Synthesis and in vivo evaluation of a PET radioligand for imaging the endothelin-A receptor

Nuclear Medicine and Biology

Volumn 33, Issue 1, 2006, Pages 15-19

  Mathews, William B ^a   Zober, Tamas G ^a   Ravert, Hayden T ^a   Scheffel, Ursula ^a   Hilton, John ^a   Sleep, Darryl ^b   Dannals, Robert F ^a   Szabo, Zsolt ^a  

^a DEPARTMENT OF PATHOLOGY   (United States)

^b ABBOTT LABORATORIES   (United States)

Author keywords

ABT 627; Atrasentan; Baboon; Endothelin; PET

Indexed keywords

ATRASENTAN; CARBON 11; ENDOTHELIN A RECEPTOR;

ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; BABOON; CONTROLLED STUDY; DRUG DISTRIBUTION; DRUG METABOLISM; DRUG RECEPTOR BINDING; DRUG UPTAKE; HEART MUSCLE; IN VIVO STUDY; MALE; MOUSE; NONHUMAN; ORGAN DISTRIBUTION; POSITRON EMISSION TOMOGRAPHY; TISSUE DISTRIBUTION;

ANIMALS; CARBON RADIOISOTOPES; FEASIBILITY STUDIES; MALE; METABOLIC CLEARANCE RATE; MICE; ORGAN SPECIFICITY; PAPIO; POSITRON-EMISSION TOMOGRAPHY; PYRROLIDINES; RADIOPHARMACEUTICALS; RECEPTOR, ENDOTHELIN A; SPECIES SPECIFICITY; TISSUE DISTRIBUTION;

EID: 31844454096     PISSN: 09698051     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.nucmedbio.2005.07.012     Document Type: Article

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