-
1
-
-
0033560699
-
PET studies of binding competition between endogenous dopamine and the D1 radiotracer [11C]NNC 756
-
Abi-Dargham A, Simpson N, Kegeles L, Parsey R, Hwang DR, Anjilvel S, Zea-Ponce Y, Lombardo I, Van Heertum R, Mann JJ, et al. (1999) PET studies of binding competition between endogenous dopamine and the D1 radiotracer [11C]NNC 756. Synapse 32:93-109.
-
(1999)
Synapse
, vol.32
, pp. 93-109
-
-
Abi-Dargham, A.1
Simpson, N.2
Kegeles, L.3
Parsey, R.4
Hwang, D.R.5
Anjilvel, S.6
Zea-Ponce, Y.7
Lombardo, I.8
Van Heertum, R.9
Mann, J.J.10
-
2
-
-
0033782021
-
Advantages of heterologous expression of human D2long dopamine receptors in human neuroblastoma SH-SY5Y over human embryonic kidney 293 cells
-
Alberts GL, Pregenzer JF, and Im WB (2000) Advantages of heterologous expression of human D2long dopamine receptors in human neuroblastoma SH-SY5Y over human embryonic kidney 293 cells. Br J Pharmacol 131:514-520.
-
(2000)
Br J Pharmacol
, vol.131
, pp. 514-520
-
-
Alberts, G.L.1
Pregenzer, J.F.2
Im, W.B.3
-
3
-
-
0015904377
-
Comparison of effects of L-dopa, amphetamine and apomorphine on firing rate of rat dopaminergic neurones
-
Bunney BS, Aghajanian GK, and Roth RH (1973a) Comparison of effects of L-dopa, amphetamine and apomorphine on firing rate of rat dopaminergic neurones. Nat New Biol 245:123-125.
-
(1973)
Nat New Biol
, vol.245
, pp. 123-125
-
-
Bunney, B.S.1
Aghajanian, G.K.2
Roth, R.H.3
-
4
-
-
0015742027
-
Dopaminergic neurons: Effect of antipsychotic drugs and amphetamine on single cell activity
-
Bunney BS, Walters JR, Roth RH, and Aghajanian GK (1973b) Dopaminergic neurons: effect of antipsychotic drugs and amphetamine on single cell activity. J Pharmacol Exp Ther 185:560-571.
-
(1973)
J Pharmacol Exp Ther
, vol.185
, pp. 560-571
-
-
Bunney, B.S.1
Walters, J.R.2
Roth, R.H.3
Aghajanian, G.K.4
-
5
-
-
0345406583
-
Scatchard analysis with bolus/infusion administration of [11C]raclopride: Amphetamine effects in anesthetized monkeys
-
Senda M, Kimura Y and Herscovitch P eds Academic Press, San Diego
-
Carson RE, Channing MA, Der MG, Herscovitch P, and Eckelman W (2002) Scatchard analysis with bolus/infusion administration of [11C]raclopride: amphetamine effects in anesthetized monkeys, in Brain Imaging Using PET (Senda M, Kimura Y and Herscovitch P eds) pp 63-69, Academic Press, San Diego.
-
(2002)
Brain Imaging Using PET
, pp. 63-69
-
-
Carson, R.E.1
Channing, M.A.2
Der, M.G.3
Herscovitch, P.4
Eckelman, W.5
-
6
-
-
0037013696
-
Density and affinity of the dopamine D2 receptors in aged symptomatic and asymptomatic MPTP-treated monkeys: PET studies with [11C]raclopride
-
Doudet DJ, Jivan S, Ruth TJ, and Holden JE (2002) Density and affinity of the dopamine D2 receptors in aged symptomatic and asymptomatic MPTP-treated monkeys: PET studies with [11C]raclopride. Synapse 44:198-202.
-
(2002)
Synapse
, vol.44
, pp. 198-202
-
-
Doudet, D.J.1
Jivan, S.2
Ruth, T.J.3
Holden, J.E.4
-
7
-
-
0022595579
-
Quantitative analysis of D2 dopamine receptor binding in the living human brain by PET
-
Farde L, Hall H, Ehrin E, and Sedvall G (1986) Quantitative analysis of D2 dopamine receptor binding in the living human brain by PET. Science (Wash DC) 231:258-261.
