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Bioorganic and Medicinal Chemistry Letters

Volumn 14, Issue 12, 2004, Pages 3295-3298

The effect of 6-substituted-4′,4″- difluorobenztropines on monoamine transporters and the muscarinic M1 receptor

(4) Grundt, Peter a Kopajtic, Theresa A a Katz, Jonathan L a Newman, Amy Hauck a

a NATIONAL INSTITUTE ON DRUG ABUSE (United States)

Author keywords

Benztropine; Ligand binding; Monoamine transporters; Muscarinic M1 receptor

Indexed keywords

3BETA (4 FLUOROPHENYL) 2BETA TROPANECARBOXYLIC ACID METHYL ESTER; 6ALPHA HYDROXY 4',4'' DIFLUOROBENZTROPINE; 6BETA ACETYL 4',4'' DIFLUOROBENZTROPINE; 6BETA FORMYL 4',4'' DIFLUOROBENZTROPINE; 6BETA HYDROXY 4',4'' DIFLUOROBENZTROPINE; 6BETA PHENYLACETYL 4',4'' DIFLUOROBENZTROPINE; 6BETA PHENYLCARBOXY 4',4'' DIFLUOROBENZTROPINE; 6BETA PHENYLPROPIONYL 4',4'' DIFLUOROBENZTROPINE; 6BETA PROPIONYL 4',4'' DIFLUOROBENZTROPINE; AHN 1 055; BENZATROPINE; BENZENE DERIVATIVE; DOPAMINE TRANSPORTER; MUSCARINIC M1 RECEPTOR; NORADRENALIN TRANSPORTER; PIRENZEPINE; SEROTONIN TRANSPORTER; TRITIUM; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; DRUG EFFECT; DRUG RECEPTOR BINDING; DRUG SCREENING; DRUG SYNTHESIS; NONHUMAN; RACEMIC MIXTURE; RAT; SUBSTITUTION REACTION;

BENZTROPINE; DOPAMINE PLASMA MEMBRANE TRANSPORT PROTEINS; MEMBRANE GLYCOPROTEINS; MEMBRANE TRANSPORT PROTEINS; NERVE TISSUE PROTEINS; NOREPINEPHRINE PLASMA MEMBRANE TRANSPORT PROTEINS; PROTEIN BINDING; RECEPTOR, MUSCARINIC M1; SEROTONIN PLASMA MEMBRANE TRANSPORT PROTEINS; SYMPORTERS;

ANIMALIA;

EID: 2442501261 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/j.bmcl.2004.03.075 Document Type: Article

Times cited : (9)

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