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Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 24, 2005, Pages 5439-5441

Indole-2-carboxamidines as novel NR2B selective NMDA receptor antagonists

(9) Borza, István a Kolok, Sándor a Ignácz Szendrei, Györgyi a Greiner, István a Tárkányi, Gábor a Galgóczy, Kornél a Horváth, Csilla a Farkas, Sándor a Domány, György a

a GEDEON RICHTER LTD (Hungary)

Author keywords

Indole 2 carboxamidine; NB2B; NMDA

Indexed keywords

AMIDINE; BENZYL DERIVATIVE; FORMALDEHYDE; INDOLE DERIVATIVE; N METHYL DEXTRO ASPARTIC ACID RECEPTOR BLOCKING AGENT;

ANALGESIC ACTIVITY; ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL MODEL; ARTICLE; CARBON NUCLEAR MAGNETIC RESONANCE; CONTROLLED STUDY; DRUG SYNTHESIS; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; INFRARED SPECTROSCOPY; MASS SPECTROMETRY; MOUSE; NONHUMAN; PAIN; PROTON NUCLEAR MAGNETIC RESONANCE; RAT; STRUCTURE ACTIVITY RELATION;

AMINOIMIDAZOLE CARBOXAMIDE; ANIMALS; CALCIUM; CELL CULTURE TECHNIQUES; CEREBRAL CORTEX; IMIDAZOLES; INDOLES; N-METHYLASPARTATE; RATS; RECEPTORS, N-METHYL-D-ASPARTATE;

ANIMALIA;

EID: 27644505056 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/j.bmcl.2005.08.110 Document Type: Article

Times cited : (19)

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