-
4
-
-
0032518922
-
-
L. Wilkström, C. Johansson, C. Saltó, C. Barlow, A.G. Barrow, F. Baas, D. Forrest, P. Thorén, and B. Vennström EMBO J. 17 1998 455
-
(1998)
EMBO J.
, vol.17
, pp. 455
-
-
Wilkström, L.1
Johansson, C.2
Saltó, C.3
Barlow, C.4
Barrow, A.G.5
Baas, F.6
Forrest, D.7
Thorén, P.8
Vennström, B.9
-
5
-
-
17444449237
-
-
C. Johansson, S. Göthe, D. Forrest, B. Vennström, and P. Thorén Am. J. Physiol. 276 1999 H2006
-
(1999)
Am. J. Physiol.
, vol.276
, pp. 2006
-
-
Johansson, C.1
Göthe, S.2
Forrest, D.3
Vennström, B.4
Thorén, P.5
-
6
-
-
17744387900
-
-
S.U. Trost, E. Swanson, B. Gloss, D.B. Wang-Iverson, H. Zhang, T. Volodarsky, G.J. Grover, J.D. Baxter, G. Chiellini, T.S. Scanlan, W.H. Dillmann, and H. Wolfgang Endocrinology 141 2000 3057
-
(2000)
Endocrinology
, vol.141
, pp. 3057
-
-
Trost, S.U.1
Swanson, E.2
Gloss, B.3
Wang-Iverson, D.B.4
Zhang, H.5
Volodarsky, T.6
Grover, G.J.7
Baxter, J.D.8
Chiellini, G.9
Scanlan, T.S.10
Dillmann, W.H.11
Wolfgang, H.12
-
7
-
-
0042734823
-
-
G.J. Grover, K. Mellström, L. Ye, J. Malm, Y.-L. Li, L.-G. Bladh, P.G. Sleph, M.A. Smith, R. George, B. Vennström, K. Mookhtiar, R. Horvath, J. Speelman, D. Egan, and J.D. Baxter Proc. Natl. Acad. Sci. U.S.A. 100 2003 10067
-
(2003)
Proc. Natl. Acad. Sci. U.S.A.
, vol.100
, pp. 10067
-
-
Grover, G.J.1
Mellström, K.2
Ye, L.3
Malm, J.4
Li, Y.-L.5
Bladh, L.-G.6
Sleph, P.G.7
Smith, M.A.8
George, R.9
Vennström, B.10
Mookhtiar, K.11
Horvath, R.12
Speelman, J.13
Egan, D.14
Baxter, J.D.15
-
8
-
-
0029643769
-
-
R.L. Wagner, J.W. Apriletti, M.E. McGrath, B.L. West, J.D. Baxter, and R.J. Fletterick Nature 378 1995 690
-
(1995)
Nature
, vol.378
, pp. 690
-
-
Wagner, R.L.1
Apriletti, J.W.2
McGrath, M.E.3
West, B.L.4
Baxter, J.D.5
Fletterick, R.J.6
-
9
-
-
0032052809
-
-
R.C.J. Ribeiro, J.W. Apriletti, R.L. Wagner, F. Feng, P.J. Kiushner, S. Nilsson, T.S. Scanlan, B.L. West, R.J. Fletterick, and J.D.J. Baxter Steroid Biochem. Mol. Biol. 65 1998 133
-
(1998)
Steroid Biochem. Mol. Biol.
, vol.65
, pp. 133
-
-
Ribeiro, R.C.J.1
Apriletti, J.W.2
Wagner, R.L.3
Feng, F.4
Kiushner, P.J.5
Nilsson, S.6
Scanlan, T.S.7
West, B.L.8
Fletterick, R.J.9
Baxter, J.D.J.10
-
13
-
-
0037464499
-
-
L. Ye, Y.-L. Li, K. Mellström, L.-G. Bladh, K. Koehler, N. Garg, A.M. Garcia Collazo, C. Litten, B. Husman, K. Persson, J. Ljunggren, G. Grover, P.G. Sleph, R. George, and J. Malm J. Med. Chem. 46 2003 1580
-
(2003)
J. Med. Chem.
, vol.46
, pp. 1580
-
-
Ye, L.1
Li, Y.-L.2
Mellström, K.3
Bladh, L.-G.4
Koehler, K.5
Garg, N.6
Garcia Collazo, A.M.7
Litten, C.8
Husman, B.9
Persson, K.10
Ljunggren, J.11
Grover, G.12
Sleph, P.G.13
George, R.14
Malm, J.15
-
14
-
-
0037330393
-
-
R.L. Dow, S.R. Schneider, E.S. Paight, R.F. Hank, P. Chaing, P. Cornelius, E. Lee, W.P. Newsome, A.G. Swick, J. Spitzer, D.E. Hargrove, T.A. Patterson, J. Pandit, B.A. Chrunyk, P.K. LeMotte, D.E. Danley, M.H. Rosner, M.J. Ammirati, S.P. Simones, G.K. Schulte, B.F. Tate, and P. DaSilva-Jardine Bioorg. Med. Chem. Lett. 13 2003 379
-
(2003)
Bioorg. Med. Chem. Lett.
, vol.13
, pp. 379
-
-
Dow, R.L.1
Schneider, S.R.2
Paight, E.S.3
Hank, R.F.4
Chaing, P.5
Cornelius, P.6
Lee, E.7
Newsome, W.P.8
Swick, A.G.9
Spitzer, J.10
Hargrove, D.E.11
Patterson, T.A.12
Pandit, J.13
Chrunyk, B.A.14
Lemotte, P.K.15
Danley, D.E.16
Rosner, M.H.17
Ammirati, M.J.18
Simones, S.P.19
Schulte, G.K.20
Tate, B.F.21
Dasilva-Jardine, P.22
more..
