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Volumn 128, Issue 1-3, 2002, Pages 129-144

Estradiol, testosterone, dehydroepiandrosterone and androstenedione: Novel derivatives and enantiomers. Interactions with rat liver microsomal cytochrome P450 and antioxidant/radical scavenger activities in vitro

(17) Klinger, W a Lupp, A a Karge, E a Baumbach, H a Eichhorn, F a Feix, A a Fuldner F a Gernhardt, S a Knels, L a Kost, B a Mertens, G a Werner, F a Oettel, M b Romer W b Schwarz, S b Elger, W c Schneider, B c

a FRIEDRICH SCHILLER UNIVERSITY JENA (Germany)

b BAYER PHARMA AG (Germany)

c EnTec GmbH (Germany)

Author keywords

Androstenedione; Chemiluminescence; Cytochromes P450; Dehydroepiandrosterone; Estrogens; Free radicals; Lipid peroxidation; Testosterone

Indexed keywords

17ALPHA ESTRADIOL 3 DIMETHYLAMIDOSULFONIC ACID; 17BETA (8,9 DEHYDRO 14ALPHA,15ALPHA METHYLENE)ESTRADIOL; ANDROGEN; ANDROSTENEDIONE DERIVATIVE; CYTOCHROME P450; ESTRADIOL DERIVATIVE; ESTRIOL; ESTRONE; ETHER DERIVATIVE; ETHINYLESTRADIOL; ETHOXYCOUMARIN; ETHOXYRESORUFIN; ETHYLMORPHINE; HYDROGEN PEROXIDE; LUCIGENIN; LUMINOL; MESTRANOL; PRASTERONE; PRASTERONE SULFATE; PROGESTERONE DERIVATIVE; SCAVENGER; SULFATE; SULFONIC ACID DERIVATIVE; TESTOSTERONE DERIVATIVE; UNCLASSIFIED DRUG; UNSPECIFIC MONOOXYGENASE;

ANIMAL CELL; ANIMAL MODEL; ANIMAL TISSUE; ANTIOXIDANT ACTIVITY; ARTICLE; CHEMICAL REACTION; CHEMOLUMINESCENCE; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG EFFECT; DRUG PROTEIN BINDING; ENZYME ACTIVITY; ENZYME INHIBITION; IN VITRO STUDY; LIPID PEROXIDATION; LIVER MICROSOME; MALE; METHYLATION; NONHUMAN; PRIORITY JOURNAL; RAT;

7-ALKOXYCOUMARIN O-DEALKYLASE; ANDROSTENEDIONE; ANIMALS; CHEMILUMINESCENT MEASUREMENTS; CYTOCHROME P-450 CYP1A1; CYTOCHROME P-450 ENZYME SYSTEM; DEHYDROEPIANDROSTERONE; ESTRADIOL; ETHYLMORPHINE-N-DEMETHYLASE; LIVER; MALE; MICROSOMES, LIVER; RATS; RATS, WISTAR; REACTIVE OXYGEN SPECIES; TESTOSTERONE;

EID: 18244404841 PISSN: 03784274 EISSN: None Source Type: Journal
DOI: 10.1016/S0378-4274(01)00540-9 Document Type: Article

Times cited : (23)

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