Design, synthesis, and structure-activity relationships of tetrahydroquinoline-based farnesyltransferase inhibitors

Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 7, 2005, Pages 1895-1899

  Lombardo, Louis J ^a   Camuso, Amy ^a   Clark, John ^a   Fager, Krista ^a   Gullo Brown, Johnni ^a   Hunt, John T ^a   Inigo, Ivan ^a   Kan, David ^a   Koplowitz, Barry ^a   Lee, Francis ^a   McGlinchey, Kelly ^a   Qian, Ligang ^a   Ricca, Carolyn ^a   Rovnyak, George ^a   Traeger, Sarah ^a   Tokarski, John ^a   Williams, David K ^a   Wu, Laurence I ^a   Zhao, Yufen ^a   Manne, Veeraswamy ^a   Bhide, Rajeev S ^a   more..

^a BRISTOL MYERS SQUIBB   (United States)

Author keywords

BMS 316810; Farnesyltransferase inhibitor

Indexed keywords

BMS 316810; PROTEIN FARNESYLTRANSFERASE INHIBITOR; QUINOLINE DERIVATIVE; TETRAHYDROQUINOLINE; UNCLASSIFIED DRUG;

ALLOGRAFT; ANIMAL CELL; ANIMAL MODEL; ANTINEOPLASTIC ACTIVITY; ARTICLE; BIOASSAY; BIOCHEMISTRY; CONTROLLED STUDY; DRUG DESIGN; DRUG SYNTHESIS; MOUSE; MUTANT; NONHUMAN; STRUCTURE ACTIVITY RELATION; TUMOR;

MUS MUSCULUS;

EID: 20144379792     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2005.02.004     Document Type: Article

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