Enantioselective binding to the human organic cation transporter-1 (hOCT1) determined using an immobilized hOCT1 liquid chromatographic stationary phase

Chirality

Volumn 17, Issue 8, 2005, Pages 501-506

  Moaddel, R ^a   Patel, S ^a,b   Jozwiak, K ^a,c   Yamaguchi, R ^a,d   Ho, P C ^a,e   Wainer, Irving W ^a,f  

^a NATIONAL INSTITUTE ON AGING   (United States)

^b UNIVERSITY OF SUNDERLAND   (United Kingdom)

^c MEDICAL UNIVERSITY OF LUBLIN   (Poland)

^d SHIONOGI AND CO LTD   (Japan)

^e NATIONAL UNIVERSITY OF SINGAPORE   (Singapore)

^f NATIONAL INSTITUTE ON AGING   (United States)

Author keywords

Affinity chromatography; Drug transporters; Immobilized cellular membranes; Pharmacophore modeling

Indexed keywords

ALPHA METHYLBENZYLAMINE; ATENOLOL; ORGANIC CATION TRANSPORTER; PROPRANOLOL; PSEUDOEPHEDRINE;

ARTICLE; CHROMATOGRAPHY; COMPETITIVE INHIBITION; ENANTIOMER; ENANTIOSELECTIVITY; HYDROGEN BOND; IC 50; LIQUID CHROMATOGRAPHY; NONHUMAN; PHASE SEPARATION; PRIORITY JOURNAL; PROTEIN BINDING; STATISTICAL SIGNIFICANCE;

ANIMALS; ATENOLOL; BINDING SITES; CELL LINE; CHROMATOGRAPHY, AFFINITY; CHROMATOGRAPHY, LIQUID; DOGS; EPHEDRINE; HUMANS; HYDROGEN BONDING; ORGANIC CATION TRANSPORTER 1; PHENETHYLAMINES; PROPRANOLOL; STEREOISOMERISM;

EID: 25844475717     PISSN: 08990042     EISSN: None     Source Type: Journal    
DOI: 10.1002/chir.20195     Document Type: Article

References (13)

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