Synthesis of 3-substituted 1,4-benzodiazepin-2-ones

Journal of the Brazilian Chemical Society

Volumn 9, Issue 4, 1998, Pages 375-379

  Kim, Kyungjin ^a   Volkman, Steven K ^a   Ellman, Jonathan A ^a  

^a UNIVERSITY OF CALIFORNIA   (United States)

Author keywords

Benzodiazepine enolate alkylation; Systemic lupus erythematosus

Indexed keywords

EID: 3042861425     PISSN: 01035053     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (21)

1. Sternbach, L.H. J. Med. Chem. 1979, 22, 1.
2. Bock, M.G.; Dipardo, R.M.; Evans, B.E.; Rittle, K.E.; Whitter, W.L.; Veber, D.F.; Anderson, P.S.; Freidinger, R.M. J. Med. Chem. 1989, 32, 13.
3. Romer, D.; Buschler, H.H.; Hill, R.C.; Maurer, R.; Petcher, T.J.; Zeugner, H.; Benson, W.; Finner, E.; Milkowski, W.; Thies, P.W. Nature 1982, 298, 759.
4. Komeki, E.; Erlich, Y.H.; Lenox, R.H. Science 1984, 226, 1454.
5. Hsu, M.C.; Schutt, A.D.; Holly, M.; Slice, L.W.; Sherman, M.I.; Richman, D.D.; Potash, J.M.; Volsky, D.F. Science 1991, 254, 1799.
6. Pauwels, R.; Andries, K.; Desmyter, J.; Schols, D.; Kukla, M.J.; Breslin, H.; Raeymaeckers, A.; Van, G. Nature 1990, 343, 470.
7. James, G.L.; Goldstein, J.L.; Brown, M.S.; Rawson, I.E.; Somers, T.C.; Medowell, R.S.; Crowley, C.W.; Lucas, B.K.; Levinson, A.D.; Marsters, J.C. Science 1993, 260, 1937.
8. Bunin, B.A.; Ellman, J.A. J. Am. Chem. Soc. 1992, 114, 10997.
9. Bunin, B.A.; Plunkett, M.J.; Ellman, J.A. Proc. Natl. Acad. Sci. U.S.A. 1994, 6, 4708.
10. Plunkett, M.J.; Ellman, J.A. J. Am. Chem. Soc. 1995, 117, 3306.
11. Bunin, B.A.; Plunkett, M.J.; Ellman, J.A. Methods Enzymol. 1995, 267, 448.
12. Boojamra, C.G.; Burow, K.M.; Ellman, J.A. J. Org. Chem. 1997, 62, 1240.
13. Stevens, S.Y.; Bunin, B.A.; Plunkett, M.J.; Swanson, P.C.; Ellman, J.A.; Glick, G.D. J. Am. Chem. Soc. 1996, 118, 10650.
14. Hahn, B.H. N. Eng. J. Med. 1998, 338, 1359.
15. Bock, M.G.; Dipardo, R.M.; Evans, B.E.; Rittle, K.E.; Veber, D.F.; Freidinger, R.M.; Hirshfield, J.; Springer, J.P. J. Org. Chem. 1987, 52, 3232.
16. Fryer, R.I.; Earley, J.V.; Sternbach, L.H. J. Org. Chem. 1969, 34, 649.
17. Reitter, B.E.; Sachdeva, Y.P.; Wolfe, J.F. J. Org. Chem. 1981, 46, 3945.
18. Butcher, J. W.; Liverton, N.J.; Seinick, H.G.; Elliot, J.; Smith, G.R. Tetrahedron Lett. 1996, 37, 6685.
19. Davis, R.B.; Pizzini, L.C. J. Org. Chem. 1960, 25, 1884.
20. Sternbach, L.H.; Fryer, R.I.; Metlesics, W.; Reeder, E.; Sach, G.; Saucy, G.; Stempel, A. J. Org. Chem. 1962, 27, 3788.
21. Node, M.; Nishide, K.; Fujita, E. J. Org. Chem. 1980, 45, 4275.