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Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 13, 2005, Pages 3257-3262

Design, synthesis, and biological evaluation of novel 4-hydroxypyrone derivatives as HIV-1 protease inhibitors

(4) Sun, Chun Lai a Pang, Rui Fang a Zhang, Hang a Yang, Ming a

a PEKING UNIVERSITY (China)

Author keywords

4 Hydroxypyrone; Antiviral activity; Protease inhibitor

Indexed keywords

PROTEINASE INHIBITOR; PYRONE DERIVATIVE;

ANTIVIRAL ACTIVITY; ARTICLE; CONTROLLED STUDY; DRUG ACTIVITY; DRUG DESIGN; DRUG SYNTHESIS; HUMAN; HUMAN CELL; HUMAN IMMUNODEFICIENCY VIRUS 1; IC 50; SIMIAN IMMUNODEFICIENCY VIRUS;

CELL LINE; CELL SURVIVAL; HIV PROTEASE INHIBITORS; HUMANS; INHIBITORY CONCENTRATION 50; MODELS, MOLECULAR; PYRONES; SIMIAN IMMUNODEFICIENCY VIRUS; STRUCTURE-ACTIVITY RELATIONSHIP;

HUMAN IMMUNODEFICIENCY VIRUS 1; SIMIAN IMMUNODEFICIENCY VIRUS;

EID: 20444416295 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/j.bmcl.2005.04.057 Document Type: Article

Times cited : (15)

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