In vitro dermal disposition of abamectin (avermectin B1) in livestock

Research in Veterinary Science

Volumn 76, Issue 3, 2004, Pages 235-242

  Baynes, Ronald E ^a  

^a NORTH CAROLINA STATE UNIVERSITY   (United States)

Author keywords

Abamectin; Avermectins; Bovine; Caprine; Dermal absorption; Formulation; Ovine; Porcine

Indexed keywords

2 PROPANOL; ABAMECTIN; EPRINEX; EPRINOMECTIN; IVERMECTIN; TOPICAL ANTIINFECTIVE AGENT;

ANALYSIS OF VARIANCE; ANIMAL TISSUE; ARTICLE; BOVIDS; CATTLE; CONTROLLED STUDY; DOMESTIC ANIMAL; DRUG ABSORPTION; DRUG APPROVAL; DRUG FORMULATION; IN VITRO STUDY; LIVESTOCK; NONHUMAN; PARTITION COEFFICIENT; SHEEP; SKIN ABSORPTION; SKIN SURFACE; SPECIES DIFFERENCE; STRATUM CORNEUM; SWINE;

ANIMALIA; BOVINAE; CAPRA; OVIS; SUIDAE;

EID: 1842737746     PISSN: 00345288     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.rvsc.2003.10.006     Document Type: Article

References (28)

