Rheological, mucoadhesive and release properties of Pluronic F-127 gel and Pluronic F-127/polycarbophil mixed gel systems

Pharmazie

Volumn 60, Issue 7, 2005, Pages 518-523

  Tirnaksiz, Figen ^a,b   Robinson, J R ^a  

^a UNIVERSITY OF WISCONSIN MADISON   (United States)

^b GAZI UNIVERSITY   (Turkey)

Author keywords

[No Author keywords available]

Indexed keywords

CARBOXYLIC ACID; MANNITOL; NOVEON; POLOXAMER; POLYCARBOPHIL;

ADHESION; AQUEOUS SOLUTION; ARTICLE; CONCENTRATION (PARAMETERS); CONTROLLED DRUG RELEASE; DIFFUSION; FLOW KINETICS; FORCE; GEL; HEAT SENSITIVITY; MOLECULAR INTERACTION; TEMPERATURE DEPENDENCE; VISCOSITY;

ACRYLIC RESINS; ADHESIVENESS; ANIMALS; GASTRIC MUCOSA; GELS; MANNITOL; MUCOUS MEMBRANE; POLOXAMER; RABBITS; RHEOLOGY; TEMPERATURE; VISCOSITY;

EID: 22644443288     PISSN: 00317144     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (35)

1. Attwood D, Collett JH, Tait CJ (1985) The micellar properties of the poly (oxyethylene) - poly (oxypropylene) copolymer Pluronic F127 in water and electrolyte solution. Int J Pharm 26: 25-33.
2. BASF Performance Chemicals (1996), Technical data on Pluronic and Tetronic Surfactants, Mount Olive, New Jersey.
3. Bhardwaj R, Blanchard J (1996) Controlled release delivery system for the α-MSH analog melanotan-I using poloxamer 407. J Pharm Sci 85: 915-919.
4. Chen-Chow P-C, Frank SG (1981) In vitro release of lidocaine from Pluronic F-127 gels. Int J Pharm 8: 89-99.
5. Chi SC, Jun HW (1990) Anti-inflammatory activity of ketoprofen gel on carrageenan-induced paw edema in rats. J Pharm Sci 79: 974-977.
6. Chi SC, Jun HW (1991) Release rates of ketoprofen from poloxamer gels in a membraneless diffusion cell. J Pharm Sci 80: 280-283.
7. Ch'ng HS, Park H, Kelly P, Robinson JR (1985) Bioadhesive polymers as platforms for oral controlled drug delivery II: Synthesis and evaluation of some swelling, water-insoluble bioadhesive polymers. J Pharm Sci 74: 399-405.
8. Choi H-g, Jung J-h, Ryu J-m, Yoon S-j, Oh Y-k, Kim C-k (1998) Development of in situ-gelling and mucoadhesive acetaminophen liquid suppository. Int J Pharm 165: 33-44.
9. Cole ML, Whateley TL (1996) Interaction of nonionic block copolymeric (poloxamer) surfactants with poly(acrylic acid), studied by photon correlation spectroscopy. J Colloid Interface Sci 180: 421-427.
10. Collett JH, Tait CJ, Atwood D, Sharma HL, Smith AM (1985) In vivo evaluation of poloxamer gels as controlled release systems using gama scintigraphy. Proceed Intern Symp Control Rel Bioact Mater 12: 28-29.
11. DiBiase MD, Rhodes CT (1996) Formulation and evaluation of epidermal growth factor in Pluronic F-127 gel. Drug Dev Ind Pharm 22: 823-831.
12. Fults KA, Johnston TP (1990) Sustained release of urease from a poloxamer gel matrix. J Parenter Sci Technol 44: 58-65.
13. Guzman M, Aberturas MR, Garcia F, Molpeceres J (1994) Gelatine gels and polyoxyethylene-polyoxypropylene gels: Comparative study of their properties. Drug Dev Ind Pharm 20: 2041-2048.
14. Johnston TP, Punjabi MA (1990) Froelich CJ Sustained delivery of interleukin-2 from a poloxamer 407 gel matrix following intraperitoneal injection in mice. Pharm Res 9: 425-434.
