Demonstration of a specific site of covalent labeling of the human motilin receptor using a biologically active photolabile motilin analog

Journal of Pharmacology and Experimental Therapeutics

Volumn 313, Issue 3, 2005, Pages 1101-1108

  Matsuura, Bunzo ^a,b   Dong, Maoqing ^a   Coulie, Bernard ^a,c   Pinon, Delia I ^a   Miller, Laurence J ^a,d  

^a MAYO GRADUATE SCHOOL   (United States)

^b EHIME UNIVERSITY SCHOOL OF MEDICINE   (Japan)

^c JANSSEN RESEARCH AND DEVELOPMENT   (Belgium)

^d MAYO CLINIC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

BENZOYLPHENYLALANINE; CYANOGEN BROMIDE; G PROTEIN COUPLED RECEPTOR; IODINE 125; LIGAND; MOTILIN; MOTILIN DERIVATIVE; MOTILIN RECEPTOR; PEPTIDE; PHENYLALANINE; PHENYLALANINE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; CELL STRAIN COS1; CHO CELL; COVALENT BOND; DRUG BINDING SITE; DRUG CONFORMATION; DRUG DESIGN; DRUG RECEPTOR BINDING; MOLECULAR PROBE; NONHUMAN; PRIORITY JOURNAL; PROTEIN DEGRADATION; PROTEIN LOCALIZATION; PROTEIN STRUCTURE; RADIOCHEMISTRY; RADIOIODINATION; RECEPTOR AFFINITY;

AMINO ACID SEQUENCE; ANIMALS; BINDING SITES; CHO CELLS; COS CELLS; CRICETINAE; HUMANS; MOLECULAR SEQUENCE DATA; MOTILIN; PHOTOAFFINITY LABELS; PROTEIN CONFORMATION; RECEPTORS, GASTROINTESTINAL HORMONE; RECEPTORS, NEUROPEPTIDE;

EID: 19444381509     PISSN: 00223565     EISSN: None     Source Type: Journal    
DOI: 10.1124/jpet.104.081562     Document Type: Article

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