Prodrugs of Ara-CMP and Ara-AMP with a S-acyl-2-thioethyl (SATE) biolabile phosphate protecting group: Synthesis and biological evaluation

Nucleosides and Nucleotides

Volumn 18, Issue 4-5, 1999, Pages 971-972

  Bazzanini, R ^a   Manfredini, S ^b   Durini, E ^b   Groschel B ^c   Cinatl, J ^c   Balzarini, J ^d   De Clercq, E ^d   Imbach, J L ^e   Perigaud C ^e   Gosselin, G ^e  

^a CNR   (Italy)

^b UNIVERSITY OF FERRARA   (Italy)

^c GOETHE UNIVERSITY   (Germany)

^d REGA INSTITUTE FOR MEDICAL RESEARCH   (Belgium)

^e CNRS   (France)

Author keywords

[No Author keywords available]

Indexed keywords

ANTINEOPLASTIC AGENT; ANTIVIRUS AGENT; BIS(PIVALOYL 2 THIOETHYL)PHOSPHOTRIESTER DERIVATIVE; CYTARABINE; CYTARABINE DERIVATIVE; PRODRUG; UNCLASSIFIED DRUG; VIDARABINE; VIDARABINE DERIVATIVE;

ACYLATION; ANTINEOPLASTIC ACTIVITY; ANTIVIRAL ACTIVITY; CONFERENCE PAPER; DRUG SYNTHESIS; LIPOPHILICITY; NONHUMAN; TUMOR CELL;

ARA;

EID: 0032991960     PISSN: 07328311     EISSN: None     Source Type: Journal    
DOI: 10.1080/15257779908041616     Document Type: Conference Paper

References (2)

1. Lefebvre, I., Périgaud, C., Pompon, A., Aubertin, A.-M., Girardet, J.-L., Kim, A., Gosselin, G., and Imbach, J.-L. J Med Chem , 1995, 33, 3941-3950.
2. Gröschel B., Cinatl J., Kotchetkov R., Köhl U., Rohrbach E, Kornhuber B, Bazzanini R., Périgaud C., Gosselin G., Imbach J.-L., Doerr H.W., Cinatl J. In: Haematology and Blood Transfusion 39. Acute Leukemias VII, Experimental Approaches and Novel Therapies. W. Hiddemann, T. et al. Eds., Springer-Verlag Berlin Heidelberg 1998, pp. 628-632.