Design and synthesis of novel diphenacoum-derived, conformation-restricted vitamin K 2,3-epoxide reductase inhibitors

Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 10, 2005, Pages 2665-2668

  Chen, Ding Uei ^a   Kuo, Pei Yu ^a   Yang, Ding Yah ^a  

^a TUNGHAI UNIVERSITY   (Taiwan)

Author keywords

Conformation restricted; VKOR inhibitor

Indexed keywords

ENZYME INHIBITOR; UNCLASSIFIED DRUG; VITAMIN K 2,3 EPOXIDE REDUCTASE INHIBITOR;

ARTICLE; DRUG CONFORMATION; DRUG DESIGN; DRUG POTENCY; DRUG SYNTHESIS; ENZYME INHIBITION; INHIBITION KINETICS;

EID: 18144423865     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2005.03.005     Document Type: Article

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