1. Alvinerie, M., Sutra, J.F., Galtier, P., Mage, C., 1999a. Pharmacokinetics of eprinomectin in plasma and milk following topical administration to lactating dairy cattle. Research in Veterinary Science 67, 229-232.
2. Alvinerie, M., Lacoste, E., Sutra, JF., Chartier, C., 1999b. Some pharmacokinetic parameters of eprinomectin in goats following pour-on administration. Veterinary Research Communications 23, 449 455.
3. Baynes, R.E., Payne, M.. Martin-Jimenez, T., Abdullah, A.R., Anderson, K.L., Webb, A.I., Craigmill, A., Riviere, J.E., 2000. Extralabel use of ivermectin and moxidectin in food animals. Journal ofthe American Veterinary Medical Association 217, 668-671.
4. Baynes, R.E., Brooks, J.D., Mumtaz, M., Riviere, J.E., 2002. Effect of chemical interactions in pentachlorophenol mixtures on skin and membrane transport. Toxicological Sciences 69, 295-305.
5. Bronaugh, R.L., Stewart, R.F., 1985. Methods for in vitro percutaneous absorption studies IV: The flow-though diffusion cell. Journal of Pharmaceutical Science 74, 64-67.
6. Egerton, J.R., Birnbaum, J., Blair, L.S., Chabala, J.C., Conroy, J., Fisher, M.H., Mrozik, H., Ostlind, D.A., Wilkins, C.A., Campbell, W.C., 1980. 22,23-dihydroavermectin B1, a new broad-spectrum antiparasitic agent. British Veterinary Journal 136, 88-97.
7. Gayrard, V., Alvinerie, M., Toutain, P.L., 1999. Comparison of pharmacokietic profiles of doramectin and ivermectin pour-on formulations in cattle. Veterinary Parasitology 81, 47-55.
8. Jenkinson, D.M., Lloyd, D.H., 1979. The topography of the skin surface of cattle and sheep. British Veterinary Journal 135, 376-379.
9. Kitagawa, S., Li, H., 1999. Effects of removal of stratum corneum, delipidization and addition of enhancers, ethanol and 1-menthol, on skin permeation of benzoic acid and its 4-n-alkyl substituents in excised guinea pig dorsal skin. Chemical Pharmaceutical Bulletin (Tokyo) 47, 44-47.
10. Klink, P.R., Ferguson, T.H., Magruder, J.A., 1998. Formulation of veterinary dosage forms. In: Hardee, G.E., Baggot, J.D. (Eds.), Development and Formulation of Veterinary Dosage Forms. Marcel Dekker, New York, pp. 145-229.
11. Lo, P.-K.A., Fink, D.W., Williams, J.B., Blodinger, J., 1985. Pharmacokinetic studies of ivermectin: Effects of formulation. Veterinary Research Communications 9, 251-268.
12. Magnusson, B.M., Walters, K.A., Roberts, M.S., 2001. Veterinary drug delivery: Potential for skin penetration enhancement. Advanced Drug Delivery Reviews 50, 205-227.
13. Marriner, S.E., McKinnon, L, Bogan, J.A., 1987. The pharmacokinetics of ivermectin after oral and subcutaneous administration to sheep and horses. Journal of Veterinary Pharmacology and Therapeutics 10, 175-179.
14. Monteiro-Riviere, N.A., 1991. Comparative anatomy, physiology, and biochemistry of mammalian skin. In: Hobson, D.W. (Ed.), Fundamentals and Methods of Dermal and Ocular Toxicology. CRC Press, Boca Raton, FL, pp. 3-71.
15. Nicolaides, N., Fu, H.C., Rice, G.R., 1968. The skin surface lipids of man compared to those of eighteen species of animals. Journal of Investigative Dermatology 51, 83-89.
16. Okamoto, H., Muta, K., Hashida, M., Sezaki, H., 1990. Percutaneous penetration of acyclovir through excised hairless mouse and rat skin: Effect of vehicle and percutaneous penetration enhancer. Pharmaceutical Research 7, 64-68.
17. Pitman, I.H., Rostas, S.J., 1981. Topical drug delivery to cattle and sheep. Journal of Pharmaceutical Sciences 70, 1181-1194.
18. Pitman, I.H., Rostas, S.J., Downes, L.M., 1983. Effects of breed, season, temperature, and solvents on the permeability of frozen and reconstituted cattle skin to levamisole. Journal of Pharmaceutical Science 72, 218-221.
19. Ryder, M.L., 1975. A survey of the follicle populations in a range of British breeds of sheep. Journal of Agricultural Science 49, 275-280.
20. Sato, K., Sugibayashi, K., Morimoto, Y., 1988. Effect and mode of action of aliphatic esters on in vitro skin permeation of nicorandil. International Journal of Pharmaceutics 43, 31-42.
21. Sato, K., Sugibayashi, K., Morimoto, Y., 1991. Species differences in percutaneous absorption of nicorandil. Journal of Pharmaceutical Science 80, 104-107.
22. Scott, E.W., Kinabo, L.D., McKellar, Q.A., 1990. Pharmacokinctics of ivermectin after oral or percutaneous administration to adult milking goats. Journal of Veterinary Pharmacology and Therapeutics 13, 432-435.
23. Sznitowska, M., Janicki, S., Williams, A.C., 1998. Intracellular or intercellular localization of the polar pathway of penetration across stratum corneum. Journal of Pharmaceutical Science 87, 1109-1114.
24. Walters, K.A., Roberts, M.S., 1993. Veterinary applications of skin penetration enhancers. In: Walters, K.A., Hadgraft, J. (Eds.), Pharmaceutical Skin Penetration Enhancement. Marcel Dekker, New York, pp. 345-364.
25. Wicks, S.R., Kaye, B., Weatherley, A.J., Lewis, D., Davison, E., Gibson, S.P., Smith, D.G., 1993. Efect of formulation on the pharmacokinetics and efficacy of doramectin. Veterinary Parasitology 49, 17-26.
26. Williams, A.C., Barry, BW., 1991. Terpenes and the lipid-protein-partitioning theory of skin penetration enhancement. Pharmaceutical Research 8, 17-24.
27. 1a in the rhesus monkey. Toxicology and Applied Pharmacology 94, 38-245.
28. Yazdanian, M., Chen, E., 1995. The effects of diethylene glycol monoethyl ether as a vehicle for topical delivery of ivermectin. Veterinary Research Communications 19, 309-319.