New routes to oxindole derivatives

Monatshefte fur Chemie

Volumn 135, Issue 6, 2004, Pages 697-711

  Porcs Makkay, Márta ^a   Volk, Balázs ^a   Kapiller Dezsöfi, Rita ^a   Mezei, Tibor ^a   Simig, Gyula ^a  

^a EGIS PHARMACEUTICALS LTD   (Hungary)

Author keywords

Acylation; Alkylation; Isatins; Oxindoles; Regioselectivity

Indexed keywords

INDOLE DERIVATIVE; OXINDOLE;

ACYLATION; ALKYLATION; CHEMICAL PROCEDURES; CHEMICAL REACTION; CONFERENCE PAPER; DRUG SYNTHESIS; STEREOCHEMISTRY;

EID: 2942594801     PISSN: 00269247     EISSN: None     Source Type: Journal    
DOI: 10.1007/s00706-003-0127-9     Document Type: Conference Paper

References (46)

1. Howard HR, Prakash C, Seeger TF (1994) Drugs Future 19: 560
2. DeMarinis RM, Hieble JP (1989) Drugs Future 14: 781
3. Robertson DW, Hayes JS (1986) Drugs Future 11: 377
4. Robinson C (1990) Drugs Future 15: 898
5. (1993) Drugs Future 18: 875
6. Robinson RP, Reiter LA, Barth WE, Campeta AM, Cooper K, Cronin BJ, Destito R, Donahue KM, Falkner FC, Fiese EF, Johnson DL, Kuperman AV, Liston TE, Malloy D, Martin JJ, Mitchell DY, Rusek FW, Shamblin SL, Wright CF (1996) J Med Chem 39: 10
7. Junge H (1973) Ger Offen 2158955; (1973) Chem Abstr 79: 66169z
8. Kadin SB (1985) EP 153818; (1986) Chem Abstr 104: 88427u
9. Crawford ThCh (1985) EP 155828; (1986) Chem Abstr 104: 109466y
10. Kadin SB (1985) EP 156 603; (1986) Chem Abstr 104: 109468a
11. Blaskó G, Lukács Gy, Reiter J, Flórián E, Porcs-Makkay M, Mezei T, Simig Gy (1997) WO 9736895; (1997) Chem Abstr 127: 318879z
12. Porcs-Makkay M, Simig Gy (2000) Org Process Res Dev 4: 10
13. Caramella P, Coda Corsico A, Corsaro A, Del Monte D, Marinone Albini F (1982) Tetrahedron 38: 173
14. a) Beccalli EM, Marchesini A (1992) Synthesis 265;
15. b) Beccalli EM, Marchesini A, Pilati T (1992) Synthesis 891;
16. c) Beccalli EM, Marchesini A (1992) Tetrahedron 48: 5359;
17. d) Beccalli EM, Marchesini A, Pilati T (1993) Tetrahedron 49: 4741;
18. e) Beccalli EM, Marchesini A (1993) Synth Comm 23: 2945;
19. f) Beccalli EM, Marchesini A, Pilati T (1994) Tetrahedron 50: 12697;
20. g) Beccalli EM, Marchesini A, Pilati T (1994) J Chem Soc Perkin Trans 1 579;
21. h) Beccalli EM, Marchesini A (1995) Org Prep Proc Int 27: 113;
22. i) Beccalli EM, Marchesini A, Pilati T (1996) Tetrahedron 52: 3029
23. Robinson RP, Donahue KM (1994) J Het Chem 31: 1541
24. Porcs-Makkay M, Simig Gy (2001) J Het Chem 38: 451
25. a) Kadin SB (1986) EP 208510; (1987) Chem Abstr 106: 138254z;
26. b) Kadin SB (1987) US 4725616; (1989) Chem Abstr 110: 23728x
27. Porcs-Makkay M, Kálmán A, Argay Gy, Simig Gy (2000) Tetrahedron 56: 5893
28. a) Gruda I (1972) Can J Chem 50: 18;
29. b) Reisch J, Müller M, Labitzke H (1984) Arch Pharm (Weinheim, Germany) 317: 639;
30. c) Kende AS, Hodges JC (1982) Synth Commun 12: 1
31. a) Nozoye T, Nakai T, Kubo A (1977) Chem Pharm Bull 25: 196;
32. b) Mertens A, Müller-Beckmann B, Kampe W, Hölck JP, von der Saal W (1987) J Med Chem 30: 1279;
33. c) Tacconi G, Maggi LD, Righetti P, Desimoni G, Azzolina O, Ghislandi V (1976) J Chem Soc Perkin Trans 2 150
34. Wenkert E, Bringi NV (1958) J Am Chem Soc 80: 5575
35. Wenkert E, Bringi NV, Choulett HE (1982) Acta Chem Scand Ser B 36: 348
36. Volk B, Mezei T, Simig Gy (2002) Synthesis 595
37. a) McEvoy FJ, Allen GR Jr (1973) J Org Chem 38: 3350;
38. b) Wenkert E, Bindra JS, Chang CJ, Cochran DW, Rearick DE (1974) J Org Chem 39: 1662;
39. c) Nozoye T, Shibanuma Y (1975) Yakugaku Zasshi 95: 710; (1975) Chem Abstr 83: 131400;
40. c) Nozoye T, Shibanuma Y (1975) Yakugaku Zasshi 95: 710; (1975) Chem Abstr 83: 131400;
41. d) Rajanbabu TV, Chenard BL, Petti MA (1986) J Org Chem 51: 1704;
42. e) Rasmussen HB, MacLeod JK (1997) J Nat Prod 60: 1152
43. a) Karp GM (1993) Org Prep Proc Int 25: 481 and references cited therein;
44. b) Muchowski JM (1969) Can J Chem 47: 857;
45. c) Wells AS, Lewis NJ, Walsgrove TC, Oxley P, Fortunak JM (1994) WO 9415918; (1994) Chem Abstr 121: 179494f
46. Volk B, Simig Gy (2003) Eur J Org Chem 3991.