15. Johnson TP, Miller SC (1989) Inulin disposition following intramuscular administration of an inulin/poloxamer gel matrix. J Parenter Sci Technol 43: 279-286.
16. Juhasz J, Lenaerts V, Raymond P, Ong H (1989) Diffusion of rat natriuretic factor in thermoreversible poloxamer gels. Biomaterials 10: 265-268.
17. Juhasz J, Pimienta C, Lenaerts V (1991) Adhesion of poloxamer 407 formulations on dog ileal segments in vitro. Eur J Pharm Biopharm 37: 262-265.
18. Katakam M, Ravis WR, Banga AK (1997) Controlled release of human growth hormone in rats following parenteral administration of poloxamer gels. J Contr Rel 49: 21-26.
19. Lenaerts V, Triqueneaux C, Quarton M, Rieg-Falson F, Couvreur P (1987) Temperature-dependent rheological behavior of Pluronic F-127 aqueous solutions. Int J Pharm 39: 121-127.
20. Lu G, Jun HW (1998) Diffusion studies of methotrexate in Carbopol and poloxamer gels. Int J Pharm 160: 1-9.
21. Malmsten M, Lindman B (1993) Effects of homopolymers on the gel formation in aqueous block copolymer solutions. Macromolecules 26: 1282-1286.
22. Miller S, Donovan MD (1982) Effect of poloxamer 407 gel on the miotic activity of pilocarpine nitrate in rabbits. Int J Pharm 12: 147-152.
23. Miller SC, Drabik BR (1984) Rheological properties of poloxamer vehicles. Int J Pharm 18: 269-276.
24. Miyazaki S, Takeuchi S, Yokouchi C, Takada M (1984) Pluronic F-127 gels as a vehicle for topical administration of anticancer agents. Chem Pharm Bull 32: 4205-4208.
25. Moore T, Croy S, Mallapragada S, Pandit N (2000) Experimental investigation and mathematical modeling of Pluronic F127 gel dissolution: drug release in stirred systems. J Cont Rel 67: 91-202.
26. Park H, Robinson JR (1985) Physicochemical properties of water insoluble polymers important to mucin/epithelial adhesion. J Cont Rel 2: 47-57.
27. Saettone MF, Giannaccini B, Delmonte G, Campigli V, Tota G, Marca FL (1988) Solubilization of tropicamide by poloxamers: Physicochemical data and activity data in rabbits and humans. Int J Pharm 43: 67-76.
28. Schmolka IR (1967) Application of Pluronic® polyols in the cosmetic industry. Am Perfumer Cosmet 82: 25-30.
29. Schmolka IR (1972) Artificial skin I. preparation and properties of Pluronic F-127 gels for treatment of burns. J Biomed Mater Res 6: 571-582.
30. Schmolka IR (1991) A comparison of block copolymer surfactant gels. J Am Oil Chem Soc 68: 206-209.
31. Suh H, Jun H (1996) Physicochemical and release studies of naproxen in poloxamer gels. Int J Pharm 129: 13-20.
32. Tung IC (1994) Rheological behavior of poloxamer 407 aqueous solutions during sol-gel and dehydration processes. Int J Pharm 107: 85-90.
33. Vadnere M, Amidon G, Lindenbaum S, Haslam JL (1984) Thermodynamic studies on the gel-sol transition of some Pluronic polyols. Int J Pharm 22: 207-218.
34. Veyries ML, Couarraze G, Geiger S, Agnely F, Massias L, Kunzli B, Faurisson F, Rouveix B (1999) Controlled release of vancomycin from poloxamer 407 gels. Int J Pharm 192: 183-193.
35. Wang PL, Johnston TP (1995) Sustained release interleukin-2 following intramuscular injection in rats. Int J Pharm 113: 73-81.