New practical synthesis of tenidap

Organic Process Research and Development

Volumn 4, Issue 1, 2000, Pages 10-16

  Porcs Makkay, Márta ^a   Simig, Gyula ^a  

^a EGIS PHARMACEUTICALS LTD   (Hungary)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 0034404019     PISSN: 10836160     EISSN: None     Source Type: Journal    
DOI: 10.1021/op990067a     Document Type: Article

References (21)

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2. (b) Drugs Future 1993, 18 (9), 875.
3. Robinson R. P.; Reiter, L. A.; Barth, W. E.; Campeta, A. M.; Cooper, K.; Cronin, B. J.; Destito, R.; Donahue, K. M.; Falkner, F. C.; Fiese, E. F.; Johnson, D. L.; Kuperman, A. V.; Liston, T. E.; Malloy, D.; Martin, J. J.; Mitchell, D. Y.; Rusek, F. W.; Shamblin, S. L.; Wright, C. F. J. Med. Chem. 1996, 39, 10.
4. Junge, H. (BASF AG). Ger Offen. 21 58955, May 30, 1973; Chem. Abstr. 1973, 79, 66169z.
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6. Crawford, Th. Ch. (Pfizer Inc.). EPA 155,828, March 15, 1985; Chem. Abstr. 1986, 104, 109466y.
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8. Blaskó, G.; Lukács, G.; Reiter, J.; Flórián, E.; Porcs-Makkay, M.; Mezei, T.; Simig, G. (Egis Pharmaceuticals Ltd.). WO 97 36,895, April 3, 1997; Chem. Abstr. 1997, 127, 318879z.
9. 3 at room temperature: Rajeswaran, W. G.; Cohen, L. A. Tetrahedron 1998, 54, 11375.
10. Caramella, P.; Coda Corsico, A.; Corsaro, A.; Del Monte, D.; Marinone Albini, F. Tetrahedron 1982, 38, 173.
11. (a) Beccalli, E. M.; Marchesini, A. Synthesis 1992, 265.
12. (b) Beccalli, E. M.; Marchesini, A.; Pilati T. Synthesis 1992, 891.
13. (c) Beccalli, E. M.; Marchesini, A.; Pilati, T. Tetrahedron 1992, 48, 5359.
14. (d) Beccalli, E. M.; Marchesini, A.; Pilati, T. Tetrahedron 1993, 49, 4741.
15. (e) Beccalli, E. M.; Marchesini, A. Synthetic Comm., 1993, 23, 2945.
16. (f) Beccalli, E. M.; Marchesini, A.; Pilati T. Tetrahedron 1994, 50, 12697.
17. (g) Beccalli, E. M.; Marchesini, A.; Pilati T. J. Chem. Soc., Perkin Trans. 1 1994, 579.
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19. (i) Beccalli, E. M.; Marchesini A.; Pilati, T. Tetrahedron 1996, 52, 3029.
20. Sun, L.; Tran, N.; Tang, F.; App. H.; Hirth, P.; McMahon, G.; Tang, C. J. Med. Chem. 1998, 41, 2588.
21. The authors have deposited atomic coordinates for 11a and 12a with the Cambridge Crystallographic Data Centre. The coordinates can be obtained, on request, from the Director, Cambridge Crystallographic Data Centre, 12 Union Road, Cambridge, CB2 1EZ, UK.