Solubility and prediction of the heat of solution of sodium naproxen in aqueous solutions

Journal of Pharmaceutical Sciences

Volumn 94, Issue 9, 2005, Pages 1941-1948

  Kim, Young Soo ^a   Méndez Del Río, José R ^a   Rousseau, Ronald W ^a  

^a Georgia Institute of Technology   (United States)

Author keywords

Focused beam reflectance method; Heat of solution; Pseudopolymorphism; Sodium naproxen; Solubility

Indexed keywords

NAPROXEN; NONSTEROID ANTIINFLAMMATORY AGENT; WATER;

AQUEOUS SOLUTION; ARTICLE; DEHYDRATION; DIFFERENTIAL SCANNING CALORIMETRY; DRUG SOLUBILITY; FOCUSED BEAM REFLECTANCE METHOD; HEAT OF SOLUTION; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; HUMAN; REFLECTOMETRY; TEMPERATURE; THERMOGRAVIMETRY;

EID: 27644533755     PISSN: 00223549     EISSN: None     Source Type: Journal    
DOI: 10.1002/jps.20391     Document Type: Article

References (23)

1. Shefter E, Higuchi T. 1963. Dissolution behavior of crystalline solvated and nonsolvated forms of some pharmaceuticals. J Pharm Sci 52:781-791.
2. Peterson ML, McIlroy D, Shaw P, Mustonen JP, Oliveira M, Almarsson Ö. 2003. Crystallization and transformation of acetaminophen trihydrate. Cryst Growth Des 3:761-765.
3. Bettinetti G, Mura P, Sorrenti M, Faucci MT, Negri A. 1999. Physical characterization of picotamide monohydrate and anhydrous picotamide. J Pharm Sci 88:1133-1139.
4. Shefter E, Kmack G. 1967. Phase transitions I. Preliminary study of theophylline hydrate-anhydrate system. J Pharm Sci 56:1028-1029.
5. Reutzel-Edens SM, Bush JK, Magee PA, Stephenson GA, Byrn SR. 2003. Anhydrates and hydrates of olanzapine: Crystallization, solid-state characterization, and structural relationships. Cryst Growth Des 3:897-907.
6. Vippagunta SR, Brittain HG, Grant DJW. 2001. Crystalline solids. Adv Drug Delivery Rev 48:3-26.
7. Byrn SR, Pfeiffer RR, Stephenson G, Grant DJW, Gleason WB. 1994. Solid-state pharmaceutical chemistry. Chem Mater 6:1148-1158.
8. Urakami K, Shono Y, Higashi A, Umemoto K, Godo M. 2002. A Novel method for estimation of transition temperature for polymorphic pairs in pharmaceuticals using heat of solution and solubility data. Chem Pharm Bull 50:263-267.
9. Terada K, Kitano H, Yoshihashi Y, Yonemochi E. 2000. Quantitative correlation between initial dissolution rate and heat of solution of drug. Pharm Res 17:920-924.
10. Suryanarayanan R, Mitchell AG. 1986. Phase transitions of calcium gluceptate. Int J Pharm 32:213-221.
11. Gandhi R, Pillai O, Thilagavathi R, Gopalakrishnan B, Kaul CL, Panchagnula R. 2002. Characterization of azithromycin hydrates. Eur J Pharm Sci 16:175-184.
12. Suryanarayanan R, Mitchell AG. 1985. Evaluation of two concepts of crystallinity using calcium gluceptate as a model compound. Int J Pharm 24:1-17.
13. Kim Y, VanDerveer D, Rousseau RW, Wilkinson AP. 2004. Anhydrous sodium naproxen. Acta Crystallogr E60:m419-m420.
14. 3Na), a non-steroidal antiinflammatory agent. Arch Pharmacol Res 13:166-173.
15. Kim Y, Rousseau RW. 2004. Characterization and solid-state transformations of the pseudopolymorphic forms of sodium naproxen. Cryst Growth Des 4:1211-1216.
16. Shi B, Frederick WJ, Rousseau RW. 2003. Effects of calcium and other ionic impurities on the primary nucleation of burkeite. Ind Eng Chem Res 42:2861-2869.
17. Packer JL, Werner JJ, Latch DE, McNeill K, Arnold WA. 2003. Photochemical fate of pharmaceuticals in the environment: Naproxen, diclofenac, clofibric acid, and ibuprofen. Aquat Sci 65:342-351.
18. Valero M, Carrillo C. 2004. Effect of binary and ternary polyethyleneglycol and/or beta-cyclodextrin complexes on the photochemical and photosensitizing properties of naproxen. J Photochem Photobiol 674:151-160.
19. Barrett P, Glennon B. 2002. Characterizing the metastable zone width and solubility curve using lasentec FBRM and PVM. Chem Eng Res Des 80:799-805.
20. Fujiwara M, Chow PS, Ma DL, Braatz RD. 2002. Paracetamol crystallization using laser backscattering and ATR-FTIR spectroscopy: Metastability, agglomeration, and control. Cryst Growth Des 2:363-370.
21. Stark JG, Wallace HG. 1976. Chemistry data book. SI Ed. London: John Murray.
22. Khankari RK, Law D, Grant DJW. 1992. Determination of water-content in pharmaceutical hydrates by differential scanning calorimetry. Int J Pharm 82:117-127.
23. Grant DJW, Higuchi T. 1990. Solubility behavior of organic compounds. New York: John Wiley.