Synthesis and pharmacological evaluation of a new class of peroxisome proliferator-activated receptor modulators

Bioorganic and Medicinal Chemistry Letters

Volumn 12, Issue 24, 2002, Pages 3565-3567

  Thor, Markus ^a   Beierlein, Katarina ^a   Dykes, Graeme ^a   Gustavsson, Anna Lena ^a   Heidrich, Jessica ^a   Jendeberg, Lena ^a   Lindqvist, Bengt ^a   Pegurier, Cecile ^b   Roussel, Patrick ^c   Slater, Martin ^b   Svensson, Stefan ^a   Sydow Bäckman, Mona ^a   Thornström, Ulla ^a   Uppenberg, Jonas ^a  

^a BIOVITRUM AB   (Sweden)

^b BioFocus DPI   (United Kingdom)

^c PFIZER INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

AMINOBENZOIC ACID DERIVATIVE; PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR AGONIST; PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR ALPHA; PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR GAMMA; CELL RECEPTOR; TRANSCRIPTION FACTOR;

ARTICLE; BINDING AFFINITY; BINDING ASSAY; BINDING COMPETITION; DRUG BINDING SITE; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; STRUCTURE ACTIVITY RELATION; X RAY CRYSTALLOGRAPHY; BINDING SITE; CELL CULTURE; DRUG EFFECT; DRUG POTENTIATION; GENETIC TRANSFECTION; GENETICS; HUMAN; SYNTHESIS; TRANSACTIVATION;

AMINOBENZOIC ACIDS; BINDING SITES; CRYSTALLOGRAPHY, X-RAY; HUMANS; RECEPTORS, CYTOPLASMIC AND NUCLEAR; STRUCTURE-ACTIVITY RELATIONSHIP; TRANS-ACTIVATION (GENETICS); TRANSCRIPTION FACTORS; TRANSFECTION; TUMOR CELLS, CULTURED;

EID: 18744365476     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(02)00791-6     Document Type: Article

References (9)

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