QSAR study on thiazole and thiadiazole analogues as antagonists for the adenosine A1 and A3 receptors

Bioorganic and Medicinal Chemistry

Volumn 13, Issue 18, 2005, Pages 5330-5337

  Borghini, Alice ^a   Pietra, Daniele ^a   Domenichelli, Patrick ^a   Bianucci, Anna Maria ^a  

^a UNIVERSITY OF PISA   (Italy)

Author keywords

Adenosine receptors; Model validation; QSAR; Thiazole and thiadiazole analogues

Indexed keywords

ADENOSINE A1 RECEPTOR ANTAGONIST; ADENOSINE A3 RECEPTOR ANTAGONIST; LIGAND; THIADIAZOLE DERIVATIVE; THIAZOLE;

ACCURACY; ARTICLE; CHEMICAL MODEL; COMPUTER PROGRAM; CORRELATION ANALYSIS; DATA BASE; DRUG STRUCTURE; DRUG TARGETING; QUANTITATIVE STRUCTURE ACTIVITY RELATION; RELIABILITY; STRUCTURE ANALYSIS;

COMPUTER SIMULATION; LIGANDS; MODELS, CHEMICAL; QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIP; RECEPTOR, ADENOSINE A1; RECEPTOR, ADENOSINE A3; THIADIAZOLES; THIAZOLES;

EID: 23644458559     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2005.05.041     Document Type: Article

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