Inhibition of the Staphylococcus aureus sortase transpeptidase SrtA by phosphinic peptidomimetics

Bioorganic and Medicinal Chemistry

Volumn 12, Issue 13, 2004, Pages 3723-3729

  Kruger, Ryan G ^a   Barkallah, Salim ^a   Frankel, Brenda A ^a   McCafferty, Dewey G ^a  

^a UNIVERSITY OF PENNSYLVANIA   (United States)

Author keywords

Antivirulence; Peptidomimetic; Phosphinate; Sortase; Transpeptidase

Indexed keywords

BACTERIAL ENZYME; ENZYME INHIBITOR; GAMMA GLUTAMYLTRANSFERASE; PEPTIDE DERIVATIVE; PHOSPHINIC ACID DERIVATIVE; SORTASE;

AMINO ACID SEQUENCE; ARTICLE; CONTROLLED STUDY; DRUG SYNTHESIS; ENZYME INHIBITION; ENZYME SUBSTRATE; NONHUMAN; STAPHYLOCOCCUS AUREUS;

AMINO ACID SEQUENCE; AMINOACYLTRANSFERASES; BACTERIAL PROTEINS; BIOMIMETIC MATERIALS; CATALYSIS; CYSTEINE ENDOPEPTIDASES; ENZYME INHIBITORS; KINETICS; MOLECULAR STRUCTURE; PHOSPHOPEPTIDES; STAPHYLOCOCCUS AUREUS;

POSIBACTERIA; STAPHYLOCOCCUS; STAPHYLOCOCCUS AUREUS;

EID: 2942546536     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2004.03.066     Document Type: Article

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