Design, synthesis, and evaluation of proline based melanocortin receptor ligands

Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 11, 2005, Pages 2819-2823

  Tian, Xinrong ^a   Field, Timothy ^a   Mazur, Adam W ^a   Ebetino, Frank H ^a   Wos, John A ^a   Crossdoersen, Doreen ^a   Pinney, Beth B ^a   Sheldon, Russell J ^a  

^a PROCTER AND GAMBLE PHARMACEUTICALS   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

HORMONE RECEPTOR BLOCKING AGENT; HORMONE RECEPTOR STIMULATING AGENT; MELANOCORTIN RECEPTOR; PROLINE DERIVATIVE;

ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; DRUG DESIGN; DRUG SCREENING; DRUG SYNTHESIS; EMBRYO; HUMAN; HUMAN CELL; IC 50; RECEPTOR BINDING;

DRUG DESIGN; HUMANS; LIGANDS; PROLINE; RECEPTORS, MELANOCORTIN; STEREOISOMERISM;

EID: 19544388588     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2005.03.120     Document Type: Article

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