials with a different compaction behaviour. Int. J. Pharm. 203:2000;71-79
40. Yu A.B., Hall J.S. Packing of fine powders subjected to tapping. Powder Technol. 78:1994;247-256
41. Zenz, F.A., Othmer, D.F., 1960. Fluidization and Fluid-Particle Systems. New York, Reinhold Publishing Corporation.