Tyrphostins are inhibitors of guanylyl and adenylyl cyclases

Biochemistry

Volumn 43, Issue 25, 2004, Pages 8247-8255

  Jaleel, Mahaboobi ^a   Shenoy, Avinash R ^a   Visweswariah, Sandhya S ^a  

^a INDIAN INSTITUTE OF SCIENCE   (India)

Author keywords

[No Author keywords available]

Indexed keywords

BIOLOGICAL MEMBRANES; CHEMICAL MODIFICATION; ENZYME INHIBITION; ENZYME KINETICS; GENETIC ENGINEERING; PROTEINS; SUBSTRATES;

FLUID BALANCE; INTRACELLULAR DOMAINS; TRANSMEMBRANE DOMAINS (TMD);

BIOCHEMISTRY;

ADENINE NUCLEOTIDE; ADENYLATE CYCLASE INHIBITOR; ENTEROTOXIN; GUANYLATE CYCLASE INHIBITOR; GUANYLIN; PROTEIN TYROSINE KINASE INHIBITOR; TYRPHOSTIN; UNCLASSIFIED DRUG; UROGUANYLIN;

ARTICLE; CARBOXY TERMINAL SEQUENCE; COMPETITIVE INHIBITION; CONTROLLED STUDY; COVALENT BOND; DRUG POTENCY; ENZYME ANALYSIS; ENZYME INHIBITION; ENZYME STRUCTURE; EVALUATION; HUMAN; HUMAN CELL; HUMAN TISSUE; IC 50; INHIBITION KINETICS; INTESTINE; PRIORITY JOURNAL; PROTEIN DOMAIN; PROTEIN STRUCTURE; STRUCTURE ACTIVITY RELATION;

ADENYLATE CYCLASE; ANIMALS; CATALYTIC DOMAIN; CELL LINE; CYCLIC GMP; CYTOSOL; DOGS; ENZYME INHIBITORS; ESCHERICHIA COLI; GUANOSINE TRIPHOSPHATE; GUANYLATE CYCLASE; HUMANS; INHIBITORY CONCENTRATION 50; KINETICS; MANGANESE; MEMBRANE PROTEINS; PROTEIN-TYROSINE KINASES; RABBITS; RADIOLIGAND ASSAY; RECEPTORS, PEPTIDE; RECOMBINANT PROTEINS; SPODOPTERA; STRUCTURE-ACTIVITY RELATIONSHIP; TYRPHOSTINS;

INSECTA;

EID: 3042604812     PISSN: 00062960     EISSN: None     Source Type: Journal    
DOI: 10.1021/bi036234n     Document Type: Article

References (44)

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