-
(1986)
Science (Wash DC)
, vol.231
, pp. 258-261
-
-
Farde, L.1
Hall, H.2
Ehrin, E.3
Sedvall, G.4
-
8
-
-
0028981192
-
Variability in D2-dopamine receptor density and affinity: A PET study with [11C]raclopride in man
-
Farde L, Hall H, Pauli S, and Halldin C (1995) Variability in D2-dopamine receptor density and affinity: a PET study with [11C]raclopride in man. Synapse 20:200-208.
-
(1995)
Synapse
, vol.20
, pp. 200-208
-
-
Farde, L.1
Hall, H.2
Pauli, S.3
Halldin, C.4
-
9
-
-
0031595716
-
Agonist action at D2(long) dopamine receptors: Ligand binding and functional assays
-
Gardner B and Strange PG (1998) Agonist action at D2(long) dopamine receptors: ligand binding and functional assays. Br J Pharmacol 124:978-984.
-
(1998)
Br J Pharmacol
, vol.124
, pp. 978-984
-
-
Gardner, B.1
Strange, P.G.2
-
10
-
-
0021894675
-
Dopamine D2 receptors in the anterior pituitary: A single population without reciprocal antagonist/agonist states
-
George SR, Watanabe M, and Seeman P (1985) Dopamine D2 receptors in the anterior pituitary: a single population without reciprocal antagonist/agonist states. J Neurochem 44:1168-1177.
-
(1985)
J Neurochem
, vol.44
, pp. 1168-1177
-
-
George, S.R.1
Watanabe, M.2
Seeman, P.3
-
11
-
-
0030949522
-
Effect of reserpine-induced depletion of synaptic dopamine on [C-11]raclopride binding to D-2-dopamine receptors in the monkey brain
-
Ginovart N, Farde L, Halldin C, and Swahn CG (1997) Effect of reserpine-induced depletion of synaptic dopamine on [C-11]raclopride binding to D-2-dopamine receptors in the monkey brain. Synapse 25:321-325.
-
(1997)
Synapse
, vol.25
, pp. 321-325
-
-
Ginovart, N.1
Farde, L.2
Halldin, C.3
Swahn, C.G.4
-
12
-
-
0021870454
-
Complete conversion of brain D2 dopamine receptors from the high- to the low-affinity state for dopamine agonists, using sodium ions and guanine nucleotide
-
Grigoriadis D and Seeman P (1985) Complete conversion of brain D2 dopamine receptors from the high- to the low-affinity state for dopamine agonists, using sodium ions and guanine nucleotide. J Neurochem 44:1925-1935.
-
(1985)
J Neurochem
, vol.44
, pp. 1925-1935
-
-
Grigoriadis, D.1
Seeman, P.2
-
13
-
-
0026599216
-
Gpp(NH)p stimulates [3H]raclopride binding to homogenates from human putamen and accumbens
-
Hall H, Halldin C, and Sedvall G (1992) Gpp(NH)p stimulates [3H]raclopride binding to homogenates from human putamen and accumbens. Neurosci Lett 136:79-82.
-
(1992)
Neurosci Lett
, vol.136
, pp. 79-82
-
-
Hall, H.1
Halldin, C.2
Sedvall, G.3
-
14
-
-
0023790321
-
Effects of temperature on the in vitro binding of 3H-raclopride to rat striatal dopamine-D2 receptors
-
Hall H, Wedel I, and Sallemark M (1988) Effects of temperature on the in vitro binding of 3H-raclopride to rat striatal dopamine-D2 receptors. Pharmacol Toxicol 63:118-121.
