Synthesis and dopamine receptor binding of sulfur-containing aporphines

Bioorganic and Medicinal Chemistry

Volumn 14, Issue 6, 2006, Pages 1918-1923

  Tóth, Miklós ^a   Berényi, Sándor ^a   Csutorás, Csaba ^b   Kula, Nora S ^c   Zhang, Kehong ^c   Baldessarini, Ross J ^c   Neumeyer, John L ^c  

^a UNIVERSITY OF DEBRECEN   (Hungary)

^b ESZTERHÁZY KÁROLY UNIVERSITY   (Hungary)

^c MCLEAN HOSPITAL   (United States)

Author keywords

Apomorphine; Aporphine derivatives; D2 receptors; Dopamine agonists

Indexed keywords

2 ETHYLTHIO N N PROPYLNORAPOMORPHINE; 2 MERCAPTOAPOCODEINE DERIVATIVE; 2 MERCAPTOAPOMORPHINE DERIVATIVE; 2 METHYLTHIO N N PROPYLNORAPOMORPHINE; 2 METHYLTHIO N PROPYLNORAPOCODEINE; 2 METHYLTHIOAPOCODEINE; 2 METHYLTHIOAPOMORPHINE; 2 PROPYLTHIO N N PROPYLNORAPOMORPHINE; APOMORPHINE; APORPHINE DERIVATIVE; DI ( N PROPYLNORAPOCODEINE 2 YL)SULFIDE; DI (APOCODEINE 2 YL)SULFIDE; DI (APOMORPHINE 2 YL)SULFIDE; DI (N PROPYLNORAPOMORPHINE 2 YL)SULFIDE; DOPAMINE 2 RECEPTOR; DOPAMINE RECEPTOR STIMULATING AGENT; HYDROGEN SULFIDE; MESYLIC ACID; METHANETHIOL; PROPYLNORAPOMORPHINE; SULFUR DERIVATIVE; THEBAINE; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; CATALYSIS; CONTROLLED STUDY; DRUG BIOAVAILABILITY; DRUG MECHANISM; DRUG RECEPTOR BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; LOCOMOTION; MALE; MOTOR ACTIVITY; NONHUMAN; RAT; REACTION ANALYSIS;

ANIMALS; APORPHINES; BRAIN; DRUG EVALUATION, PRECLINICAL; MALE; MOLECULAR STRUCTURE; MOTOR ACTIVITY; RATS; RECEPTORS, DOPAMINE; SULFUR;

ANIMALIA;

EID: 32144458938     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2005.10.049     Document Type: Article

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