Synthesis of modulators of chloroquine resistance in Plasmodium falciparum, analogues of malagashanine from strychnobrasiline

Tetrahedron

Volumn 60, Issue 25, 2004, Pages 5471-5474

  Trigalo, François ^a   Joyeau, Roger ^a   Pham, Van Cuong ^a   Youté, Jean Jacques ^a   Rasoanaivoa, Philippe ^b   Frappier, François ^a  

^a MUSÉUM NATIONAL D'HISTOIRE NATURELLE   (France)

^b Inst Malgache de Rech Appl   (Madagascar)

Author keywords

Alkaloid; Malagashanine; Reductive amination; Strychnobrasiline; Strychnos myrto des

Indexed keywords

BENZENE; CARBON; CHLOROQUINE;

ACETYLATION; ANTIBIOTIC RESISTANCE; ARTICLE; CHEMICAL BOND; CYCLIZATION; DRUG SYNTHESIS; HYDROGENATION; HYDROLYSIS; METHYLATION; OXIDATION; PLASMODIUM FALCIPARUM; PRIORITY JOURNAL; REDUCTION;

PLASMODIUM FALCIPARUM; STRYCHNOS; STRYCHNOS MYRTOIDES;

EID: 2542447175     PISSN: 00404020     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.tet.2004.04.068     Document Type: Article

References (9)

1. Caira M.R., Rasoanivo P. J. Chem. Crystallogr. 25:1995;725-729
2. Rasoanivo P., Ratsimamanga-Urverg D., Milijaona R., Rafatro H., Ratsimamanga A., Galeffi C., Nicoletti M. Planta Med. 27:1994;2551-2552
3. Trigalo F., Martin M.T., Blond A., Brouard J.P., Herintsoa R., Ramanitrahasimbola D., Frappier F. Tetrahedron. 55:1999;6139-6146
4. Hudlicky M. J. Org. Chem. 45:1980;5377-5378
5. Woodward R.B., Cava M.P., Ollis W.D., Hunger H.U., Daeniker H.U., Schenker K. Tetrahedron. 19:1963;247-288
6. Ingold C.K. Structure and Mechanism in Organic Chemistry. 2nd ed. 1969;Cornell University Press, Ithaca, NY. pp 1129
7. Abdel-Magid A.F., Carson K.G., Harris B.D., Maryanoff C.A., Shah R.D. J. Org. Chem. 61:1996;3849-3862
8. Boit H.G. Chem. Ber. 83:1950;217-226
9. Frappier, F.; Trigalo, A.; Ratsimamanga, S.; Rasoainavo, P. French Patent Application: No. 02/05740, 7 May, 2002.