-
(1988)
Pharmacol Toxicol
, vol.63
, pp. 118-121
-
-
Hall, H.1
Wedel, I.2
Sallemark, M.3
-
15
-
-
0032587503
-
Measurement of striatal D2 dopamine receptor density and affinity with [11C]-raclopride in vivo: A test-retest analysis
-
Hietala J, Nagren K, Lehikoinen P, Ruotsalainen U, and Syvalahti E (1999) Measurement of striatal D2 dopamine receptor density and affinity with [11C]-raclopride in vivo: a test-retest analysis. J Cereb Blood Flow Metab 19:210-217.
-
(1999)
J Cereb Blood Flow Metab
, vol.19
, pp. 210-217
-
-
Hietala, J.1
Nagren, K.2
Lehikoinen, P.3
Ruotsalainen, U.4
Syvalahti, E.5
-
16
-
-
0036714078
-
In vivo receptor assay with multiple ligand concentrations: An equilibrium approach
-
Holden JE, Jivan S, Ruth TJ, and Doudet DJ (2002) In vivo receptor assay with multiple ligand concentrations: an equilibrium approach. J Cereb Blood Flow Metab 22:1132-1141.
-
(2002)
J Cereb Blood Flow Metab
, vol.22
, pp. 1132-1141
-
-
Holden, J.E.1
Jivan, S.2
Ruth, T.J.3
Doudet, D.J.4
-
17
-
-
0033623451
-
(-)-N-[(11)C]Propyl-norapomorphine: A positron-labeled dopamine agonist for PET imaging of D(2) receptors
-
Hwang D, Kegeles LS, and Laruelle M (2000) (-)-N-[(11)C]Propyl- norapomorphine: a positron-labeled dopamine agonist for PET imaging of D(2) receptors. Nucl Med Biol 27:533-539.
-
(2000)
Nucl Med Biol
, vol.27
, pp. 533-539
-
-
Hwang, D.1
Kegeles, L.S.2
Laruelle, M.3
-
18
-
-
1542399582
-
Quantitative analysis of (-)-N-(11)C-propyl-norapomorphine in vivo binding in nonhuman primates
-
Hwang DR, Narendran R, Huang Y, Slifstein M, Talbot PS, Sudo Y, Van Berckel BN, Kegeles LS, Martinez D, and Laruelle M (2004) Quantitative analysis of (-)-N-(11)C-propyl-norapomorphine in vivo binding in nonhuman primates. J Nucl Med 45:338-346.
-
(2004)
J Nucl Med
, vol.45
, pp. 338-346
-
-
Hwang, D.R.1
Narendran, R.2
Huang, Y.3
Slifstein, M.4
Talbot, P.S.5
Sudo, Y.6
Van Berckel, B.N.7
Kegeles, L.S.8
Martinez, D.9
Laruelle, M.10
-
19
-
-
0021844076
-
Specific in vitro and in vivo binding of 3H-raclopride. A potent substituted benzamide drug with high affinity for dopamine D-2 receptors in the rat brain
-
Kohler C, Hall H, Ogren SO, and Gawell L (1985) Specific in vitro and in vivo binding of 3H-raclopride. A potent substituted benzamide drug with high affinity for dopamine D-2 receptors in the rat brain. Biochem Pharmacol 34:2251-2259.
-
(1985)
Biochem Pharmacol
, vol.34
, pp. 2251-2259
-
-
Kohler, C.1
Hall, H.2
Ogren, S.O.3
Gawell, L.4
-
20
-
-
2342543198
-
In vivo binding behavior of dopamine receptor agonist (+)-PD 128907 and implications for the "ceiling effect" in endogenous competition studies with [(11)C]raclopride-a positron emission tomography study in Macaca mulatta
-
Kortekaas R, Maguire RP, Cremers TI, Dijkstra D, van Waarde A, and Leenders KL (2004) In vivo binding behavior of dopamine receptor agonist (+)-PD 128907 and implications for the "ceiling effect" in endogenous competition studies with [(11)C]raclopride-a positron emission tomography study in Macaca mulatta. J Cereb Blood Flow Metab 24:531-535.
