Synthesis of 4-substituted and 3,4-disubstituted indazole derivatives by palladium-mediated cross-coupling reactions

Tetrahedron Letters

Volumn 46, Issue 36, 2005, Pages 6163-6167

  El Kazzouli, Saïd ^a,b   Bouissane, Latifa ^a,b   Khouili, Mostafa ^b   Guillaumet, Gérald ^a  

^a UNIVERSITÉ D'ORLÉANS   (France)

^b FACULTÉ DES SCIENCES ET TECHNIQUES GUÉLIZ   (Morocco)

Author keywords

3 Bromo 4 iodoindazole; Indazoles; Palladium

Indexed keywords

INDAZOLE DERIVATIVE; PALLADIUM; VINYL DERIVATIVE;

ALKYLATION; ARTICLE; DEHALOGENATION; DRUG SYNTHESIS; HECK REACTION; PROTON NUCLEAR MAGNETIC RESONANCE; SONOGASHIRA REACTION; STILLE REACTION; SUZUKI REACTION;

EID: 23244451883     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.tetlet.2005.06.080     Document Type: Article

References (22)

1. V. Collot, P. Dallemagne, P.R. Bovy, and S. Rault Tetrahedron 55 1999 6917
2. J.-H. Sun, C.A. Teleha, J.-S. Yan, J.D. Rodgers, and D.A. Nugiel J. Org. Chem. 62 1997 5627
3. D.G. Batt, J.J. Petraitis, G.C. Houghton, D.P. Modi, G.A. Cain, M.H. Corjay, S.A. Mousa, P.J. Bouchard, M.S. Forsythe, P.P. Harlow, F.A. Barbera, S.M. Spitz, R.R. Wexler, and P.K. Jadhav J. Med. Chem. 43 2000 41
4. A. Amautu, V. Collot, J.C. Ros, C. Alayrac, B. Witulski, and S. Rault Tetrahedron Lett. 43 2002 2695
5. V. Collot, P.R. Bovy, and S. Rault Tetrahedron Lett. 41 2000 9053
6. V. Collot, D. Varlet, and S. Rault Tetrahedron Lett. 41 2000 4363
7. D.W. Gordon Synlett 1998 1065
8. W.M. Welch, C.E. Hanau, and W.M. Whalen Synthesis 1992 937
9. L. Bouissane, S. El Kazzouli, J.-M. Leger, C. Jarry, E.M. Rakib, M. Khouili, and G. Guillaumet Tetrahedron 61 2005 8218
10. Bouissane, L.; El Kazzouli, S.; Léonce, S.; Pfeiffer, B.; Rakib, E. M.; Khouili, M.; Guillaumet, G. Bioorg. Med. Chem., submitted for publication.
11. E. Noelting Berichte 37 1904 2556
12. +].
13. B.I. Alo, A. Kandil, P.A. Patil, M.J. Sharp, M.A. Siddiqui, and V. Snieckus J. Org. Chem. 56 1991 3763
14. +].
15. B. Ruhland, A. Bombrun, and M.A. Gallop J. Org. Chem. 62 1997 7820
16. +].
17. V. Farina, S. Kapadia, B. Krishnan, C. Wang, and L.S. Liebeskind J. Org. Chem. 59 1994 5905
18. +].
19. +].
20. +].
21. During the submission of this article, similar results were published. B. Witulski, J.R. Azcon, C. Alayrac, A. Arnautu, V. Collot, and S. Rault Synthesis 2005 771
22. +].