Synthesis of irreversibly binding bicalutamide analogs for imaging studies

Tetrahedron Letters

Volumn 46, Issue 28, 2005, Pages 4821-4823

  Nair, Vipin A ^a   Mustafa, Suni M ^a   Mohler, Michael L ^a   Yang, Jun ^b   Kirkovsky, Leonid I ^a   Dalton, James T ^b   Miller, Duane D ^a  

^a UNIVERSITY OF TENNESSEE HEALTH SCIENCE CENTER   (United States)

^b OHIO STATE UNIVERSITY   (United States)

Author keywords

Androgen; Bicalutamide; Iodine; Radioactive; Receptor

Indexed keywords

ANDROGEN RECEPTOR; BICALUTAMIDE;

ARTICLE; COLUMN CHROMATOGRAPHY; DRUG SYNTHESIS; IMAGING; RECEPTOR BINDING; RING OPENING; ROOM TEMPERATURE;

EID: 20444419774     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.tetlet.2005.04.143     Document Type: Article

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