Sulfamide derivatives as transition state analogue inhibitors for carboxypeptidase A

Bioorganic and Medicinal Chemistry

Volumn 12, Issue 9, 2004, Pages 2349-2356

  Park, Jung Dae ^a   Kim, Dong H ^a  

^a Pohang University of Science and Technology (POSTECH)   (South Korea)

Author keywords

Carboxypeptidase A; Enzyme inhibition; Hydroxysulfamide; Sulfamide; Transition state analogue inhibitor

Indexed keywords

CARBOXYPEPTIDASE A; SULFAMIDE DERIVATIVE;

ARTICLE; COMPETITIVE INHIBITION; DEGRADATION KINETICS; DRUG BINDING SITE; DRUG SCREENING; DRUG SYNTHESIS; ENZYME INHIBITION; PHASE TRANSITION; X RAY CRYSTALLOGRAPHY;

CARBOXYPEPTIDASES A; KINETICS; PROTEASE INHIBITORS; SPECTRUM ANALYSIS; SULFONIC ACIDS;

EID: 1842817739     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2004.02.012     Document Type: Article

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