Peptide T-araC conjugates: Solid-phase synthesis and biological activity of N4-(acylpeptidyl)-araC

Bioorganic and Medicinal Chemistry

Volumn 8, Issue 3, 2000, Pages 539-547

  Manfredini, Stefano ^a   Marastoni, Mauro ^a   Tomatis, Roberto ^a   Durini, Elisa ^a   Spisani, Susanna ^a   Pani, Alessandra ^b   Marceddu, Tiziana ^b   Musiu, Chiara ^b   Marongiu, Maria Elena ^b   La Colla, Paolo ^b  

^a UNIVERSITY OF FERRARA   (Italy)

^b UNIVERSITY OF CAGLIARI   (Italy)

Author keywords

[No Author keywords available]

Indexed keywords

ANTINEOPLASTIC AGENT; CD4 ANTIGEN; CYTARABINE; CYTARABINE DERIVATIVE; GLYCOSIDE; NUCLEOSIDE; PEPTIDE DERIVATIVE; PEPTIDE T; PRODRUG;

ANTINEOPLASTIC ACTIVITY; ARTICLE; CANCER CELL CULTURE; CARCINOMA CELL; CELL LINE; CELL MEMBRANE; CHEMOTAXIS; CONCENTRATION RESPONSE; CONJUGATE; CONTROLLED STUDY; CULTURE MEDIUM; DRUG ACTIVITY; DRUG SYNTHESIS; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; HUMAN; HUMAN CELL; LEUKEMIA CELL LINE; LYMPHOCYTE PROLIFERATION; LYMPHOMA CELL LINE; MASS SPECTROMETRY; MONOCYTE; PLASMA; PROTON NUCLEAR MAGNETIC RESONANCE; SOLID PHASE SYNTHESIS; T LYMPHOCYTE;

ANTIGENS, CD4; ANTIMETABOLITES, ANTINEOPLASTIC; CELL DIVISION; CHEMOTAXIS; CYTARABINE; DOSE-RESPONSE RELATIONSHIP, DRUG; DRUG CARRIERS; DRUG STABILITY; HUMANS; INHIBITORY CONCENTRATION 50; MONOCYTES; OLIGOPEPTIDES; PEPTIDE HYDROLASES; PEPTIDE T; PRODRUGS; TIME FACTORS; TUMOR CELLS, CULTURED;

EID: 17944395774     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0968-0896(99)00317-X     Document Type: Article

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