-
(2004)
J Cereb Blood Flow Metab
, vol.24
, pp. 531-535
-
-
Kortekaas, R.1
Maguire, R.P.2
Cremers, T.I.3
Dijkstra, D.4
Van Waarde, A.5
Leenders, K.L.6
-
21
-
-
0029972880
-
Affinities and intrinsic activities of dopamine receptor agonists for the hD21 and hD4.4 receptors
-
Lahti RA, Mutin A, Cochrane EV, Tepper PG, Dijkstra D, Wikstrom H, and Tamminga CA (1996) Affinities and intrinsic activities of dopamine receptor agonists for the hD21 and hD4.4 receptors. Eur J Pharmacol 301:R11-R13.
-
(1996)
Eur J Pharmacol
, vol.301
-
-
Lahti, R.A.1
Mutin, A.2
Cochrane, E.V.3
Tepper, P.G.4
Dijkstra, D.5
Wikstrom, H.6
Tamminga, C.A.7
-
22
-
-
0028179235
-
SPECT quantification of [123I]iomazenil binding to benzodiazepine receptors in nonhuman primates. II. Equilibrium analysis of constant infusion experiments and correlation with in vitro parameters
-
Laruelle M, Abi-Dargham A, Al-Tikriti MS, Baldwin RM, Zea-Ponce Y, Zoghbi SS, Charney DS, Hoffer PB, and Innis RB (1994a) SPECT quantification of [123I]iomazenil binding to benzodiazepine receptors in nonhuman primates. II. Equilibrium analysis of constant infusion experiments and correlation with in vitro parameters. J Cereb Blood Flow Metab 14:453-465.
-
(1994)
J Cereb Blood Flow Metab
, vol.14
, pp. 453-465
-
-
Laruelle, M.1
Abi-Dargham, A.2
Al-Tikriti, M.S.3
Baldwin, R.M.4
Zea-Ponce, Y.5
Zoghbi, S.S.6
Charney, D.S.7
Hoffer, P.B.8
Innis, R.B.9
-
23
-
-
0028147183
-
123I]iodobenzofuran and single photon emission computerized tomography
-
123I] iodobenzofuran and single photon emission computerized tomography. Eur J Pharmacol 263:39-51.
-
(1994)
Eur J Pharmacol
, vol.263
, pp. 39-51
-
-
Laruelle, M.1
Al-Tikriti, M.S.2
Zea-Ponce, Y.3
Zoghbi, S.S.4
Baldwin, R.M.5
Charney, D.S.6
Hoffer, P.B.7
Kung, H.F.8
Innis, R.B.9
-
24
-
-
0031030271
-
Microdialysis and SPECT measurements of amphetamine-induced dopamine release in nonhuman primates
-
Laruelle M, Iyer RN, Al-Tikriti MS, Zea-Ponce Y, Malison R, Zoghbi SS, Baldwin RM, Kung HF, Charney DS, Hoffer PB, Innis RB, and Bradberry CW (1997) Microdialysis and SPECT measurements of amphetamine-induced dopamine release in nonhuman primates. Synapse 25:1-14.
-
(1997)
Synapse
, vol.25
, pp. 1-14
-
-
Laruelle, M.1
Iyer, R.N.2
Al-Tikriti, M.S.3
Zea-Ponce, Y.4
Malison, R.5
Zoghbi, S.S.6
Baldwin, R.M.7
Kung, H.F.8
Charney, D.S.9
Hoffer, P.B.10
Innis, R.B.11
Bradberry, C.W.12
-
25
-
-
0034840454
-
Imaging human mesolimbic dopamine transmission with positron emission tomography: I. Accuracy and precision of D2 receptor parameter measurements in ventral striatum
-
Mawlawi O, Martinez D, Slifstein M, Broft A, Chatterjee R, Hwang DR, Huang Y, Simpson N, Ngo K, Van Heertum R, and Laruelle M (2001) Imaging human mesolimbic dopamine transmission with positron emission tomography: I. Accuracy and precision of D2 receptor parameter measurements in ventral striatum. J Cereb Blood Flow Metab 21:1034-1057.
