Pharmacological characterization of indisetron hydrochloride, as a novel 5-HT 3 receptor antagonist

Japanese Pharmacology and Therapeutics

Volumn 32, Issue 11, 2004, Pages 789-797

  Taniguchi, Sugure ^a   Watanabe, Fumiko ^a   Hagihara, Koichiro ^a  

^a KYORIN PHARMACEUTICAL CO LTD   (Japan)

Author keywords

5 HT 4 receptor antagonist; 5 HT 3 receptor antagonist; Guinea pig; Indisetron hydrochloride; Rat

Indexed keywords

2 METHYLSEROTONIN; 3 (5 METHYL 1H IMIDAZOL 4 YL) 1 (1 METHYL 1H INDOL 3 YL) 1 PROPANONE; 5 METHYLTRYPTAMINE; 8 CHLORO 2,3,4,5 TETRAHYDRO 3 METHYL 5 PHENYL 1H 3 BENZAZEPIN 7 OL HYDROGEN MALEATE; ALPHA 1 ADRENERGIC RECEPTOR; ALPHA 2 ADRENERGIC RECEPTOR; AZASETRON; BENZODIAZEPINE RECEPTOR; BETA ADRENERGIC RECEPTOR; BUTACLAMOL; CLONIDINE; DIAZEPAM; DOPAMINE 1 RECEPTOR; DOPAMINE 2 RECEPTOR; FLUNITRAZEPAM; GRANISETRON; INDISETRON; KETANSERIN; ONDANSETRON; PHENTOLAMINE; PRAZOSIN; PROPRANOLOL; RACLOPRIDE; SEROTONIN; SEROTONIN 1 RECEPTOR; SEROTONIN 2 RECEPTOR; SEROTONIN 3 ANTAGONIST; SEROTONIN 3 RECEPTOR; SEROTONIN 4 RECEPTOR; TROPISETRON;

ARTICLE; BINDING AFFINITY; BRADYCARDIA; BRAIN CORTEX; DRUG POTENCY; DRUG RECEPTOR BINDING; ESOPHAGUS MUSCLE; GUINEA PIG; IC 50; INTESTINE CONTRACTION; MUSCLE RELAXATION; NONHUMAN; RAT;

EID: 21044454109     PISSN: 03863603     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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