Evaluation of rapidly disintegrating tablets manufactured by phase transition of sugar alcohols

Journal of Controlled Release

Volumn 105, Issue 1-2, 2005, Pages 16-22

  Kuno, Yoshio ^a   Kojima, Masazumi ^a   Ando, Shuichi ^a   Nakagami, Hiroaki ^a  

^a DAIICHI SANKYO CO   (Japan)

Author keywords

Phase transition; Rapidly disintegrating tablets; Sugar alcohol

Indexed keywords

CRYSTALLIZATION; HEATING; MELTING; PHASE TRANSITIONS; PORE SIZE; SUGARS;

ERYTHRITOL; PHYSICOCHEMICAL PROPERTIES; RAPIDLY DISINTEGRATING (RD) TABLETS; XYLITOL;

DRUG PRODUCTS;

ERYTHRITOL; SUGAR ALCOHOL; XYLITOL;

ARTICLE; CHEMICAL COMPOSITION; DRUG MANUFACTURE; EVALUATION; HARDNESS; HEATING; MELTING POINT; PHASE TRANSITION; PHYSICAL CHEMISTRY; POWDER; PRIORITY JOURNAL; STORAGE; TABLET; TECHNIQUE;

DELAYED-ACTION PREPARATIONS; DRUG COMPOUNDING; EXCIPIENTS; HARDNESS; POROSITY; POWDERS; SOLUBILITY; SUGAR ALCOHOLS; TABLETS;

EID: 20444425824     PISSN: 01683659     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.jconrel.2005.01.018     Document Type: Article

References (21)

1. Y. Kuno, M. Kojima, S. Ando, and H. Nakagami Preparation of interoral rapid disintegrating tablets by a novel method involving phase transition of sugar alcohol Controlled Release Society 30th Annual Meeting ProceedingsGlasgow, Scotland, United Kingdom, July 19-23, 2003 2003 #649
2. A. Watanabe, T. Hanada, and M. Sugihara New oral dosage form for the elderly-rapid dissolving tablet in mouth without addition of water Yakuzaigaku 54 1998 103 110
3. Y. Jin, H. Ohkuma, H. Wang, H. Natsume, K. Sugibayashi, and Y. Morimoto Fast-disintegration oral tablets having sustained release property Yakuzaigaku 122 11 2002 989 994
4. Y. Bi, H. Sunada, Y. Yonezawa, K. Danjo, A. Otsuka, and K. Iida Preparation and evaluation of a compressed tablet rapidly disintegrating in the oral cavity Chem. Pharm. Bull. 44 11 1996 2121 2127
5. Y. Bi, H. Sunada, and Y. Yonezawa Rapidly disintegrating tablets prepared by the wet compression method: mechanism and optimization J. Pharm. Sci. 88 10 1999 1004 1010
6. Y. Bi, H. Sunada, Y. Yonezawa, and K. Danjo Evaluation of rapidly disintegrating tablets prepared by a direct compression method Drug Dev. Ind. Pharm. 25 5 1999 571 581
7. H. Sunada, and Y. Bi Preparation, evaluation and optimization of rapidly disintegrating tablets Powder Technol. 122 2002 188 198
8. M. Sugimoto, K. Matsubara, Y. Koida, and M. Kobayashi The preparation of rapidly disintegrating tablets in the mouth Pharm. Dev. Technol. 6 4 2001 487 493
9. K. Masaki Orally disintegrating famotidine tablet The Collected Papers of the 22nd Conference on Pharmaceutical Technology 1997 (July) Academy of Pharmaceutical Science and Technology Japan 79 84
10. H. Seager Drug-delivery products and the zydis fast-dissolving dosage form J. Pharm. Pharmacol. 50 1998 375 382
11. Y. Tsushima Tablets that are easily to be taken-dosage form developed for elderly patients Farumashia 33 10 1997 1119 1123
12. T. Shimizu, Y. Nakano, S. Morimoto, T. Tabata, N. Hmaguchi, and Y. Igari Formulation study for lansoprazole fast-disintegrating tablet: I. Effect of compression on dissolution behavior Chem. Pharm. Bull. 51 9 2003 942 947
13. T. Shimizu, N. Kameoka, H. Iki, T. Tabata, N. Hamaguchi, and Y. Igari Formulation study for lansoprazole fast-disintegrating tablet: II. Effect of triethyl citrate on the quality of the products Chem. Pharm. Bull. 51 9 2003 1029 1035
14. T. Mizumoto, Y. Masuda, M. Fukui, Intraorally soluble compressed molding and process for producing the same, PCT patent, PCT/JP95/00102, December 4, 1996.
15. T. Shimizu, M. Shugaya, Y. Nakao, Rapidly disintegrating solid dosage form, JP patent, 2000-103731, April 11, 2000.
16. K. Nishimura, H. Aibara, Y. Nakagawa, S. Aoki, Orally dissolving tablet, JP patent, 2000-273038, October 3, 2000.
17. M.J. Anne Relation between breaking force and pore structure of lactose, glucose and mannitol tablets Int. J. Pharm. 127 1996 95 102
18. S. Mattsson, and C. Nystrom The use of mercury porosimetry in assessing the effect of different binders on the pore structure and bonding properties of tablets Eur. J. Pharm. Biopharm. 52 2001 237 247
19. C. Nystrom, and P.G. Karehill Studies on direct compression of tablets: XVI. The use of surface area measurements for the evaluation of bonding surface area in compressed powders Powder Technol. 47 1986 201 209
20. C. Nystrom, G. Alderborn, M. Duberg, and P.G. Karehill Bonding surface area and bonding mechanism-two important factors for the understanding of powder compactabillity Drug Dev. Ind. Pharm. 19 17 & 18 1993 2143 2196
21. E.W. Washburn The dynamics of capillary flow Phys. Rev. 17 1921 273 281