Identification of a region of the ileal-type sodium/bile acid cotransporter interacting with a competitive bile acid transport inhibitor

Biochemistry

Volumn 41, Issue 50, 2002, Pages 14916-14924

  Hallen S ^a,b   Bjorquist A ^b   Ostlund Lindqvist A M ^b   Sachs, G ^a,c  

^a VETERANS AFFAIRS MEDICAL CENTER   (United States)

^b ASTRAZENECA R AND D   (Sweden)

^c VA GREATER LOS ANGELES HEALTHCARE SYSTEM   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ABSORPTION; AMINO ACIDS; CHOLESTEROL; DRUG PRODUCTS; HYDROPHOBICITY; PATIENT TREATMENT; SODIUM;

DRUG INTERVENTION;

BIOCHEMISTRY;

2164 U90; 3 BUTYL 3 ETHYL 5 PHENYL 2,3,4,5 TETRAHYDRO 1,4 BENZOTHIAZEPINE 1,1 DIOXIDE; AMINO ACID; BENZOTHIAZEPINE DERIVATIVE; BILE ACID; COTRANSPORTER; CYSTEINE; ISOLEUCINE; METHANETHIOSULFONATE; SERINE; SODIUM BILE ACID COTRANSPORTER; SULFONIC ACID DERIVATIVE; UNCLASSIFIED DRUG; VALINE;

ALKYLATION; AMINO ACID SUBSTITUTION; ANIMAL CELL; ARTICLE; CARBOXY TERMINAL SEQUENCE; CHOLESTEROL BLOOD LEVEL; DRUG BINDING; DRUG PROTEIN BINDING; DRUG STRUCTURE; HAMSTER; HUMAN; HUMAN CELL; HYDROPHOBICITY; ILEUM; MOUSE; NONHUMAN; PRIORITY JOURNAL; PROTEIN DOMAIN; RAT; SPECIES DIFFERENTIATION;

AMINO ACID SEQUENCE; ANIMALS; BILE ACIDS AND SALTS; BINDING, COMPETITIVE; BIOLOGICAL TRANSPORT, ACTIVE; CARRIER PROTEINS; CELL LINE; CHO CELLS; CRICETINAE; CYSTEINE; HUMANS; HYDROXYSTEROID DEHYDROGENASES; ILEUM; KINETICS; MEMBRANE GLYCOPROTEINS; MESYLATES; MICE; MOLECULAR SEQUENCE DATA; MUTAGENESIS, SITE-DIRECTED; ORGANIC ANION TRANSPORTERS, SODIUM-DEPENDENT; PEPTIDE FRAGMENTS; RATS; RECOMBINANT FUSION PROTEINS; SEQUENCE ALIGNMENT; SERINE; SYMPORTERS; TAUROCHOLIC ACID; THIAZEPINES; THREONINE; VALINE;

ANIMALIA; CRICETINAE;

EID: 2242424505     PISSN: 00062960     EISSN: None     Source Type: Journal    
DOI: 10.1021/bi0205404     Document Type: Article

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