Synthesis and structure-activity relationships of isoxazole carboxamides as growth hormone secretagogue receptor antagonists

Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 4, 2005, Pages 1201-1204

  Xin, Zhili ^a   Zhao, Hongyu ^a   Serby, Michael D ^a   Liu, Bo ^a   Schaefer, Verlyn G ^a   Falls, Douglas H ^a   Kaszubska, Wiweka ^a   Colins, Christine A ^a   Sham, Hing L ^a   Liu, Gang ^a  

^a ABBOTT LABORATORIES   (United States)

Author keywords

Growth hormone secretagogue receptor antagonist

Indexed keywords

GHRELIN; GROWTH HORMONE SECRETAGOGUE RECEPTOR; GROWTH HORMONE SECRETAGOGUE RECEPTOR ANTAGONIST; HORMONE RECEPTOR BLOCKING AGENT; ISOXAZOLE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; CONTROLLED STUDY; DRUG BIOAVAILABILITY; DRUG METABOLISM; DRUG POTENCY; DRUG SCREENING; DRUG SYNTHESIS; NONHUMAN; RAT; STRUCTURE ACTIVITY RELATION;

EID: 20144389487     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2004.11.075     Document Type: Article

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