-
(2001)
J Cereb Blood Flow Metab
, vol.21
, pp. 1034-1057
-
-
Mawlawi, O.1
Martinez, D.2
Slifstein, M.3
Broft, A.4
Chatterjee, R.5
Hwang, D.R.6
Huang, Y.7
Simpson, N.8
Ngo, K.9
Van Heertum, R.10
Laruelle, M.11
-
26
-
-
2342595176
-
In vivo vulnerability to competition by endogenous dopamine: Comparison of the D2 receptor agonist radiotracer (-)-N-[11C]propyl-norapomorphine ([11C]NPA) with the D2 receptor antagonist radiotracer [11C]-raclopride
-
Narendran R, Hwang DR, Slifstein M, Talbot PS, Erritzoe D, Huang Y, Cooper TB, Martinez D, Kegeles LS, Abi-Dargham A, et al. (2004) In vivo vulnerability to competition by endogenous dopamine: comparison of the D2 receptor agonist radiotracer (-)-N-[11C]propyl-norapomorphine ([11C]NPA) with the D2 receptor antagonist radiotracer [11C]-raclopride. Synapse 52:188-208.
-
(2004)
Synapse
, vol.52
, pp. 188-208
-
-
Narendran, R.1
Hwang, D.R.2
Slifstein, M.3
Talbot, P.S.4
Erritzoe, D.5
Huang, Y.6
Cooper, T.B.7
Martinez, D.8
Kegeles, L.S.9
Abi-Dargham, A.10
-
27
-
-
0015856184
-
Aporphines. 8. Total synthesis and pharmacological evaluation of (±)-apomorphine, (±)-apocodeine, (±)-N-n- propylnorapomorphine and (±)-N-npropylnorapocodeine
-
Neumeyer JL, Neustadt BR, Oh KH, Weinhardt KK, Boyce CB, Rosenberg FJ, and Teiger DG (1973) Aporphines. 8. Total synthesis and pharmacological evaluation of (±)-apomorphine, (±)-apocodeine, (±)-N-n-propylnorapomorphine and (±)-N-npropylnorapocodeine. J Med Chem 16:1223-1228.
-
(1973)
J Med Chem
, vol.16
, pp. 1223-1228
-
-
Neumeyer, J.L.1
Neustadt, B.R.2
Oh, K.H.3
Weinhardt, K.K.4
Boyce, C.B.5
Rosenberg, F.J.6
Teiger, D.G.7
-
28
-
-
0024399617
-
Anatomical and affinity state comparisons between dopamine D1 and D2 receptors in the rat central nervous system
-
Richfield EK, Penney JB, and Young AB (1989) Anatomical and affinity state comparisons between dopamine D1 and D2 receptors in the rat central nervous system. Neuroscience 30:767-777.
-
(1989)
Neuroscience
, vol.30
, pp. 767-777
-
-
Richfield, E.K.1
Penney, J.B.2
Young, A.B.3
-
29
-
-
18744362461
-
Mechanisms of inverse agonist action at D2 dopamine receptors
-
Roberts DJ and Strange PG (2005) Mechanisms of inverse agonist action at D2 dopamine receptors. Br J Pharmacol 145:34-42.
-
(2005)
Br J Pharmacol
, vol.145
, pp. 34-42
-
-
Roberts, D.J.1
Strange, P.G.2
-
30
-
-
0026063942
-
11C]diprenorphine and positron emission tomography
-
11C]diprenorphine and positron emission tomography. J Cereb Blood Flow Metab 11:204-219.
-
(1991)
J Cereb Blood Flow Metab
, vol.11
, pp. 204-219
-
-
Sadzot, B.1
Price, J.C.2
Mayberg, H.S.3
Douglass, K.H.4
Dannals, R.F.5
Lever, J.R.6
Ravert, H.T.7
Wilson, A.A.8
Wagner Jr., H.N.9
Feldman, M.A.10
-
31
-
-
84969001783
-
The attraction of proteins for small molecules and ions
-
Scatchard G (1949) The attraction of proteins for small molecules and ions. Ann NY Acad Sci 51:660-672.
-
(1949)
Ann NY Acad Sci
, vol.51
, pp. 660-672
-
-
Scatchard, G.1
-
32
-
-
0036221550
-
Atypical antipsychotics: Mechanism of action
-
Seeman P (2002) Atypical antipsychotics: mechanism of action. Can J Psychiatry 47:27-38.
