Preclinical pharmacology of bilastine, a new selective histamine H 1 receptor antagonist: Receptor selectivity and in Vitro antihistaminic activity

Drugs in R and D

Volumn 6, Issue 6, 2005, Pages 371-384

  Corcóstegui, Reyes ^a   Labeaga, Luis ^a   Innerárity, Ana ^a   Berisa, Agustin ^a   Orjales, Aurelio ^a  

^a FAES SA   (Spain)

Author keywords

[No Author keywords available]

Indexed keywords

ALPHA 1 ADRENERGIC RECEPTOR; BILASTINE; BRADYKININ; CALCIUM; HISTAMINE H1 RECEPTOR; HISTAMINE H1 RECEPTOR ANTAGONIST; HISTAMINE H2 RECEPTOR; HISTAMINE H3 RECEPTOR; LEUKOTRIENE D4; MEPYRAMINE; MUSCARINIC M3 RECEPTOR; SEROTONIN; TRITIUM; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ANTIINFLAMMATORY ACTIVITY; ARTICLE; BINDING AFFINITY; CELL LINE; CEREBELLUM; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG SCREENING; DRUG SELECTIVITY; EMBRYO; GUINEA PIG; HUMAN; HUMAN CELL; ILEUM; IN VITRO STUDY; MALE; NONHUMAN; PRIORITY JOURNAL; PROTEIN EXPRESSION; RAT; RECEPTOR BLOCKING; SMOOTH MUSCLE;

ANIMALS; BENZIMIDAZOLES; BINDING, COMPETITIVE; CELL LINE; DRUG EVALUATION, PRECLINICAL; GUINEA PIGS; HISTAMINE H1 ANTAGONISTS; HUMANS; MALE; ORGAN SPECIFICITY; PIPERIDINES; PROTEIN BINDING; RABBITS; RATS; RECEPTORS, HISTAMINE H1;

EID: 27744581978     PISSN: 11745886     EISSN: 11745886     Source Type: Journal    
DOI: 10.2165/00126839-200506060-00005     Document Type: Article

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