(4-Substituted-phenyl)-(5H-10,11-dihydro-pyrrolo [2,1-c][1,4] benzodiazepin-10-yl)-methanone derivatives as vasopressin receptor modulators

Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 22, 2005, Pages 5003-5006

  Venkatesan, Aranapakam M ^a   Grosu, George T ^a   Failli, Amedeo A ^b   Chan, Peter S ^b   Coupet, Joseph ^b   Saunders, Trina ^b   Mazandarani, Hussain ^b   Ru, Xun ^b  

^a WYETH RESEARCH   (United States)

^b PFIZER INC   (United States)

Author keywords

Vasopressin receptor modulators

Indexed keywords

ARGIPRESSIN RECEPTOR; BENZODIAZEPINE DERIVATIVE; LIXIVAPTAN; VASOPRESSIN RECEPTOR ANTAGONIST;

ANIMAL CELL; ANIMAL EXPERIMENT; ARTICLE; CHEMICAL BOND; CONTROLLED STUDY; DRUG POTENCY; DRUG SYNTHESIS; MOUSE; NONHUMAN; RAT; STRUCTURE ACTIVITY RELATION;

BENZODIAZEPINES; BLOOD PLATELETS; HUMANS; INHIBITORY CONCENTRATION 50; MOLECULAR STRUCTURE; PYRROLES; RECEPTORS, VASOPRESSIN; SENSITIVITY AND SPECIFICITY; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 25844449154     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2005.08.007     Document Type: Article

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