-
(2002)
Can J Psychiatry
, vol.47
, pp. 27-38
-
-
Seeman, P.1
-
33
-
-
0042421942
-
Anesthetics inhibit high-affinity states of dopamine D2 and other G-linked receptors
-
Seeman P and Kapur S (2003) Anesthetics inhibit high-affinity states of dopamine D2 and other G-linked receptors. Synapse 50:35-40.
-
(2003)
Synapse
, vol.50
, pp. 35-40
-
-
Seeman, P.1
Kapur, S.2
-
34
-
-
0024854498
-
Link between D1 and D2 dopamine receptors is reduced in schizophrenia and Huntington diseased brain
-
Seeman P, Niznik HB, Guan HC, Booth G, and Ulpian C (1989) Link between D1 and D2 dopamine receptors is reduced in schizophrenia and Huntington diseased brain. Proc Natl Acad Sci USA 86:10156-10160.
-
(1989)
Proc Natl Acad Sci USA
, vol.86
, pp. 10156-10160
-
-
Seeman, P.1
Niznik, H.B.2
Guan, H.C.3
Booth, G.4
Ulpian, C.5
-
35
-
-
0037114070
-
Amphetamine-sensitized animals show a marked increase in dopamine D2 high receptors occupied by endogenous dopamine, even in the absence of acute challenges
-
Seeman P, Tallerico T, Ko F, Tenn C, and Kapur S (2002) Amphetamine-sensitized animals show a marked increase in dopamine D2 high receptors occupied by endogenous dopamine, even in the absence of acute challenges. Synapse 46:235-239.
-
(2002)
Synapse
, vol.46
, pp. 235-239
-
-
Seeman, P.1
Tallerico, T.2
Ko, F.3
Tenn, C.4
Kapur, S.5
-
37
-
-
0022271046
-
Dopamine D2 receptor binding sites for agonists. a tetrahedral model
-
Seeman P, Watanabe M, Grigoriadis D, Tedesco JL, George SR, Svensson U, Nilsson JL, and Neumeyer JL (1985) Dopamine D2 receptor binding sites for agonists. A tetrahedral model. Mol Pharmacol 28:391-399.
-
(1985)
Mol Pharmacol
, vol.28
, pp. 391-399
-
-
Seeman, P.1
Watanabe, M.2
Grigoriadis, D.3
Tedesco, J.L.4
George, S.R.5
Svensson, U.6
Nilsson, J.L.7
Neumeyer, J.L.8
-
39
-
-
4344664800
-
In vivo affinity of [18F]fallypride for striatal and extrastriatal dopamine D2 receptors in nonhuman primates
-
Slifstein M, Hwang DR, Huang Y, Guo N, Sudo Y, Narendran R, Talbot P, and Laruelle M (2004a) In vivo affinity of [18F]fallypride for striatal and extrastriatal dopamine D2 receptors in nonhuman primates. Psychopharmacology 175:274-286.
-
(2004)
Psychopharmacology
, vol.175
, pp. 274-286
-
-
Slifstein, M.1
Hwang, D.R.2
Huang, Y.3
Guo, N.4
Sudo, Y.5
Narendran, R.6
Talbot, P.7
Laruelle, M.8
-
40
-
-
4344664800
-
In vivo affinity of [18F]fallypride for striatal and extrastriatal dopamine D2 receptors in nonhuman primates
-
Slifstein M, Hwang DR, Huang Y, Guo NN, Sudo Y, Narendran R, Talbot P, and Laruelle M (2004b) In vivo affinity of [18F]fallypride for striatal and extrastriatal dopamine D2 receptors in nonhuman primates. Psychopharmacology 175:274-286.
-
(2004)
Psychopharmacology
, vol.175
, pp. 274-286
-
-
Slifstein, M.1
Hwang, D.R.2
Huang, Y.3
Guo, N.N.4
Sudo, Y.5
Narendran, R.6
Talbot, P.7
Laruelle, M.8
|