-
15
-
-
24344435819
-
-
S. Borngraeber, M.-J. Budny, G. Chiellini, S.T. Cunha-Lima, M. Togashi, P. Webb, J.D. Baxter, T.S. Scanlan, and R.J. Fletterick Proc. Natl. Acad. Sci. U.S.A. 2003 100
-
(2003)
Proc. Natl. Acad. Sci. U.S.A.
, pp. 100
-
-
Borngraeber, S.1
Budny, M.-J.2
Chiellini, G.3
Cunha-Lima, S.T.4
Togashi, M.5
Webb, P.6
Baxter, J.D.7
Scanlan, T.S.8
Fletterick, R.J.9
-
16
-
-
2942596255
-
-
J.J. Hangeland, A.M. Doweyko, T. Dejneka, T.J. Friends, P. Devasthale, K. Mellström, J. Sandberg, M. Grynfarb, J.S. Sack, H. Einspahr, M. Färnegårdh, B. Husma, J. Ljunggren, K. Koehler, C. Sheppard, J. Malm, and D.E. Ryono Bioorg. Med. Chem. Lett. 14 2004 3549
-
(2004)
Bioorg. Med. Chem. Lett.
, vol.14
, pp. 3549
-
-
Hangeland, J.J.1
Doweyko, A.M.2
Dejneka, T.3
Friends, T.J.4
Devasthale, P.5
Mellström, K.6
Sandberg, J.7
Grynfarb, M.8
Sack, J.S.9
Einspahr, H.10
Färnegårdh, M.11
Husma, B.12
Ljunggren, J.13
Koehler, K.14
Sheppard, C.15
Malm, J.16
Ryono, D.E.17
-
17
-
-
0016395135
-
-
The description of the conformational relationship between the two phenyl rings has been adapted from: V. Cody J. Am. Chem. Soc. 96 1974 6720
-
(1974)
J. Am. Chem. Soc.
, vol.96
, pp. 6720
-
-
Cody, V.1
-
18
-
-
0032101890
-
-
G. Chiellini, J.W. Apriletti, H.A.I. Yoshihara, J.D. Baxter, R.C. Riberio, and T.S. Scanlan Chem. Biol. 5 1998 299
-
(1998)
Chem. Biol.
, vol.5
, pp. 299
-
-
Chiellini, G.1
Apriletti, J.W.2
Yoshihara, H.A.I.3
Baxter, J.D.4
Riberio, R.C.5
Scanlan, T.S.6
-
21
-
-
24344479055
-
-
note
-
Compounds 5 and 6 were synthesized using procedures reported in Refs. 8 and 9c.
-
-
-
-
23
-
-
24344481177
-
-
note
-
8,17.
-
-
-
-
24
-
-
0037203995
-
-
B. Carlsson, B.N. Singh, M. Temciuc, S. Nilsson, Y.-L. Li, C. Mellin, and J. Malm J. Med. Chem. 45 2002 623
-
(2002)
J. Med. Chem.
, vol.45
, pp. 623
-
-
Carlsson, B.1
Singh, B.N.2
Temciuc, M.3
Nilsson, S.4
Li, Y.-L.5
Mellin, C.6
Malm, J.7
-
25
-
-
0025881963
-
-
T. Barkhem, B. Carlsson, J. Simons, B. Moeller, A. Berkenstam, J.-Å. Gustafsson, and S. Nilsson J. Steroid Biochem. Mol. Biol. 38 1991 667
-
(1991)
J. Steroid Biochem. Mol. Biol.
, vol.38
, pp. 667
-
-
Barkhem, T.1
Carlsson, B.2
Simons, J.3
Moeller, B.4
Berkenstam, A.5
Gustafsson, J.-Å.6
Nilsson, S.7
-
26
-
-
0029044699
-
-
N. Yokoyama, G.N. Walker, A.J. Main, J.L. Stanton, M.M. Morrissey, C. Boehm, A. Engle, A.D. Neubert, J.M. Wasvary, Z.F. Stephan, and R.E. Steele J. Med. Chem. 38 1995 695
-
(1995)
J. Med. Chem.
, vol.38
, pp. 695
-
-
Yokoyama, N.1
Walker, G.N.2
Main, A.J.3
Stanton, J.L.4
Morrissey, M.M.5
Boehm, C.6
Engle, A.7
Neubert, A.D.8
Wasvary, J.M.9
Stephan, Z.F.10
Steele, R.E.11
-
27
-
-
0002247632
-
-
T. Harada, T. Yoshida, A. Inoue, M. Takeuchi, and A. Oku Synlett 1995 283
-
(1995)
Synlett
, pp. 283
-
-
Harada, T.1
Yoshida, T.2
Inoue, A.3
Takeuchi, M.4
Oku, A.5
-
32
-
-
24344473622
-
-
Colin McMartin, Thistlesoft, Colebrook, CT.
-
Flo/QXP molecular modeling program; Colin McMartin, Thistlesoft, Colebrook, CT.
-
Flo/QXP Molecular Modeling Program
-
-
-
33
-
-
24344447673
-
-
note
-
Semi-empirical molecular orbital calculations carried out using SAM1D within the AMPAC package as implemented within Sybyl Version 7.0 (Tripos, Inc., St. Louis, MO).
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